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Compile Data Set for Download or QSAR

Found 107 hits of ph data with Target = 'Metabotropic glutamate receptor 5'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196506
PNG
(US9212165, 3)
Show SMILES Fc1cccc(c1)C#CC12CCC(C1)(CCC2)NC(=O)c1cnccn1
Show InChI InChI=1S/C21H20FN3O/c22-17-4-1-3-16(13-17)5-8-20-6-2-7-21(15-20,10-9-20)25-19(26)18-14-23-11-12-24-18/h1,3-4,11-14H,2,6-7,9-10,15H2,(H,25,26)
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US Patent
3 -48.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196508
PNG
(US9212165, 16)
Show SMILES O=C(N[C@]12CC[C@](C1)(CCC2)C#Cc1ccccn1)c1ccccn1
Show InChI InChI=1S/C21H21N3O/c25-19(18-7-2-4-15-23-18)24-21-10-5-9-20(16-21,12-13-21)11-8-17-6-1-3-14-22-17/h1-4,6-7,14-15H,5,9-10,12-13,16H2,(H,24,25)/t20-,21+/m0/s1
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US Patent
4.5 -47.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196528
PNG
(US9212165, 71)
Show SMILES O=C(NC12CC3CC(C1)CC(C3)(C2)C#Cc1ccccn1)c1cnccn1
Show InChI InChI=1S/C22H22N4O/c27-20(19-14-23-7-8-25-19)26-22-12-16-9-17(13-22)11-21(10-16,15-22)5-4-18-3-1-2-6-24-18/h1-3,6-8,14,16-17H,9-13,15H2,(H,26,27)
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4.70 -47.5n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196520
PNG
(US9212165, 45)
Show SMILES Cc1csc(n1)C(=O)N[C@]12CC[C@](C1)(CCC2)C#Cc1cnccn1
Show InChI InChI=1S/C19H20N4OS/c1-14-12-25-17(22-14)16(24)23-19-5-2-4-18(13-19,7-8-19)6-3-15-11-20-9-10-21-15/h9-12H,2,4-5,7-8,13H2,1H3,(H,23,24)/t18-,19+/m0/s1
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6.20 -46.8n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196510
PNG
(US9212165, 18)
Show SMILES Cc1nccc(n1)C(=O)N[C@]12CC[C@](C1)(CCC2)C#Cc1ccccn1
Show InChI InChI=1S/C21H22N4O/c1-16-22-14-7-18(24-16)19(26)25-21-9-4-8-20(15-21,11-12-21)10-6-17-5-2-3-13-23-17/h2-3,5,7,13-14H,4,8-9,11-12,15H2,1H3,(H,25,26)/t20-,21+/m0/s1
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10 -45.7n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196511
PNG
(US9212165, 20)
Show SMILES Fc1ccc(nc1)C(=O)N[C@]12CC[C@](C1)(CCC2)C#Cc1ccccn1
Show InChI InChI=1S/C21H20FN3O/c22-16-5-6-18(24-14-16)19(26)25-21-9-3-8-20(15-21,11-12-21)10-7-17-4-1-2-13-23-17/h1-2,4-6,13-14H,3,8-9,11-12,15H2,(H,25,26)/t20-,21+/m0/s1
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11 -45.4n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196514
PNG
(US9212165, 28)
Show SMILES Cc1nccc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)C#Cc1ccccn1
Show InChI InChI=1S/C21H22N4O/c1-16-22-14-7-18(24-16)19(26)25-21-9-4-8-20(15-21,11-12-21)10-6-17-5-2-3-13-23-17/h2-3,5,7,13-14H,4,8-9,11-12,15H2,1H3,(H,25,26)/t20-,21+/m1/s1
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17 -44.3n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196513
PNG
(US9212165, 26)
Show SMILES O=C(N[C@@]12CC[C@@](C1)(CCC2)C#Cc1ccccn1)c1ccccn1
Show InChI InChI=1S/C21H21N3O/c25-19(18-7-2-4-15-23-18)24-21-10-5-9-20(16-21,12-13-21)11-8-17-6-1-3-14-22-17/h1-4,6-7,14-15H,5,9-10,12-13,16H2,(H,24,25)/t20-,21+/m1/s1
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22 -43.7n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141501
PNG
(US8921370, 2 | US9656975, 2)
Show SMILES Cc1cccc(n1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C22H24ClN3O2/c1-15-5-2-8-18(24-15)20(28)26-22-10-4-9-21(14-22,11-12-22)25-19(27)16-6-3-7-17(23)13-16/h2-3,5-8,13H,4,9-12,14H2,1H3,(H,25,27)(H,26,28)
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US Patent
27 -43.2n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196519
PNG
(US9212165, 44)
Show SMILES Cn1ccc(n1)C(=O)N[C@]12CC[C@](C1)(CCC2)C#Cc1cnccn1
Show InChI InChI=1S/C19H21N5O/c1-24-12-4-16(23-24)17(25)22-19-6-2-5-18(14-19,8-9-19)7-3-15-13-20-10-11-21-15/h4,10-13H,2,5-6,8-9,14H2,1H3,(H,22,25)/t18-,19+/m0/s1
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34 -42.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141506
PNG
(US8921370, 160 | US9656975, 160)
Show SMILES Cc1cncc(n1)C(=O)N[C@]12CC[C@](C1)(CCC2)NC(=O)c1cccc(F)c1
Show InChI InChI=1S/C21H23FN4O2/c1-14-11-23-12-17(24-14)19(28)26-21-7-3-6-20(13-21,8-9-21)25-18(27)15-4-2-5-16(22)10-15/h2,4-5,10-12H,3,6-9,13H2,1H3,(H,25,27)(H,26,28)/t20-,21+/m0/s1
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35 -42.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196515
PNG
(US9212165, 30)
Show SMILES Fc1ccc(nc1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)C#Cc1ccccn1
Show InChI InChI=1S/C21H20FN3O/c22-16-5-6-18(24-14-16)19(26)25-21-9-3-8-20(15-21,11-12-21)10-7-17-4-1-2-13-23-17/h1-2,4-6,13-14H,3,8-9,11-12,15H2,(H,25,26)/t20-,21+/m1/s1
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35 -42.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196523
PNG
(US9212165, 50)
Show SMILES Cc1csc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)C#Cc1cnccn1
Show InChI InChI=1S/C19H20N4OS/c1-14-12-25-17(22-14)16(24)23-19-5-2-4-18(13-19,7-8-19)6-3-15-11-20-9-10-21-15/h9-12H,2,4-5,7-8,13H2,1H3,(H,23,24)/t18-,19+/m1/s1
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38 -42.4n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141505
PNG
(US8921370, 126 | US9656975, 126)
Show SMILES Cc1cccc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)NC(=O)c1ccccn1
Show InChI InChI=1S/C21H24N4O2/c1-15-6-4-8-17(23-15)19(27)25-21-10-5-9-20(14-21,11-12-21)24-18(26)16-7-2-3-13-22-16/h2-4,6-8,13H,5,9-12,14H2,1H3,(H,24,26)(H,25,27)/t20-,21+/m1/s1
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39 -42.3n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141508
PNG
(US8921370, 171 | US9656975, 171)
Show SMILES Cc1csc(n1)C(=O)NC12CCC(C1)(CCC2)C(=O)Nc1cccc(C)n1
Show InChI InChI=1S/C20H24N4O2S/c1-13-5-3-6-15(21-13)23-18(26)19-7-4-8-20(12-19,10-9-19)24-16(25)17-22-14(2)11-27-17/h3,5-6,11H,4,7-10,12H2,1-2H3,(H,24,25)(H,21,23,26)
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65 -41.0n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141502
PNG
(US8921370, 6 | US9656975, 6)
Show SMILES Cc1cncc(n1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1cccc(F)c1
Show InChI InChI=1S/C21H23FN4O2/c1-14-11-23-12-17(24-14)19(28)26-21-7-3-6-20(13-21,8-9-21)25-18(27)15-4-2-5-16(22)10-15/h2,4-5,10-12H,3,6-9,13H2,1H3,(H,25,27)(H,26,28)
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78 -40.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196507
PNG
(US9212165, 13)
Show SMILES Clc1cccc(c1)C(=O)NC12CCC(C1)(CCC2)C#Cc1cnccn1
Show InChI InChI=1S/C21H20ClN3O/c22-17-4-1-3-16(13-17)19(26)25-21-7-2-6-20(15-21,9-10-21)8-5-18-14-23-11-12-24-18/h1,3-4,11-14H,2,6-7,9-10,15H2,(H,25,26)
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91 -40.2n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196530
PNG
(US9212165, 81)
Show SMILES Cc1csc(n1)C#CC12CC3CC(CC(C3)(C1)NC(=O)c1ccn(C)n1)C2
Show InChI InChI=1S/C21H24N4OS/c1-14-12-27-18(22-14)3-5-20-8-15-7-16(9-20)11-21(10-15,13-20)23-19(26)17-4-6-25(2)24-17/h4,6,12,15-16H,7-11,13H2,1-2H3,(H,23,26)
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120 -39.5n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141504
PNG
(US8921370, 36 | US9656975, 36)
Show SMILES Cc1cccc(c1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1ccncc1
Show InChI InChI=1S/C22H25N3O2/c1-16-4-2-5-18(14-16)20(27)25-22-9-3-8-21(15-22,10-11-22)24-19(26)17-6-12-23-13-7-17/h2,4-7,12-14H,3,8-11,15H2,1H3,(H,24,26)(H,25,27)
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280 -37.4n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141503
PNG
(US8921370, 15 | US9656975, 15)
Show SMILES Cc1ncc(s1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C20H22ClN3O2S/c1-13-22-11-16(27-13)18(26)24-20-7-3-6-19(12-20,8-9-20)23-17(25)14-4-2-5-15(21)10-14/h2,4-5,10-11H,3,6-9,12H2,1H3,(H,23,25)(H,24,26)
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340 -36.9n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141510
PNG
(US8921370, 178 | US9656975, 178)
Show SMILES Cc1cccc(n1)C(=O)NC12CCC(C1)(CCC2)C(=O)Nc1ccnc(C)n1
Show InChI InChI=1S/C21H25N5O2/c1-14-5-3-6-16(23-14)18(27)26-21-9-4-8-20(13-21,10-11-21)19(28)25-17-7-12-22-15(2)24-17/h3,5-7,12H,4,8-11,13H2,1-2H3,(H,26,27)(H,22,24,25,28)
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370 -36.7n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141509
PNG
(US8921370, 176 | US9656975, 176)
Show SMILES Cc1cccc(NC(=O)C23CCC(C2)(CCC3)NC(=O)c2cccc(Cl)c2)n1
Show InChI InChI=1S/C22H24ClN3O2/c1-15-5-2-8-18(24-15)25-20(28)21-9-4-10-22(14-21,12-11-21)26-19(27)16-6-3-7-17(23)13-16/h2-3,5-8,13H,4,9-12,14H2,1H3,(H,26,27)(H,24,25,28)
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500 -36.0n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196522
PNG
(US9212165, 49)
Show SMILES Cn1ccc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)C#Cc1cnccn1
Show InChI InChI=1S/C19H21N5O/c1-24-12-4-16(23-24)17(25)22-19-6-2-5-18(14-19,8-9-19)7-3-15-13-20-10-11-21-15/h4,10-13H,2,5-6,8-9,14H2,1H3,(H,22,25)/t18-,19+/m1/s1
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590 -35.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141507
PNG
(US8921370, 161 | US9656975, 161)
Show SMILES Cc1cncc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)NC(=O)c1cccc(F)c1
Show InChI InChI=1S/C21H23FN4O2/c1-14-11-23-12-17(24-14)19(28)26-21-7-3-6-20(13-21,8-9-21)25-18(27)15-4-2-5-16(22)10-15/h2,4-5,10-12H,3,6-9,13H2,1H3,(H,25,27)(H,26,28)/t20-,21+/m1/s1
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1.20E+3 -33.8n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol. Pharmacol., 2003, 64, 731-740] with slight modifications, including that a r...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196525
PNG
(US9212165, 56)
Show SMILES Cc1cncc(n1)C#CC12CC3CC(CC(C3)(C1)NC(=O)c1cccc(F)c1)C2
Show InChI InChI=1S/C24H24FN3O/c1-16-13-26-14-21(27-16)5-6-23-9-17-7-18(10-23)12-24(11-17,15-23)28-22(29)19-3-2-4-20(25)8-19/h2-4,8,13-14,17-18H,7,9-12,15H2,1H3,(H,28,29)
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1.30E+3 -33.6n/an/an/an/an/a7.425



H. Lundbeck A/S

US Patent


Assay Description
Binding assays were performed as described in [J. A. O'Brien et al. Mol Pharmacol., 2003, 64, 731-740] with slight modifications, including that ...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141501
PNG
(US8921370, 2 | US9656975, 2)
Show SMILES Cc1cccc(n1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C22H24ClN3O2/c1-15-5-2-8-18(24-15)20(28)26-22-10-4-9-21(14-22,11-12-22)25-19(27)16-6-3-7-17(23)13-16/h2-3,5-8,13H,4,9-12,14H2,1H3,(H,25,27)(H,26,28)
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n/an/a 3.70n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141502
PNG
(US8921370, 6 | US9656975, 6)
Show SMILES Cc1cncc(n1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1cccc(F)c1
Show InChI InChI=1S/C21H23FN4O2/c1-14-11-23-12-17(24-14)19(28)26-21-7-3-6-20(13-21,8-9-21)25-18(27)15-4-2-5-16(22)10-15/h2,4-5,10-12H,3,6-9,13H2,1H3,(H,25,27)(H,26,28)
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n/an/a 9n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141503
PNG
(US8921370, 15 | US9656975, 15)
Show SMILES Cc1ncc(s1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1cccc(Cl)c1
Show InChI InChI=1S/C20H22ClN3O2S/c1-13-22-11-16(27-13)18(26)24-20-7-3-6-19(12-20,8-9-20)23-17(25)14-4-2-5-15(21)10-14/h2,4-5,10-11H,3,6-9,12H2,1H3,(H,23,25)(H,24,26)
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n/an/a 26n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141504
PNG
(US8921370, 36 | US9656975, 36)
Show SMILES Cc1cccc(c1)C(=O)NC12CCC(C1)(CCC2)NC(=O)c1ccncc1
Show InChI InChI=1S/C22H25N3O2/c1-16-4-2-5-18(14-16)20(27)25-22-9-3-8-21(15-22,10-11-22)24-19(26)17-6-12-23-13-7-17/h2,4-7,12-14H,3,8-11,15H2,1H3,(H,24,26)(H,25,27)
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n/an/a 35n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141505
PNG
(US8921370, 126 | US9656975, 126)
Show SMILES Cc1cccc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)NC(=O)c1ccccn1
Show InChI InChI=1S/C21H24N4O2/c1-15-6-4-8-17(23-15)19(27)25-21-10-5-9-20(14-21,11-12-21)24-18(26)16-7-2-3-13-22-16/h2-4,6-8,13H,5,9-12,14H2,1H3,(H,24,26)(H,25,27)/t20-,21+/m1/s1
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n/an/a 0.320n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141506
PNG
(US8921370, 160 | US9656975, 160)
Show SMILES Cc1cncc(n1)C(=O)N[C@]12CC[C@](C1)(CCC2)NC(=O)c1cccc(F)c1
Show InChI InChI=1S/C21H23FN4O2/c1-14-11-23-12-17(24-14)19(28)26-21-7-3-6-20(13-21,8-9-21)25-18(27)15-4-2-5-16(22)10-15/h2,4-5,10-12H,3,6-9,13H2,1H3,(H,25,27)(H,26,28)/t20-,21+/m0/s1
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n/an/a 3.90n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141507
PNG
(US8921370, 161 | US9656975, 161)
Show SMILES Cc1cncc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)NC(=O)c1cccc(F)c1
Show InChI InChI=1S/C21H23FN4O2/c1-14-11-23-12-17(24-14)19(28)26-21-7-3-6-20(13-21,8-9-21)25-18(27)15-4-2-5-16(22)10-15/h2,4-5,10-12H,3,6-9,13H2,1H3,(H,25,27)(H,26,28)/t20-,21+/m1/s1
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n/an/a 134n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141508
PNG
(US8921370, 171 | US9656975, 171)
Show SMILES Cc1csc(n1)C(=O)NC12CCC(C1)(CCC2)C(=O)Nc1cccc(C)n1
Show InChI InChI=1S/C20H24N4O2S/c1-13-5-3-6-15(21-13)23-18(26)19-7-4-8-20(12-19,10-9-19)24-16(25)17-22-14(2)11-27-17/h3,5-6,11H,4,7-10,12H2,1-2H3,(H,24,25)(H,21,23,26)
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n/an/a 4.70n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141509
PNG
(US8921370, 176 | US9656975, 176)
Show SMILES Cc1cccc(NC(=O)C23CCC(C2)(CCC3)NC(=O)c2cccc(Cl)c2)n1
Show InChI InChI=1S/C22H24ClN3O2/c1-15-5-2-8-18(24-15)25-20(28)21-9-4-10-22(14-21,12-11-21)26-19(27)16-6-3-7-17(23)13-16/h2-3,5-8,13H,4,9-12,14H2,1H3,(H,26,27)(H,24,25,28)
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n/an/a 33n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM141510
PNG
(US8921370, 178 | US9656975, 178)
Show SMILES Cc1cccc(n1)C(=O)NC12CCC(C1)(CCC2)C(=O)Nc1ccnc(C)n1
Show InChI InChI=1S/C21H25N5O2/c1-14-5-3-6-16(23-14)18(27)26-21-9-4-8-20(13-21,10-11-21)19(28)25-17-7-12-22-15(2)24-17/h3,5-7,12H,4,8-11,13H2,1-2H3,(H,26,27)(H,22,24,25,28)
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n/an/a 38n/an/an/an/a7.437



H. Lundbeck A/S

US Patent


Assay Description
The cDNA for rat metabotropic glutamate receptor 5 (rmGluR5) and the cDNA for human metabotropic glutamate receptor 5 (rmGluR5) were generous gifts f...


US Patent US8921370 (2014)


BindingDB Entry DOI: 10.7270/Q2CR5S3C
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196506
PNG
(US9212165, 3)
Show SMILES Fc1cccc(c1)C#CC12CCC(C1)(CCC2)NC(=O)c1cnccn1
Show InChI InChI=1S/C21H20FN3O/c22-17-4-1-3-16(13-17)5-8-20-6-2-7-21(15-20,10-9-20)25-19(26)18-14-23-11-12-24-18/h1,3-4,11-14H,2,6-7,9-10,15H2,(H,25,26)
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n/an/a 1.20n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196508
PNG
(US9212165, 16)
Show SMILES O=C(N[C@]12CC[C@](C1)(CCC2)C#Cc1ccccn1)c1ccccn1
Show InChI InChI=1S/C21H21N3O/c25-19(18-7-2-4-15-23-18)24-21-10-5-9-20(16-21,12-13-21)11-8-17-6-1-3-14-22-17/h1-4,6-7,14-15H,5,9-10,12-13,16H2,(H,24,25)/t20-,21+/m0/s1
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n/an/a 1.60n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196509
PNG
(US9212165, 17)
Show SMILES O=C(N[C@]12CC[C@](C1)(CCC2)C#Cc1ccccn1)c1cnccn1
Show InChI InChI=1S/C20H20N4O/c25-18(17-14-21-12-13-23-17)24-20-7-3-6-19(15-20,9-10-20)8-5-16-4-1-2-11-22-16/h1-2,4,11-14H,3,6-7,9-10,15H2,(H,24,25)/t19-,20+/m0/s1
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n/an/a 6.60n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196512
PNG
(US9212165, 23)
Show SMILES Fc1cccnc1C(=O)N[C@]12CC[C@](C1)(CCC2)C#Cc1ccccn1
Show InChI InChI=1S/C21H20FN3O/c22-17-6-3-14-24-18(17)19(26)25-21-9-4-8-20(15-21,11-12-21)10-7-16-5-1-2-13-23-16/h1-3,5-6,13-14H,4,8-9,11-12,15H2,(H,25,26)/t20-,21+/m0/s1
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n/an/a 11n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196513
PNG
(US9212165, 26)
Show SMILES O=C(N[C@@]12CC[C@@](C1)(CCC2)C#Cc1ccccn1)c1ccccn1
Show InChI InChI=1S/C21H21N3O/c25-19(18-7-2-4-15-23-18)24-21-10-5-9-20(16-21,12-13-21)11-8-17-6-1-3-14-22-17/h1-4,6-7,14-15H,5,9-10,12-13,16H2,(H,24,25)/t20-,21+/m1/s1
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n/an/a 5.90n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196516
PNG
(US9212165, 32)
Show SMILES Cn1ccc(n1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)C#Cc1ccccn1
Show InChI InChI=1S/C20H22N4O/c1-24-14-7-17(23-24)18(25)22-20-9-4-8-19(15-20,11-12-20)10-6-16-5-2-3-13-21-16/h2-3,5,7,13-14H,4,8-9,11-12,15H2,1H3,(H,22,25)/t19-,20+/m1/s1
PDB
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KEGG

UniProtKB/SwissProt

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UniChem
US Patent
n/an/a 17n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196517
PNG
(US9212165, 37)
Show SMILES Cc1cccc(n1)C#C[C@]12CC[C@](C1)(CCC2)NC(=O)c1ccccn1
Show InChI InChI=1S/C22H23N3O/c1-17-6-4-7-18(24-17)9-12-21-10-5-11-22(16-21,14-13-21)25-20(26)19-8-2-3-15-23-19/h2-4,6-8,15H,5,10-11,13-14,16H2,1H3,(H,25,26)/t21-,22+/m1/s1
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KEGG

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n/an/a 5.30n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196518
PNG
(US9212165, 41)
Show SMILES Fc1cccnc1C#C[C@]12CC[C@](C1)(CCC2)NC(=O)c1cnccn1
Show InChI InChI=1S/C20H19FN4O/c21-15-3-1-10-23-16(15)4-7-19-5-2-6-20(14-19,9-8-19)25-18(26)17-13-22-11-12-24-17/h1,3,10-13H,2,5-6,8-9,14H2,(H,25,26)/t19-,20+/m1/s1
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KEGG

UniProtKB/SwissProt

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n/an/a 9.30n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196521
PNG
(US9212165, 46)
Show SMILES Cc1nc(cs1)C(=O)N[C@]12CC[C@](C1)(CCC2)C#Cc1cnccn1
Show InChI InChI=1S/C19H20N4OS/c1-14-22-16(12-25-14)17(24)23-19-5-2-4-18(13-19,7-8-19)6-3-15-11-20-9-10-21-15/h9-12H,2,4-5,7-8,13H2,1H3,(H,23,24)/t18-,19+/m0/s1
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KEGG

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n/an/a 12n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196524
PNG
(US9212165, 51)
Show SMILES Cc1nc(cs1)C(=O)N[C@@]12CC[C@@](C1)(CCC2)C#Cc1cnccn1
Show InChI InChI=1S/C19H20N4OS/c1-14-22-16(12-25-14)17(24)23-19-5-2-4-18(13-19,7-8-19)6-3-15-11-20-9-10-21-15/h9-12H,2,4-5,7-8,13H2,1H3,(H,23,24)/t18-,19+/m1/s1
PDB
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KEGG

UniProtKB/SwissProt

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n/an/a 83n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196526
PNG
(US9212165, 58)
Show SMILES Cc1cncc(n1)C(=O)NC12CC3CC(C1)CC(C3)(C2)C#Cc1cccnc1
Show InChI InChI=1S/C23H24N4O/c1-16-12-25-14-20(26-16)21(28)27-23-10-18-7-19(11-23)9-22(8-18,15-23)5-4-17-3-2-6-24-13-17/h2-3,6,12-14,18-19H,7-11,15H2,1H3,(H,27,28)
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n/an/a 3.80n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196527
PNG
(US9212165, 62)
Show SMILES Fc1cncc(c1)C(=O)NC12CC3CC(C1)CC(C3)(C2)C#Cc1cnccn1
Show InChI InChI=1S/C22H21FN4O/c23-18-6-17(11-25-12-18)20(28)27-22-9-15-5-16(10-22)8-21(7-15,14-22)2-1-19-13-24-3-4-26-19/h3-4,6,11-13,15-16H,5,7-10,14H2,(H,27,28)
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KEGG

UniProtKB/SwissProt

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n/an/a 30n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM196529
PNG
(US9212165, 80)
Show SMILES Cc1ccc(cn1)C#CC12CC3CC(CC(C3)(C1)NC(=O)c1cnccn1)C2
Show InChI InChI=1S/C23H24N4O/c1-16-2-3-17(13-26-16)4-5-22-9-18-8-19(10-22)12-23(11-18,15-22)27-21(28)20-14-24-6-7-25-20/h2-3,6-7,13-14,18-19H,8-12,15H2,1H3,(H,27,28)
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KEGG

UniProtKB/SwissProt

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n/an/a 700n/an/an/an/a7.4n/a



H. Lundbeck A/S

US Patent


Assay Description
The rmGluR5 or hmGluR5 was stably expressed in a HEK 293 cell line and gown in Dulbecco's Modified Eagle Medium (DMEM) (Invitrogen, Carlsbad, Cal...


US Patent US9212165 (2015)


BindingDB Entry DOI: 10.7270/Q2Z89B69
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM206000
PNG
(US9255103, 1)
Show SMILES Fc1ccc(cc1)C(=O)N1CCn2nc(COc3ccccc3)cc2C1
Show InChI InChI=1S/C20H18FN3O2/c21-16-8-6-15(7-9-16)20(25)23-10-11-24-18(13-23)12-17(22-24)14-26-19-4-2-1-3-5-19/h1-9,12H,10-11,13-14H2
PDB
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KEGG

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n/an/an/an/a 161n/an/a7.4n/a



Vanderbilt University

US Patent


Assay Description
HEK cells transfected with the human mGluR5a receptor (H10H cell line) were plated at 15,000 cells/well in clear-bottomed poly-D-lysine-coated assay ...


US Patent US9255103 (2016)


BindingDB Entry DOI: 10.7270/Q29S1PV6
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 5


(Homo sapiens (Human))
BDBM206001
PNG
(US9255103, 2)
Show SMILES Fc1ccccc1C(=O)N1CCn2nc(COc3ccccc3)cc2C1
Show InChI InChI=1S/C20H18FN3O2/c21-19-9-5-4-8-18(19)20(25)23-10-11-24-16(13-23)12-15(22-24)14-26-17-6-2-1-3-7-17/h1-9,12H,10-11,13-14H2
PDB
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KEGG

UniProtKB/SwissProt

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n/an/an/an/a 201n/an/a7.4n/a



Vanderbilt University

US Patent


Assay Description
HEK cells transfected with the human mGluR5a receptor (H10H cell line) were plated at 15,000 cells/well in clear-bottomed poly-D-lysine-coated assay ...


US Patent US9255103 (2016)


BindingDB Entry DOI: 10.7270/Q29S1PV6
More data for this
Ligand-Target Pair
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