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Found 15 Enz. Inhib. hit(s) with all data for entry = 50035488
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367068(CHEMBL3350524 | CHEMBL609795)
Affinity DataKi:  3.00E+5nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367067(CHEMBL3350514 | CHEMBL612174)
Affinity DataKi:  1.60E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367066(CHEMBL3350509 | CHEMBL610373)
Affinity DataKi:  1.80E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367073(CHEMBL3350528 | CHEMBL609819)
Affinity DataKi:  1.90E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP:AMP phosphotransferase AK3, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367067(CHEMBL3350514 | CHEMBL612174)
Affinity DataKi:  2.10E+6nMAssay Description:Ability to inhibit rat adenylate kinase III, activity expressed as Inhibition constant; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP:AMP phosphotransferase AK3, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367066(CHEMBL3350509 | CHEMBL610373)
Affinity DataKi:  2.20E+6nMAssay Description:Ability to inhibit rat adenylate kinase III, activity expressed as Inhibition constant; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP:AMP phosphotransferase AK3, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367073(CHEMBL3350528 | CHEMBL609819)
Affinity DataKi:  2.40E+6nMAssay Description:Ability to inhibit rat adenylate kinase III, activity expressed as Inhibition constant; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367071(CHEMBL607736)
Affinity DataKi:  4.70E+6nMAssay Description:Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 4, mitochondrial(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50010316(CHEMBL3251364)
Affinity DataKi:  4.80E+6nMAssay Description:Ability to inhibit Escherichia coli adenylate kinase III, activity expressed as Inhibition constant; Non competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP:AMP phosphotransferase AK3, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367075(CHEMBL3350513 | CHEMBL611859)
Affinity DataKi:  5.90E+6nMAssay Description:Ability to inhibit rat adenylate kinase III, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP:AMP phosphotransferase AK3, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010316(CHEMBL3251364)
Affinity DataKi:  6.20E+6nMAssay Description:Ability to inhibit rat adenylate kinase III, activity expressed as Inhibition constant; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367065(CHEMBL608643)
Affinity DataKi:  6.70E+6nMAssay Description:Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367072(CHEMBL3350534 | CHEMBL610134)
Affinity DataKi:  6.80E+6nMAssay Description:Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367069(CHEMBL3350522 | CHEMBL609792)
Affinity DataKi:  7.30E+6nMAssay Description:Ability to inhibit rat adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate kinase 2, mitochondrial(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367070(CHEMBL609238)
Affinity DataKi:  7.30E+6nMAssay Description:Ability to inhibit Escherichia coli adenylate kinase II, activity expressed as Inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed