Compile Data Set for Download or QSAR
maximum 50k data
Found 209 Enz. Inhib. hit(s) with all data for entry = 1497
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327284(N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)thio]-pheny...)
Affinity DataIC50:  10nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327241(N-[5-chloro-2-(methylsulfinyl)phenyl]-1-benzofuran...)
Affinity DataIC50:  11nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327214(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-3-(...)
Affinity DataIC50:  14nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327296(N-(2-{[(6-aminopyridin-2-yl)methyl]sulfonyl}-5-chl...)
Affinity DataIC50:  15nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327306(N-{5-chloro-2-[(1H-pyrazol-3-ylmethyl)thio]phenyl}...)
Affinity DataIC50:  16nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327377(N-{5-chloro-2-[(trifluoromethyl)sulfinyl]phenyl}-1...)
Affinity DataIC50:  19nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327385(N-{2-[(3-aminobenzyl)sulfonyl]-5-fluorophenyl}-1-b...)
Affinity DataIC50:  22nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327325(N-{5-chloro-2-[(pyridin-3-ylmethyl)thio]phenyl}-1-...)
Affinity DataIC50:  22nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327351(N-{2-[(3-aminobenzyl)sulfonyl]-5-chlorophenyl}-1-b...)
Affinity DataIC50:  23nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327332(N-(2-{[(5-amino-1H-pyrazol-3-yl)methyl]thio}-5-chl...)
Affinity DataIC50:  25nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327268(4-chloro-N-[5-chloro-2-(methylthio)phenyl]-2-fluor...)
Affinity DataIC50:  25nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327240(N-[5-chloro-2-(methylthio)phenyl]-1-benzofuran-2-s...)
Affinity DataIC50:  26nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327379(N-[2-(benzylsulfinyl)-5-chlorophenyl]-1-benzofuran...)
Affinity DataIC50:  27nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327295(N-(2-{[(6-aminopyridin-2-yl)methyl]sulfinyl}-5-chl...)
Affinity DataIC50:  28nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327339(N-{5-chloro-2-[(pyridin-2-ylmethyl)sulfonyl]-pheny...)
Affinity DataIC50:  29nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327338(N-{5-chloro-2-[(pyridin-2-ylmethyl)sulfinyl]-pheny...)
Affinity DataIC50:  29nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327294(N-(2-{[(6-aminopyridin-2-yl)methyl]thio}-5-chlorop...)
Affinity DataIC50:  32nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327357(N-(2-{[(5-amino-4H-1,2,4-triazol-3-yl)methyl]thio}...)
Affinity DataIC50:  32nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327328(N-{5-chloro-2-[(pyridin-3-ylmethyl)sulfonyl]-pheny...)
Affinity DataIC50:  32nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327380(N-[2-(benzylsulfonyl)-5-chlorophenyl]-1-benzofuran...)
Affinity DataIC50:  34nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327324(N-{5-chloro-2-[(pyridin-2-ylmethyl)thio]phenyl}-1-...)
Affinity DataIC50:  35nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327383(N-{2-[(3-aminobenzyl)sulfinyl]-5-fluorophenyl}-1-b...)
Affinity DataIC50:  38nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327350(N-{2-[(3-aminobenzyl)sulfinyl]-5-chlorophenyl}-1-b...)
Affinity DataIC50:  39nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327394(N-{2-[(3-aminobenzyl)sulfonyl]phenyl}-1-benzofuran...)
Affinity DataIC50:  41nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327320(N-(2-{[(2-amino-1,3-thiazol-4-yl)methyl]thio}-5-ch...)
Affinity DataIC50:  42nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327242(N-[5-chloro-2-(methylsulfonyl)phenyl]-1-benzofuran...)
Affinity DataIC50:  42nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327349(N-{2-[(3-aminobenzyl)thio]-5-chlorophenyl}-1-benzo...)
Affinity DataIC50:  42nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327250(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-3-m...)
Affinity DataIC50:  44nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327232(3,4-dichloro-N-[5-chloro-2-(methylsulfinyl)phenyl]...)
Affinity DataIC50:  44nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327238(4-chloro-N-[5-chloro-2-(ethylsulfinyl)phenyl]-3-(t...)
Affinity DataIC50:  50nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327421(N-[2-(benzylsulfinyl)-5-cyanophenyl]-1-benzofuran-...)
Affinity DataIC50:  50nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327280(4-chloro-N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)su...)
Affinity DataIC50:  51nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327261(N-[5-chloro-2-(methylsulfinyl)phenyl]-3-nitro-4-(t...)
Affinity DataIC50:  54nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327381(N-{2-[(3-aminobenzyl)thio]-5-fluorophenyl}-1-benzo...)
Affinity DataIC50:  55nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327354(N-{5-chloro-2-[(3-hydroxybenzyl)sulfonyl]phenyl}-1...)
Affinity DataIC50:  56nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327422(N-[2-(benzylsulfonyl)-5-cyanophenyl]-1-benzofuran-...)
Affinity DataIC50:  56nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327390(N-{2-[(3-aminobenzyl)sulfinyl]phenyl}-1-benzofuran...)
Affinity DataIC50:  58nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327281(N-{5-chloro-2-[(1H-imidazol-2-ylmethyl)thio]-pheny...)
Affinity DataIC50:  60nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327271(3-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]-2-f...)
Affinity DataIC50:  61nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327248(4-chloro-N-[5-chloro-2-(methylsulfinyl)phenyl]benz...)
Affinity DataIC50:  62nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327215(4-chloro-N-[5-chloro-2-(methylsulfonyl)phenyl]-3-(...)
Affinity DataIC50:  64nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327278(4-chloro-N-{5-chloro-2-[(1H-imidazol-4-ylmethyl)th...)
Affinity DataIC50:  68nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327262(N-[5-chloro-2-(methylthio)phenyl]-5-methylfuran-2-...)
Affinity DataIC50:  70nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327376(N-{5-chloro-2-[(trifluoromethyl)sulfonyl]phenyl}-1...)
Affinity DataIC50:  73nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327399(N-{5-chloro-2-[(2-nitrobenzyl)sulfinyl]phenyl}-1-b...)
Affinity DataIC50:  75nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327289(3-({2-[(1-benzofuran-2-ylsulfonyl)amino]-4-chlorop...)
Affinity DataIC50:  76nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327326(N-{5-chloro-2-[(pyridin-3-ylmethyl)sulfinyl]phenyl...)
Affinity DataIC50:  76nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327236(4-chloro-N-{5-chloro-2-[(3-hydroxycyclopentyl)sulf...)
Affinity DataIC50:  76nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327352(N-{5-chloro-2-[(3-hydroxybenzyl)thio]phenyl}-1-ben...)
Affinity DataIC50:  77nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM327373(N-(5-chloro-2-{[(2-fluoropyridin-3-yl)methyl]-sulf...)
Affinity DataIC50:  79nMAssay Description:HEK-Gqi5 cells stably expressing CCR2 were cultured in (DMEM high glucose, 10% FBS, 1% PSA, 400 μg/ml geneticin and 50 μg/ml hygromycin. Ap...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 209 total ) | Next | Last >>
Jump to: