Affinity DataEC50: 7nMAssay Description:Partial agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assay relative to SR142948aMore data for this Ligand-Target Pair
Affinity DataEC50: >10nMAssay Description:Agonist activity at rat neurotensin receptor type 2 expressed in CHOK1 cells assessed as increase in calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Partial agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at rat neurotensin receptor type 2 expressed in CHOK1 cells assessed as increase in calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at rat neurotensin receptor type 2 expressed in CHOK1 cells assessed as increase in calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at rat NTS2 receptor expressed in CHO-K1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 28nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 54nMAssay Description:Binding affinity to human NTR2 by gamma countingMore data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Agonist activity at rat NTS2 overexpressed in CHO-k1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 68nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 94nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:Agonist activity at rat neurotensin receptor type 2 expressed in CHOK1 cells assessed as increase in calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 108nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 145nMAssay Description:Agonist activity at rat neurotensin receptor type 2 expressed in CHOK1 cells assessed as increase in calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 159nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 166nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 216nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 217nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 229nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 258nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 271nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 345nMAssay Description:Partial agonist activity at rat NTS2 receptor expressed in CHOK1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 382nMAssay Description:Agonist activity at rat NTS2 stably expressed in CHOK1 cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 480nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 590nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 690nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: 840nMAssay Description:Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activit...More data for this Ligand-Target Pair
Affinity DataEC50: 951nMAssay Description:Agonist activity at rat NTS2 overexpressed in CHO-k1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.41E+3nMAssay Description:Partial agonist activity at rat NTS2 receptor expressed in CHOK1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: >8.00E+4nMAssay Description:Agonist activity at NTR2 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assayMore data for this Ligand-Target Pair
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Medical University Of South Carolina Campus
Curated by ChEMBL
Medical University Of South Carolina Campus
Curated by ChEMBL
Affinity DataEC50: >8.00E+4nMAssay Description:Agonist activity at NTR2 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assayMore data for this Ligand-Target Pair