BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 4 hits of ph data with Target = 'Membrane-bound aminopeptidase P (APP2)'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Membrane-bound aminopeptidase P (APP2)


(Homo sapiens (Human))
BDBM197051
PNG
(US9212206, III)
Show SMILES CC(C)C[C@H](S)C(=O)N1C[C@@H](F)C[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CC[C@H](C1)C(O)=O
Show InChI InChI=1S/C21H32FN3O5S/c1-12(2)8-17(31)20(28)25-11-14(22)9-16(25)19(27)24-6-3-4-15(24)18(26)23-7-5-13(10-23)21(29)30/h12-17,31H,3-11H2,1-2H3,(H,29,30)/t13-,14+,15+,16+,17+/m1/s1
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 3.70n/an/an/an/a7.4n/a



TBA

US Patent


Assay Description
Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...


US Patent US9212206 (2015)


BindingDB Entry DOI: 10.7270/Q24T6H5V
More data for this
Ligand-Target Pair
Membrane-bound aminopeptidase P (APP2)


(Homo sapiens (Human))
BDBM197054
PNG
(US9212206, VII)
Show SMILES CC(C)C[C@H](S)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N(C)[C@@H](C)C(O)=O
Show InChI InChI=1S/C20H33N3O5S/c1-12(2)11-16(29)19(26)23-10-6-8-15(23)18(25)22-9-5-7-14(22)17(24)21(4)13(3)20(27)28/h12-16,29H,5-11H2,1-4H3,(H,27,28)/t13-,14-,15-,16-/m0/s1
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 3.90n/an/an/an/a7.4n/a



TBA

US Patent


Assay Description
Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...


US Patent US9212206 (2015)


BindingDB Entry DOI: 10.7270/Q24T6H5V
More data for this
Ligand-Target Pair
Membrane-bound aminopeptidase P (APP2)


(Homo sapiens (Human))
BDBM197053
PNG
(US9212206, VI)
Show SMILES CC(C)C[C@H](S)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@@H]1C(O)=O
Show InChI InChI=1S/C21H33N3O5S/c1-13(2)12-17(30)20(27)23-10-4-7-15(23)18(25)22-9-3-6-14(22)19(26)24-11-5-8-16(24)21(28)29/h13-17,30H,3-12H2,1-2H3,(H,28,29)/t14-,15-,16+,17-/m0/s1
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 9.70n/an/an/an/a7.4n/a



TBA

US Patent


Assay Description
Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...


US Patent US9212206 (2015)


BindingDB Entry DOI: 10.7270/Q24T6H5V
More data for this
Ligand-Target Pair
Membrane-bound aminopeptidase P (APP2)


(Homo sapiens (Human))
BDBM197052
PNG
(US9212206, V)
Show SMILES CC(C)C[C@H](S)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CC[C@@H](C1)C(O)=O
Show InChI InChI=1S/C21H33N3O5S/c1-13(2)11-17(30)20(27)24-9-4-6-16(24)19(26)23-8-3-5-15(23)18(25)22-10-7-14(12-22)21(28)29/h13-17,30H,3-12H2,1-2H3,(H,28,29)/t14-,15-,16-,17-/m0/s1
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 26n/an/an/an/a7.4n/a



TBA

US Patent


Assay Description
Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...


US Patent US9212206 (2015)


BindingDB Entry DOI: 10.7270/Q24T6H5V
More data for this
Ligand-Target Pair