Compile Data Set for Download or QSAR
maximum 50k data
Found 29 of ec50 data for polymerid = 50001025,50006406
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437266(CHEMBL2407271)
Affinity DataEC50:  22nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437262(CHEMBL2407259)
Affinity DataEC50:  165nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM80521(3-Hydroxy-2-naphtho-p-phenetidide | 3-hydroxy-N-p-...)
Affinity DataEC50:  212nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437267(CHEMBL2407270)
Affinity DataEC50:  221nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437264(CHEMBL2407257)
Affinity DataEC50:  243nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50015214(6-chloro-2-methoxy-9-acridinyl(4-diethylamino-1-me...)
Affinity DataEC50:  300nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437258(CHEMBL2407263)
Affinity DataEC50:  334nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437261(CHEMBL2407260)
Affinity DataEC50:  348nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437265(CHEMBL2407256)
Affinity DataEC50:  365nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437259(CHEMBL2407262)
Affinity DataEC50:  411nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437270(CHEMBL2407267)
Affinity DataEC50:  424nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM75523(3-Methoxy-naphthalene-2-carboxylic acid (4-ethoxy-...)
Affinity DataEC50:  512nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437268(CHEMBL2407269)
Affinity DataEC50:  520nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437260(CHEMBL2407261)
Affinity DataEC50:  677nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437263(CHEMBL2407258)
Affinity DataEC50:  743nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437269(CHEMBL2407268)
Affinity DataEC50:  861nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)
Affinity DataEC50:  2.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437273(CHEMBL1332508)
Affinity DataEC50:  2.20E+3nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataEC50:  4.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50131719(CHEMBL39560 | acepromazine)
Affinity DataEC50:  5.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM67545(N,N-dimethyl-3-(10-phenothiazinyl)-1-propanamine;h...)
Affinity DataEC50:  5.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437271(CHEMBL2407266)
Affinity DataEC50:  6.66E+3nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50017696((2-dimethylamino-2-methyl)ethyl-N-dibenzoparathiaz...)
Affinity DataEC50:  8.00E+3nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataEC50: >1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437274(CHEMBL2407264)
Affinity DataEC50: >1.00E+4nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50003659(5H-dibenzo[b,f]azepine-5-carboxamide | CARBAMAZEPI...)
Affinity DataEC50: >1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Ovis aries)
University Of California

Curated by ChEMBL
LigandPNGBDBM50437272(CHEMBL2407265)
Affinity DataEC50: >1.00E+4nMAssay Description:Antiprion activity against sheep prion infected in mouse ScN2a-cl3 cells assessed as reduction in PrPSc level after 5 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50131720(9,10-diazaanthracene | CHEMBL119870 | acridizine |...)
Affinity DataEC50: >1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMajor prion protein(Homo sapiens (Human))
Institut F£R Molekularbiologie Und Biophysik

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataEC50:  1.00E+4nMAssay Description:Half maximal inhibition of Prion protein PrPsc formation was assayed in ScN2a cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed