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Found 1 hit of ph data with Target = 'Cytochrome P450 144 (CYP144A1-TRV)'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Cytochrome P450 144 (CYP144A1-TRV)


(Mycobacterium tuberculosis)
BDBM222348
PNG
(CYP144A1 ligand, 3)
Show SMILES Nc1[nH]nc(c1-c1ccc(O)c(c1)-c1cccc(N)c1)-c1ccc(O)cc1
Show InChI InChI=1S/C21H18N4O2/c22-15-3-1-2-13(10-15)17-11-14(6-9-18(17)27)19-20(24-25-21(19)23)12-4-7-16(26)8-5-12/h1-11,26-27H,22H2,(H3,23,24,25)
GoogleScholar
AffyNet 
PC cid
PC sid
PDB
UniChem
Article
PubMed
n/an/an/a 1.40E+5n/an/an/a7.525



University of Cambridge



Assay Description
ITC binding isotherms were recorded on a MicroCal ITC200 instrument (MalvernInstruments). Titrations were conducted at 25 C by injecting aliquots (2...


Biochemistry 56: 1559-1572 (2017)


Article DOI: 10.1021/acs.biochem.6b00954
BindingDB Entry DOI: 10.7270/Q2SJ1JF3
More data for this
Ligand-Target Pair