Affinity DataEC50: 0.0398nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY1 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 5.60nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >30nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <32nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 135nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 135nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 144nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 222nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: >500nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: >500nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: >500nMAssay Description:Agonist activity at human NPYY1 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 790nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y1R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair