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Found 10 of ph data with Target = 'Gag polyprotein'
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM36655(Cyclopropylmethyl cyclic urea)
Affinity DataIC50:  25nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM36656(Cyclobutylmethyl cyclic urea)
Affinity DataIC50:  7.80nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM36657(2-Naphthylmethyl cyclic urea)
Affinity DataIC50:  12nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM36646(DMP850)
Affinity DataIC50:  49nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM577((3S)-oxolan-3-yl N-[(2S,3R)-4-[(4-aminobenzene)(2-...)
Affinity DataIC50:  13nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM36658(n-Pentyl cyclic urea)
Affinity DataIC50:  41nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM36659(n-Hexyl cyclic urea)
Affinity DataIC50:  130nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM517((2S)-1-[(2S,4R)-4-benzyl-2-hydroxy-4-{[(1S,2R)-2-h...)
Affinity DataIC50:  20nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM519((2S)-N-[(2S,3R)-4-[(3S,4aS,8aS)-3-(tert-butylcarba...)
Affinity DataIC50:  13.1nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag polyprotein(Human immunodeficiency virus type 1 group M subtyp...)
Dupont Pharmaceuticals

LigandPNGBDBM50124714((4R,5S,6S,7R)-1-(3-Amino-1H-indazol-5-ylmethyl)-4,...)
Affinity DataIC50:  39.5nMpH: 6.5Assay Description:Enzyme inhibition assay using cyclic ureas to inhibit GAG polyprotein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed