Compile Data Set for Download or QSAR
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Found 14 Enz. Inhib. hit(s) with all data for entry = 50038262
TargetGlutamate receptor 1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373889(CHEMBL402444)
Affinity DataKi:  150nMAssay Description:Binding affinity at iGluR1o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373890(CHEMBL429594)
Affinity DataKi:  160nMAssay Description:Binding affinity at iGluR3o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetGlutamate receptor 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373890(CHEMBL429594)
Affinity DataKi:  182nMAssay Description:Binding affinity at iGluR4o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373890(CHEMBL429594)
Affinity DataKi:  185nMAssay Description:Binding affinity at iGluR1o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373889(CHEMBL402444)
Affinity DataKi:  234nMAssay Description:Binding affinity at iGluR2o(R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373890(CHEMBL429594)
Affinity DataKi:  273nMAssay Description:Binding affinity at iGluR2o(R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373890(CHEMBL429594)
Affinity DataKi:  323nMAssay Description:Binding affinity at iGluR2 receptor S1S2J domain expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373889(CHEMBL402444)
Affinity DataKi:  531nMAssay Description:Binding affinity at iGluR2 receptor S1S2J domain expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373889(CHEMBL402444)
Affinity DataKi:  1.06E+3nMAssay Description:Binding affinity at iGluR4o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 3(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373889(CHEMBL402444)
Affinity DataKi:  1.07E+3nMAssay Description:Binding affinity at iGluR3o receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373889(CHEMBL402444)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at iGluR5(Q) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373890(CHEMBL429594)
Affinity DataKi:  1.85E+4nMAssay Description:Binding affinity at iGluR5(Q) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373890(CHEMBL429594)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity at iGluR6(V,C,R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50373889(CHEMBL402444)
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity at iGluR6(V,C,R) receptor expressed in sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed