Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 1799
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340822(US9765040, Compound 14)
Affinity DataIC50:  16nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340823(US9765040, Compound 15)
Affinity DataIC50:  23nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340790(US9765040, Compound 3)
Affinity DataIC50:  24nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340798(US9765040, Compound 9)
Affinity DataIC50:  26nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340791(US9765040, Compound 4)
Affinity DataIC50:  32nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340796(US9765040, Compound 7)
Affinity DataIC50:  32nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340548(US9765040, Compound 1)
Affinity DataIC50:  35nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340642(US9765040, Compound 2)
Affinity DataIC50:  52nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340803(US9765040, Compound 11)
Affinity DataIC50:  64nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340814(US9765040, Compound 13)
Affinity DataIC50:  68nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340797(US9765040, Compound 8)
Affinity DataIC50:  70nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340799(US9765040, Compound 10)
Affinity DataIC50:  135nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340810(US9765040, Compound 12)
Affinity DataIC50:  182nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340792(US9765040, Compound 5)
Affinity DataIC50:  263nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target11-beta-hydroxysteroid dehydrogenase 1(Rattus norvegicus (rat))
Astellas Pharma

US Patent
LigandPNGBDBM340793(US9765040, Compound 6)
Affinity DataIC50:  322nMAssay Description:The procedure for measuring the 11β-HSD1-inhibitory activity is as follows. The enzyme reaction and the measurement were carried out using a 384...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent