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Compile Data Set for Download or QSAR

Found 1075 hits of ph data with Target = 'Serine/threonine-protein kinase PIM'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108350
PNG
(US8604217, 385)
Show SMILES CN1CCN(CC1)C1CCN(CC1)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C17H21Br4N5/c1-24-6-8-25(9-7-24)10-2-4-26(5-3-10)17-22-15-13(20)11(18)12(19)14(21)16(15)23-17/h10H,2-9H2,1H3,(H,22,23)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 45.3n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108351
PNG
(US8604217, 386)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(nc2c1Br)N1CCC(CC1)C1CCNCC1
Show InChI InChI=1S/C17H20Br4N4/c18-11-12(19)14(21)16-15(13(11)20)23-17(24-16)25-7-3-10(4-8-25)9-1-5-22-6-2-9/h9-10,22H,1-8H2,(H,23,24)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 58.0n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108353
PNG
(US8604217, 392)
Show SMILES NC(=N)N1CCN(CC1)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C12H12Br4N6/c13-5-6(14)8(16)10-9(7(5)15)19-12(20-10)22-3-1-21(2-4-22)11(17)18/h1-4H2,(H3,17,18)(H,19,20)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 6.72n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108355
PNG
(US8604217, 416)
Show SMILES CCn1c(nc2c(Br)c(Br)c(Br)c(Br)c12)N1CCNCC1
Show InChI InChI=1S/C13H14Br4N4/c1-2-21-12-10(17)8(15)7(14)9(16)11(12)19-13(21)20-5-3-18-4-6-20/h18H,2-6H2,1H3
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 6.55n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108356
PNG
(US8604217, 417)
Show SMILES CCCn1c(nc2c(Br)c(Br)c(Br)c(Br)c12)N1CCNCC1
Show InChI InChI=1S/C14H16Br4N4/c1-2-5-22-13-11(18)9(16)8(15)10(17)12(13)20-14(22)21-6-3-19-4-7-21/h19H,2-7H2,1H3
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 9.36n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108416
PNG
(US8604217, 441)
Show SMILES CCn1c(nc2c(Br)c(Br)c(Br)c(Br)c12)N1CCN(CCN2CCNCC2)CC1
Show InChI InChI=1S/C19H26Br4N6/c1-2-29-18-16(23)14(21)13(20)15(22)17(18)25-19(29)28-11-9-27(10-12-28)8-7-26-5-3-24-4-6-26/h24H,2-12H2,1H3
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 65n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108357
PNG
(US8604217, 450)
Show SMILES CCn1c(nc2c(Br)c(Br)c(Br)c(Br)c12)N1CCN(CCCN2CCOCC2)CC1
Show InChI InChI=1S/C20H27Br4N5O/c1-2-29-19-17(24)15(22)14(21)16(23)18(19)25-20(29)28-8-6-26(7-9-28)4-3-5-27-10-12-30-13-11-27/h2-13H2,1H3
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 125n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108358
PNG
(US8604217, 11)
Show SMILES NCCCNc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C10H10Br4N4/c11-4-5(12)7(14)9-8(6(4)13)17-10(18-9)16-3-1-2-15/h1-3,15H2,(H2,16,17,18)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 5.89n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108359
PNG
(US8604217, 13)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCN3CCCCC3)nc2c1Br
Show InChI InChI=1S/C14H16Br4N4/c15-8-9(16)11(18)13-12(10(8)17)20-14(21-13)19-4-7-22-5-2-1-3-6-22/h1-7H2,(H2,19,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 319n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108360
PNG
(US8604217, 14)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCN3CCCC3)nc2c1Br
Show InChI InChI=1S/C13H14Br4N4/c14-7-8(15)10(17)12-11(9(7)16)19-13(20-12)18-3-6-21-4-1-2-5-21/h1-6H2,(H2,18,19,20)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 57.8n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108361
PNG
(US8604217, 16)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCN3CCOCC3)nc2c1Br
Show InChI InChI=1S/C13H14Br4N4O/c14-7-8(15)10(17)12-11(9(7)16)19-13(20-12)18-1-2-21-3-5-22-6-4-21/h1-6H2,(H2,18,19,20)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 107n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108362
PNG
(US8604217, 28)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(Nc3ccncc3)nc2c1Br
Show InChI InChI=1S/C12H6Br4N4/c13-6-7(14)9(16)11-10(8(6)15)19-12(20-11)18-5-1-3-17-4-2-5/h1-4H,(H2,17,18,19,20)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 37.0n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108363
PNG
(US8604217, 58)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCCN3CCCC3)nc2c1Br
Show InChI InChI=1S/C14H16Br4N4/c15-8-9(16)11(18)13-12(10(8)17)20-14(21-13)19-4-3-7-22-5-1-2-6-22/h1-7H2,(H2,19,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 25.7n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108364
PNG
(US8604217, 59)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCCN3CCCCC3)nc2c1Br
Show InChI InChI=1S/C15H18Br4N4/c16-9-10(17)12(19)14-13(11(9)18)21-15(22-14)20-5-4-8-23-6-2-1-3-7-23/h1-8H2,(H2,20,21,22)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 50.8n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108365
PNG
(US8604217, 61)
Show SMILES NCCCCNc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C11H12Br4N4/c12-5-6(13)8(15)10-9(7(5)14)18-11(19-10)17-4-2-1-3-16/h1-4,16H2,(H2,17,18,19)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 8.85n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108366
PNG
(US8604217, 65)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCCn3ccnc3)nc2c1Br
Show InChI InChI=1S/C13H11Br4N5/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-2-1-4-22-5-3-18-6-22/h3,5-6H,1-2,4H2,(H2,19,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
n/an/a 22.7n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108367
PNG
(US8604217, 67)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCC3CCNCC3)nc2c1Br
Show InChI InChI=1S/C13H14Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-5-6-1-3-18-4-2-6/h6,18H,1-5H2,(H2,19,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 65.2n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108368
PNG
(US8604217, 79)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(Nc3ccccc3)nc2c1Br
Show InChI InChI=1S/C13H7Br4N3/c14-7-8(15)10(17)12-11(9(7)16)19-13(20-12)18-6-4-2-1-3-5-6/h1-5H,(H2,18,19,20)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 68.2n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108369
PNG
(US8604217, 82)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCc3ccccc3)nc2c1Br
Show InChI InChI=1S/C14H9Br4N3/c15-8-9(16)11(18)13-12(10(8)17)20-14(21-13)19-6-7-4-2-1-3-5-7/h1-5H,6H2,(H2,19,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 200n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108370
PNG
(US8604217, 85)
Show SMILES CN(C)CCCN(Cc1ccccc1)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C19H20Br4N4/c1-26(2)9-6-10-27(11-12-7-4-3-5-8-12)19-24-17-15(22)13(20)14(21)16(23)18(17)25-19/h3-5,7-8H,6,9-11H2,1-2H3,(H,24,25)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 65.3n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108371
PNG
(US8604217, 86)
Show SMILES Nc1ccc(Nc2nc3c(Br)c(Br)c(Br)c(Br)c3[nH]2)cc1
Show InChI InChI=1S/C13H8Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-3-1-5(18)2-4-6/h1-4H,18H2,(H2,19,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 66.0n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108372
PNG
(US8604217, 87)
Show SMILES NC1CCC(CC1)Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H14Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-3-1-5(18)2-4-6/h5-6H,1-4,18H2,(H2,19,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

n/an/a 15.1n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108373
PNG
(US8604217, 90)
Show SMILES NCC(O)CNc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C10H10Br4N4O/c11-4-5(12)7(14)9-8(6(4)13)17-10(18-9)16-2-3(19)1-15/h3,19H,1-2,15H2,(H2,16,17,18)
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n/an/a 13.1n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108374
PNG
(US8604217, 95)
Show SMILES CN(C)CCN(Cc1ccccc1)c1nc2c(Br)c(Br)c(Br)c(Br)c2n1Cc1ccccc1
Show InChI InChI=1S/C25H24Br4N4/c1-31(2)13-14-32(15-17-9-5-3-6-10-17)25-30-23-21(28)19(26)20(27)22(29)24(23)33(25)16-18-11-7-4-8-12-18/h3-12H,13-16H2,1-2H3
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n/an/a 75.7n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108376
PNG
(US8604217, 117)
Show SMILES CN(Cc1ccccc1)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C15H11Br4N3/c1-22(7-8-5-3-2-4-6-8)15-20-13-11(18)9(16)10(17)12(19)14(13)21-15/h2-6H,7H2,1H3,(H,20,21)
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Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108377
PNG
(US8604217, 128)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCc3ccccn3)nc2c1Br
Show InChI InChI=1S/C14H10Br4N4/c15-8-9(16)11(18)13-12(10(8)17)21-14(22-13)20-6-4-7-3-1-2-5-19-7/h1-3,5H,4,6H2,(H2,20,21,22)
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n/an/a 71.3n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108378
PNG
(US8604217, 158)
Show SMILES CN(C)CCN(Cc1ccccc1)c1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C18H18Br4N4/c1-25(2)8-9-26(10-11-6-4-3-5-7-11)18-23-16-14(21)12(19)13(20)15(22)17(16)24-18/h3-7H,8-10H2,1-2H3,(H,23,24)
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Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108379
PNG
(US8604217, 166)
Show SMILES CN(C)CCN1CCC(CNc2nc3c(Br)c(Br)c(Br)c(Br)c3[nH]2)C1
Show InChI InChI=1S/C16H21Br4N5/c1-24(2)5-6-25-4-3-9(8-25)7-21-16-22-14-12(19)10(17)11(18)13(20)15(14)23-16/h9H,3-8H2,1-2H3,(H2,21,22,23)
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Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108380
PNG
(US8604217, 192)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCCN3CCOCC3)nc2c1Br
Show InChI InChI=1S/C14H16Br4N4O/c15-8-9(16)11(18)13-12(10(8)17)20-14(21-13)19-2-1-3-22-4-6-23-7-5-22/h1-7H2,(H2,19,20,21)
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Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108383
PNG
(US8604217, 247)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NCCN3CCN(CC3)c3ncccn3)nc2c1Br
Show InChI InChI=1S/C17H17Br4N7/c18-10-11(19)13(21)15-14(12(10)20)25-16(26-15)22-4-5-27-6-8-28(9-7-27)17-23-2-1-3-24-17/h1-3H,4-9H2,(H2,22,25,26)
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Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108384
PNG
(US8604217, 248)
Show SMILES Cc1c(Nc2nc3c(Br)c(Br)c(Br)c(Br)c3[nH]2)cccc1-c1nncn1C
Show InChI InChI=1S/C17H12Br4N6/c1-7-8(16-26-22-6-27(16)2)4-3-5-9(7)23-17-24-14-12(20)10(18)11(19)13(21)15(14)25-17/h3-6H,1-2H3,(H2,23,24,25)
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n/an/a 48.9n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108386
PNG
(US8604217, 261)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(NC3CCCCCCC3)nc2c1Br
Show InChI InChI=1S/C15H17Br4N3/c16-9-10(17)12(19)14-13(11(9)18)21-15(22-14)20-8-6-4-2-1-3-5-7-8/h8H,1-7H2,(H2,20,21,22)
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n/an/a 138n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108387
PNG
(US8604217, 265a)
Show SMILES CCN1CCCC1CNc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C14H16Br4N4/c1-2-22-5-3-4-7(22)6-19-14-20-12-10(17)8(15)9(16)11(18)13(12)21-14/h7H,2-6H2,1H3,(H2,19,20,21)
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n/an/a 67.4n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108389
PNG
(US8604217, 272)
Show SMILES CN(C)CC(CNc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1)C(O)c1ccccc1
Show InChI InChI=1S/C19H20Br4N4O/c1-27(2)9-11(18(28)10-6-4-3-5-7-10)8-24-19-25-16-14(22)12(20)13(21)15(23)17(16)26-19/h3-7,11,18,28H,8-9H2,1-2H3,(H2,24,25,26)
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n/an/a 43.3n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108390
PNG
(US8604217, 296)
Show SMILES Fc1ccc(CNc2nc3c(Br)c(Br)c(Br)c(Br)c3[nH]2)cc1F
Show InChI InChI=1S/C14H7Br4F2N3/c15-8-9(16)11(18)13-12(10(8)17)22-14(23-13)21-4-5-1-2-6(19)7(20)3-5/h1-3H,4H2,(H2,21,22,23)
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n/an/a 170n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108391
PNG
(US8604217, 303)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(Nc3c[nH]c(=O)[nH]c3=O)nc2c1Br
Show InChI InChI=1S/C11H5Br4N5O2/c12-3-4(13)6(15)8-7(5(3)14)18-10(19-8)17-2-1-16-11(22)20-9(2)21/h1H,(H2,17,18,19)(H2,16,20,21,22)
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n/an/a 128n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108392
PNG
(US8604217, 304cis)
Show SMILES NC1CCCCC1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H14Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-4-2-1-3-5(6)18/h5-6H,1-4,18H2,(H2,19,20,21)
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n/an/a 6.90n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108393
PNG
(US8604217, 304RR)
Show SMILES N[C@@H]1CCCC[C@H]1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H14Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-4-2-1-3-5(6)18/h5-6H,1-4,18H2,(H2,19,20,21)/t5-,6-/m1/s1
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n/an/a 5.26n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108394
PNG
(US8604217, 304SS)
Show SMILES N[C@H]1CCCC[C@@H]1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H14Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-4-2-1-3-5(6)18/h5-6H,1-4,18H2,(H2,19,20,21)/t5-,6-/m0/s1
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n/an/a 11.6n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108396
PNG
(US8604217, 307)
Show SMILES COc1ccc(Nc2nc3c(Br)c(Br)c(Br)c(Br)c3[nH]2)cc1OC
Show InChI InChI=1S/C15H11Br4N3O2/c1-23-7-4-3-6(5-8(7)24-2)20-15-21-13-11(18)9(16)10(17)12(19)14(13)22-15/h3-5H,1-2H3,(H2,20,21,22)
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n/an/a 287n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108397
PNG
(US8604217, 309)
Show SMILES OC1CCC(CC1)Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H13Br4N3O/c14-7-8(15)10(17)12-11(9(7)16)19-13(20-12)18-5-1-3-6(21)4-2-5/h5-6,21H,1-4H2,(H2,18,19,20)
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n/an/a 15.9n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108398
PNG
(US8604217, 317)
Show SMILES Nc1cc(Br)c(Br)cc1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H6Br6N4/c14-3-1-5(20)6(2-4(3)15)21-13-22-11-9(18)7(16)8(17)10(19)12(11)23-13/h1-2H,20H2,(H2,21,22,23)
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n/an/a 598n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108399
PNG
(US8604217, 329)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(Nc3ccccn3)nc2c1Br
Show InChI InChI=1S/C12H6Br4N4/c13-6-7(14)9(16)11-10(8(6)15)19-12(20-11)18-5-3-1-2-4-17-5/h1-4H,(H2,17,18,19,20)
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n/an/a 47.0n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108400
PNG
(US8604217, 331)
Show SMILES NC1CC=CCC1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H12Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-4-2-1-3-5(6)18/h1-2,5-6H,3-4,18H2,(H2,19,20,21)
PDB
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UniProtKB/SwissProt

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PC sid
UniChem
n/an/a 14.8n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108401
PNG
(US8604217, 332)
Show SMILES Nc1ccccc1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H8Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-4-2-1-3-5(6)18/h1-4H,18H2,(H2,19,20,21)
PDB
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n/an/a 16.2n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108402
PNG
(US8604217, 333)
Show SMILES Nc1cc(F)c(F)cc1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H6Br4F2N4/c14-7-8(15)10(17)12-11(9(7)16)22-13(23-12)21-6-2-4(19)3(18)1-5(6)20/h1-2H,20H2,(H2,21,22,23)
PDB
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KEGG

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n/an/a 48.5n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108403
PNG
(US8604217, 334)
Show SMILES OC1CCCCC1Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H13Br4N3O/c14-7-8(15)10(17)12-11(9(7)16)19-13(20-12)18-5-3-1-2-4-6(5)21/h5-6,21H,1-4H2,(H2,18,19,20)
PDB
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KEGG

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n/an/a 14.1n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108404
PNG
(US8604217, 336)
Show SMILES NC1CCCC(C1)Nc1nc2c(Br)c(Br)c(Br)c(Br)c2[nH]1
Show InChI InChI=1S/C13H14Br4N4/c14-7-8(15)10(17)12-11(9(7)16)20-13(21-12)19-6-3-1-2-5(18)4-6/h5-6H,1-4,18H2,(H2,19,20,21)
PDB
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KEGG

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n/an/a 18.8n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108405
PNG
(US8604217, 337)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(N[C@H]3COC[C@@H]3N3CCCC3)nc2c1Br
Show InChI InChI=1S/C15H16Br4N4O/c16-9-10(17)12(19)14-13(11(9)18)21-15(22-14)20-7-5-24-6-8(7)23-3-1-2-4-23/h7-8H,1-6H2,(H2,20,21,22)/t7-,8-/m0/s1
PDB
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KEGG

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n/an/a 25.6n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
Serine/threonine-protein kinase PIM


(Homo sapiens (Human))
BDBM108406
PNG
(US8604217, 338)
Show SMILES Brc1c(Br)c(Br)c2[nH]c(N[C@H]3COC[C@@H]3N3CCCCC3)nc2c1Br
Show InChI InChI=1S/C16H18Br4N4O/c17-10-11(18)13(20)15-14(12(10)19)22-16(23-15)21-8-6-25-7-9(8)24-4-2-1-3-5-24/h8-9H,1-7H2,(H2,21,22,23)/t8-,9-/m0/s1
PDB
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KEGG

UniProtKB/SwissProt

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Similars

n/an/a 21.7n/an/an/an/a7.0n/a



Selvita S.A.

US Patent


Assay Description
Kinase assay was performed using luminescent Kinase-Glo (Promega) system. The Kinase-Glo Luminescent Kinase Assay Platform provides a homogeneous, hi...


US Patent US8604217 (2013)


BindingDB Entry DOI: 10.7270/Q2RJ4H31
More data for this
Ligand-Target Pair
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