Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM23120![]() (7-phenyl-1-[5-(pyridin-2-yl)-1,3-oxazol-2-yl]hepta...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 297 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26741![]() (N-phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26740![]() (N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 595 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26741![]() (N-phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 991 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM23120![]() (7-phenyl-1-[5-(pyridin-2-yl)-1,3-oxazol-2-yl]hepta...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 208 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26739![]() (3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 856 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26740![]() (N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 248 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26741![]() (N-phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 687 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM23120![]() (7-phenyl-1-[5-(pyridin-2-yl)-1,3-oxazol-2-yl]hepta...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 252 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26739![]() (3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 572 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26740![]() (N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 51.9 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26741![]() (N-phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 473 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM23120![]() (7-phenyl-1-[5-(pyridin-2-yl)-1,3-oxazol-2-yl]hepta...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26739![]() (3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 109 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26740![]() (N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carbo...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 16.2 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26739![]() (3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 986 | n/a | n/a | n/a | n/a | 7.4 | 30 |
Pfizer | Assay Description FAAH activity was measured by following the production of ammonia generated from the hydrolysis of oleamide by FAAH. GDH catalyzes the condensation o... | Biochemistry 46: 13019-30 (2007) Article DOI: 10.1021/bi701378g BindingDB Entry DOI: 10.7270/Q2VT1QCN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26732![]() (Benzothiazole-based analogue, 1 | N-[4-(4-methoxy-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | 8.0 | 22 |
AstraZeneca Pharmaceuticals | Assay Description the enzyme activity of recombinant human FAAH was measured according to published procedures with minor modifications by either a fluorescent assay u... | Biochemistry 50: 6867-78 (2011) Article DOI: 10.1021/bi200552p BindingDB Entry DOI: 10.7270/Q2RJ4H2K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26750![]() (D, L mixtures | bisarylimidazole derivative, 9 | e...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26742![]() (bisarylimidazole derivative, 1 | methyl 2-[4-(4,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 670 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26752![]() (D, L mixtures | bisarylimidazole derivative, 11 | ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26753![]() (N-methyl-7-(2-methyl-4,5-diphenyl-1H-imidazol-1-yl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26754![]() (N,N-dimethyl-7-(2-methyl-4,5-diphenyl-1H-imidazol-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 970 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26755![]() (3-methyl-1-[6-(2-methyl-4,5-diphenyl-1H-imidazol-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26756![]() (3-[6-(2-methyl-4,5-diphenyl-1H-imidazol-1-yl)hexyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26757![]() (bisarylimidazole derivative, 16 | phenyl N-[6-(2-m...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26758![]() (2-fluorophenyl N-[6-(2-methyl-4,5-diphenyl-1H-imid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26759![]() (2-fluorophenyl N-[7-(2-methyl-4,5-diphenyl-1H-imid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26760![]() (2-fluorophenyl N-[8-(2-methyl-4,5-diphenyl-1H-imid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26761![]() (2-fluorophenyl N-[2-methyl-8-(2-methyl-4,5-dipheny...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26762![]() (2-fluorophenyl N-[6-(2-methyl-4,5-diphenyl-1H-imid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26763![]() (2-fluorophenyl N-ethyl-N-[6-(2-methyl-4,5-diphenyl...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26764![]() (2-fluorophenyl N-[6-(2-methyl-4,5-diphenyl-1H-imid...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26765![]() (bisarylimidazole derivative, 24 | ethyl 7-[4,5-bis...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 64 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26766![]() (2-fluorophenyl N-{6-[4,5-bis(4-fluorophenyl)-2-met...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26767![]() (2,6-difluorophenyl N-{6-[4,5-bis(4-fluorophenyl)-2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26749![]() (bisarylimidazole derivative, 8 | ethyl 8-(2-ethyl-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 31 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26748![]() (CHEMBL237044 | bisarylimidazole derivative, 7 | et...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26747![]() (bisarylimidazole derivative, 6 | ethyl 6-(2-ethyl-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26746![]() (bisarylimidazole derivative, 5 | ethyl 4-[3-(4,5-d...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 91 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26745![]() (bisarylimidazole derivative, 4 | methyl 2-[3-(4,5-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26744![]() (bisarylimidazole derivative, 3 | ethyl 5-[4-(4,5-d...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26743![]() (bisarylimidazole derivative, 2 | ethyl 4-[4-(4,5-d...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 64 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fatty-acid amide hydrolase 1 (FAAH) (Homo sapiens (Human)) | BDBM26751![]() (D, L mixtures | bisarylimidazole derivative, 10 | ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9.90E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
Bristol-Myers Squibb Company | Assay Description FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin... | Bioorg Med Chem Lett 17: 3287-91 (2007) Article DOI: 10.1016/j.bmcl.2007.04.009 BindingDB Entry DOI: 10.7270/Q2R20ZPP | |||||||||||
More data for this Ligand-Target Pair |