Compile Data Set for Download or QSAR
maximum 50k data
Found 43 of ec50 data for polymerid = 50000958
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50459972(CHEMBL4226003)
Affinity DataEC50:  4nMAssay Description:Agonist activity at B6D2F1 mouse insulin receptor assessed as increase in glucose incorporation into lipid phase after 2 hrs in presence of D-[3-3H]g...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377967(CHEMBL1627107)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253185(2-Chloro-5-{[(7-{[(7-{[(4-chloro-3-sulfophenyl)ami...)
Affinity DataEC50:  6.00E+3nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253181(2-Hydroxy-5-{[(7-{[(7-sulfo(2-naphthyl))amino]carb...)
Affinity DataEC50:  9.00E+3nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253179(5-{[(7-{[(7-{[(3-Carboxy-4-chlorophenyl)amino]sulf...)
Affinity DataEC50:  1.60E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253178(5-{[(7-{[(7-{[(3-Carboxy-4-chlorophenyl)amino]sulf...)
Affinity DataEC50:  1.80E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377968(CHEMBL1627106)
Affinity DataEC50:  2.20E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253166(3-{7-[({7-[(3-carboxyphenyl)sulfamoyl]naphthalen-2...)
Affinity DataEC50:  2.40E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253159(3-{[(4-Hydroxy-7-{[(5-hydroxy-7-{[(3-sulfophenyl)a...)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253182(5-{7-[({7-[(3-carboxy-4-nitrophenyl)sulfamoyl]naph...)
Affinity DataEC50:  4.00E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253177(2-{7-[({7-[(2-carboxyphenyl)sulfamoyl]naphthalen-2...)
Affinity DataEC50:  4.10E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253165(3-{7-[({7-[(3-carboxyphenyl)sulfamoyl]-5-hydroxyna...)
Affinity DataEC50:  4.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253180(5-{[(7-{[(7-{[(3-Carboxy-4-hydroxyphenyl)amino]sul...)
Affinity DataEC50:  4.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253168(1,3-bis(7-{[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]sul...)
Affinity DataEC50:  5.40E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253189(5-[({7-[3-(7-{[(3-Carboxy-4-chlorophenyl)amino]sul...)
Affinity DataEC50:  5.60E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253167(1,3-bis(5-hydroxy-7-{[3-(1H-1,2,3,4-tetrazol-1-yl)...)
Affinity DataEC50:  7.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377965(CHEMBL436679)
Affinity DataEC50:  9.00E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253192(CHEMBL505538 | disodium 3-{N-methyl7-[({7-[methyl(...)
Affinity DataEC50:  9.10E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253175(2-{7-[({7-[(2-carboxyphenyl)sulfamoyl]-5-hydroxyna...)
Affinity DataEC50:  9.30E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253173(CHEMBL499172 | disodium 4-{7-[({7-[(4-sulfonatophe...)
Affinity DataEC50:  9.40E+4nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253174(4-{7-[({7-[(4-carboxyphenyl)sulfamoyl]-5-hydroxyna...)
Affinity DataEC50:  1.03E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253184(3-{7-[({7-[(3-carboxy-2-chlorophenyl)sulfamoyl]-5-...)
Affinity DataEC50:  1.21E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253183(3-{7-[({7-[(3-carboxy-2-hydroxyphenyl)sulfamoyl]na...)
Affinity DataEC50:  1.50E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253195(5-({[7-({[(7-{[(3-Carboxy-4-chlorophenyl)amino]sul...)
Affinity DataEC50:  1.62E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253196(5-{[(7-{2-Amino-1-aza-2-[(7-{[(3-carboxy-4-chlorop...)
Affinity DataEC50:  1.79E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253176(4-{7-[({7-[(4-carboxyphenyl)sulfamoyl]naphthalen-2...)
Affinity DataEC50:  1.83E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253164(1,3-bis(5-hydroxy-7-{[3-(trifluoromethyl)phenyl]su...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253163(1,3-bis({7-[(3-cyanophenyl)sulfamoyl]naphthalen-2-...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253188(CHEMBL453256 | sodium 7-[({7-[(3-carboxy-4-hydroxy...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253191(CHEMBL442662 | disodium 3-{7-[({7-[(3-sulfonatophe...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253169(1,3-bis(5-hydroxy-7-{[3-(hydroxymethyl)phenyl]sulf...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253190(3-({7-[(N-{7-[N-(3-Carboxyphenyl)carbamoyl]-2-naph...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253171(1,3-bis({7-[(3-sulfamoylphenyl)sulfamoyl]naphthale...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253193(5-({[7-(N-{2-[N-(7-{[(3-Carboxy-4-chlorophenyl)ami...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253170(1,3-bis({7-[(3-hydroxyphenyl)sulfamoyl]naphthalen-...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253172(2-[3-(7-{[(7-{[3-(carboxymethyl)phenyl]sulfamoyl}-...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253194(5-({[7-({2-[(7-{[(3-Carboxy-4-chlorophenyl)amino]s...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253199(5-{[(7-{[N-(7-{[(3-Carboxy-4-chlorophenyl)amino]su...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253162(1,3-bis({7-[(3-nitrophenyl)sulfamoyl]naphthalen-2-...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253161(7,7'-carbonylbis(azanediyl)bis(N-phenylnaphthalene...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253198(5-[7-(1-{7-[(3-carboxy-4-chlorophenyl)sulfamoyl]na...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50253197(5-[7-(1-{7-[(3-carboxy-4-chlorophenyl)sulfamoyl]na...)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Mus musculus)
University Of Melbourne

Curated by ChEMBL
LigandPNGBDBM50377966(CHEMBL1627108)
Affinity DataEC50: >2.00E+5nMAssay Description:Activation of insulin receptor tyrosine kinase in mouse 3T3-L1 cells assessed as increase in 2-deoxy-D-[14C]glucose transport in presence of insulinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed