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Found 14 of ph data with Target = 'Methionine aminopeptidase 1'
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17587(bestatin-type inhibitor, 2 | ethyl (2S)-2-[(2S,3R)...)
Affinity DataIC50:  6.90E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17593(CHEMBL170733 | N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2...)
Affinity DataIC50:  8.10E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17592(CHEMBL169958 | N'-[(2S,3R)-3-amino-5-(ethylsulfany...)
Affinity DataIC50:  2.00E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17591((2S,3R)-3-amino-2-hydroxy-N-[(1S)-1-(naphthalen-1-...)
Affinity DataIC50:  1.20E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17590((2S,3S)-3-amino-2-hydroxy-4-[(2-methylpropyl)sulfa...)
Affinity DataIC50:  2.20E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17586(bestatin-type inhibitor, 1 | ethyl (2S)-2-[(2S,3R)...)
Affinity DataIC50:  6.30E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17594(A-357300 | CHEMBL352764 | N'-[(2S,3R)-3-amino-2-hy...)
Affinity DataIC50:  5.70E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17588(bestatin-type inhibitor, 3 | ethyl (2S)-2-[(2S,3S)...)
Affinity DataIC50:  6.60E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17589((2S,3R)-3-amino-5-(ethylsulfanyl)-2-hydroxy-N-[(1S...)
Affinity DataIC50:  370nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17852(3-octanamido-N-(1,3-thiazol-2-yl)pyridine-2-carbox...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17851(3-[(E)-(2-methylpropylidene)amino]-N-(1,3-thiazol-...)
Affinity DataIC50:  6.40E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17850(3-(3-phenylpropanamido)-N-(1,3-thiazol-2-yl)pyridi...)
Affinity DataIC50:  3.50E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17849(3-(2,2-dimethylpropanamido)-N-(1,3-thiazol-2-yl)py...)
Affinity DataIC50:  2.90E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM17847(CHEMBL327579 | pyridine-2-carboxylic acid inhibito...)
Affinity DataIC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair