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Found 4 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 3204
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Reviva Pharmaceuticals

US Patent
LigandPNGBDBM312156(6-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-2H...)
Affinity DataKi:  0.650nMAssay Description:Serotonin, 5HT1A:Receptor Source: Human recombinant expressed in HEK-293 cellsRadioligand: [3H]-8-OH-DPAT (221 Ci/mmol)Control Compound: 8-OH-DPATInc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Reviva Pharmaceuticals

US Patent
LigandPNGBDBM312188(6-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butoxy)...)
Affinity DataKi:  1.5nMAssay Description:Serotonin, 5HT1A:Receptor Source: Human recombinant expressed in HEK-293 cellsRadioligand: [3H]-8-OH-DPAT (221 Ci/mmol)Control Compound: 8-OH-DPATInc...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Reviva Pharmaceuticals

US Patent
LigandPNGBDBM312156(6-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butoxy)-2H...)
Affinity DataIC50:  0.970nMAssay Description:Serotonin, 5HT1A:Receptor Source: Human recombinant expressed in HEK-293 cellsRadioligand: [3H]-8-OH-DPAT (221 Ci/mmol)Control Compound: 8-OH-DPATInc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Reviva Pharmaceuticals

US Patent
LigandPNGBDBM312188(6-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butoxy)...)
Affinity DataIC50:  2.25nMAssay Description:Serotonin, 5HT1A:Receptor Source: Human recombinant expressed in HEK-293 cellsRadioligand: [3H]-8-OH-DPAT (221 Ci/mmol)Control Compound: 8-OH-DPATInc...More data for this Ligand-Target Pair
In DepthDetails US Patent