Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 7645
TargetAcyl-protein thioesterase 2 [S122A](Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207992(ML349)
Affinity DataIC50:  1.00E+3nM Kd:  160nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207992(ML349)
Affinity DataIC50:  1.10E+3nM Kd:  240nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
TargetAcyl-protein thioesterase 2 [S122A](Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207994(ML349-sulfoxide)
Affinity DataIC50:  7.10E+3nM Kd:  2.60E+3nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207994(ML349-sulfoxide)
Affinity DataIC50:  1.20E+4nM Kd:  5.20E+3nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2 [S122A](Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207995(ML349-thioether)
Affinity DataIC50: >1.00E+5nM Kd: >1.00E+4nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207995(ML349-thioether)
Affinity DataIC50: >1.00E+5nM Kd: >1.00E+4nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207993(ML349-FL)
Affinity DataKd:  1.02E+3nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2 [S122A](Homo sapiens (Human))
University Of Michigan

LigandPNGBDBM207993(ML349-FL)
Affinity DataKd:  770nMT: 2°CAssay Description:Varying amounts of enzyme were diluted in PBS supplemented with 0.5 g/L pluronic F127 and incubated with 500 nM ML349-FL for 30 minutes at room tempe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed