Compile Data Set for Download or QSAR
maximum 50k data
Found 84 Enz. Inhib. hit(s) with all data for entry = 50041329
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409669(CHEMBL155514)
Affinity DataIC50:  0.178nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409669(CHEMBL155514)
Affinity DataIC50:  0.457nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409669(CHEMBL155514)
Affinity DataIC50:  0.501nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409669(CHEMBL155514)
Affinity DataIC50:  0.537nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409660(CHEMBL155513)
Affinity DataIC50:  3.39nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409657(CHEMBL153015)
Affinity DataIC50:  5.25nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409672(CHEMBL153080)
Affinity DataIC50:  5.5nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371971(CHEMBL440542)
Affinity DataIC50:  6.92nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371971(CHEMBL440542)
Affinity DataIC50:  8.32nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409660(CHEMBL155513)
Affinity DataIC50:  10.5nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371971(CHEMBL440542)
Affinity DataIC50:  12.6nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409660(CHEMBL155513)
Affinity DataIC50:  13.2nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409672(CHEMBL153080)
Affinity DataIC50:  17.0nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409672(CHEMBL153080)
Affinity DataIC50:  22.4nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371971(CHEMBL440542)
Affinity DataIC50:  30.9nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409657(CHEMBL153015)
Affinity DataIC50:  32.4nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409660(CHEMBL155513)
Affinity DataIC50:  36.3nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409670(CHEMBL421992)
Affinity DataIC50:  43.6nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371960(CHEMBL155621)
Affinity DataIC50:  46.8nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409670(CHEMBL421992)
Affinity DataIC50:  47.9nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409672(CHEMBL153080)
Affinity DataIC50:  74.1nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409670(CHEMBL421992)
Affinity DataIC50:  83.2nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409658(CHEMBL153177)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409657(CHEMBL153015)
Affinity DataIC50:  115nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409670(CHEMBL421992)
Affinity DataIC50:  120nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371960(CHEMBL155621)
Affinity DataIC50:  148nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409657(CHEMBL153015)
Affinity DataIC50:  162nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371962(CHEMBL155396)
Affinity DataIC50:  170nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50371962(CHEMBL155396)
Affinity DataIC50:  309nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409658(CHEMBL153177)
Affinity DataIC50:  347nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409658(CHEMBL153177)
Affinity DataIC50:  380nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409671(CHEMBL356917)
Affinity DataIC50:  398nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371960(CHEMBL155621)
Affinity DataIC50:  447nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371962(CHEMBL155396)
Affinity DataIC50:  447nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409658(CHEMBL153177)
Affinity DataIC50:  575nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371960(CHEMBL155621)
Affinity DataIC50:  676nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50371962(CHEMBL155396)
Affinity DataIC50:  1.41E+3nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409666(CHEMBL152225)
Affinity DataIC50:  2.04E+3nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409661(CHEMBL152843)
Affinity DataIC50:  4.37E+3nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409662(CHEMBL152698)
Affinity DataIC50:  5.01E+3nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409661(CHEMBL152843)
Affinity DataIC50:  6.76E+3nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409666(CHEMBL152225)
Affinity DataIC50:  9.33E+3nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409662(CHEMBL152698)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409667(CHEMBL152376)
Affinity DataIC50:  1.17E+4nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcylcarnitine hydrolase(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409666(CHEMBL152225)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of carboxylesterase in murine liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409661(CHEMBL152843)
Affinity DataIC50:  2.14E+4nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase(Sus scrofa)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409662(CHEMBL152698)
Affinity DataIC50:  2.45E+4nMAssay Description:In vitro inhibition of porcine carboxylesterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409668(CHEMBL153107)
Affinity DataIC50:  2.82E+4nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCocaine esterase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50409663(CHEMBL150821)
Affinity DataIC50:  2.88E+4nMAssay Description:In vitro inhibition of carboxylesterase in human liver microsomes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Drosophila melanogaster)
University Of California

Curated by ChEMBL
LigandPNGBDBM50409666(CHEMBL152225)
Affinity DataIC50:  3.55E+4nMAssay Description:In vitro inhibition of Trichoplusia Juvenile Hormone Esterase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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