Affinity DataKi: 0.790nM ΔG°: -51.4kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nM ΔG°: -47.5kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
Affinity DataKi: 4.70nM ΔG°: -47.1kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nM ΔG°: -47.0kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
Affinity DataKi: 5.30nM ΔG°: -46.8kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
Affinity DataKi: 6.60nM ΔG°: -46.2kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
Affinity DataKi: 16nM ΔG°: -44.0kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
Affinity DataKi: 26nM ΔG°: -42.9kJ/molepH: 7.4 T: 2°CAssay Description:A radioligand-binding assay was developed using scintillation proximity assay (SPA) technology. The wheat germ agglutinin SPA beads (Amersham) (0.2 m...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 920nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 110nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 200nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 220nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 48nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 150nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 250nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 299nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 59nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 8nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 19nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 15nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 91nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 25nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 23nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 7.60nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 9.5nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 110nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 64nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 26nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 120nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 950nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 88nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 340nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 66nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Regents Of The University Of Minnesota
US Patent
Regents Of The University Of Minnesota
US Patent
Affinity DataIC50: 43nMpH: 7.43 T: 2°CAssay Description:The entire lactate uptake studies for the inhibition of MCT1 were carried out on RBE4 (Rat Brain Endothelial 4) cells. The expression of MCT1 on thes...More data for this Ligand-Target Pair
Affinity DataKi: 0.0900nM ΔG°: -56.8kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.100nM ΔG°: -56.5kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.280nM ΔG°: -54.0kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.290nM ΔG°: -53.9kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.310nM ΔG°: -53.7kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nM ΔG°: -53.6kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.350nM ΔG°: -53.4kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.420nM ΔG°: -53.0kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.430nM ΔG°: -52.9kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.520nM ΔG°: -52.5kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.680nM ΔG°: -51.8kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 0.810nM ΔG°: -51.4kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nM ΔG°: -50.6kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nM ΔG°: -50.4kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nM ΔG°: -49.6kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nM ΔG°: -48.9kJ/molepH: 7.8 T: 2°CAssay Description:Jurkat cell membranes were incubated with [3H]-labeled ligand in the absence or presence of increasing concentrations of test compound. The reagents ...More data for this Ligand-Target Pair