Compile Data Set for Download or QSAR
maximum 50k data
Found 151 of ec50 data for polymerid = 50001093,50002355,50004898
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085044((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-...)
Affinity DataEC50:  0.350nMAssay Description:Compound was tested functionally in vitro for inducing 50% of the maximum alkaline phosphatase activity (Transactivation) against murine Peroxisome p...Checked by AuthorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085044((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-...)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085046(2-((S)-1-carboxy-2-{4-[2-(5-methyl-2-phenyl-oxazol...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50306508(4'-((2,3-dimethyl-5-(1-phenylpropylcarbamoyl)-1H-i...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse PPARgamma expressed in african green monkey CV1 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50448033(CHEMBL3115237)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse PPARgamma expressed in CV-1 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50615950(CHEMBL5288454)
Affinity DataEC50:  4.10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50418564(CHEMBL423026)
Affinity DataEC50:  4.70nMAssay Description:Compound was tested functionally in vitro for inducing 50% of the maximum alkaline phosphatase activity (Transactivation) against murine Peroxisome p...Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50448032(CHEMBL3115238)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse PPARgamma expressed in CV-1 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085040(CHEMBL278994 | L-796449 | {3-Chloro-4-[3-(3-phenyl...)
Affinity DataEC50:  10nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50246525(2-(4-((5-(4-tert-butylphenyl)-1-methyl-1H-pyrazole...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at mouse PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50081222(2-(4-{2-[1-Cycloheptyl-3-(2,4-difluoro-phenyl)-ure...)
Affinity DataEC50:  12nMAssay Description:Compound was tested for its agonist activity against murine Peroxisome proliferator activated receptor gamma-Gal4 chimeric receptor in transfected CV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50049244(5-{4-[2-(Benzooxazol-2-yl-methyl-amino)-ethoxy]-be...)
Affinity DataEC50:  13nMAssay Description:In vitro transcriptional activation of Peroxisome proliferator activated receptor gamma (PPAR) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataEC50:  13nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at mouse PPARgamma expressed in african green monkey CV1 cells by Gal4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-Benzoyl-phenylamino)-3-{4-[2-(methyl-pyri...)
Affinity DataEC50:  13nMAssay Description:Compound was tested functionally in vitro for inducing 50% of the maximum alkaline phosphatase activity (Transactivation) against murine Peroxisome p...Checked by AuthorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50245782(2-(4-((5-(4-isopropylphenyl)-1-methyl-1H-pyrazole-...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at mouse PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  28nMAssay Description:Agonist activity against PPAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50200403((S)-2-(5-(3-((2-(4-isopropylphenyl)-5-methylpyrimi...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARgamma expressed in HEK293 cells co-expressing with Gal4 reporter vector after 24 hrs by dual-luciferase reporter assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50200402(2-((S)-5-(3-(5-(5-acetyl-4-methylthiazol-2-yl)pyri...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50245843(2-(4-((5-(4-tert-butylphenyl)-1-ethyl-1H-pyrazole-...)
Affinity DataEC50:  36nMAssay Description:Agonist activity at mouse PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50615962(CHEMBL5272996)
Affinity DataEC50:  40nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  60nMAssay Description:In vitro transcriptional activation of Peroxisome proliferator activated receptor gamma (PPAR) expressed in CV-1 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50246088(2-methyl-2-[2-methyl-4-({[1-methyl-5-(2'-methyl-bi...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at mouse PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  76nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50064455(4-{4-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-be...)
Affinity DataEC50:  89nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50085043(3-{4-[2-(Benzooxazol-2-yl-methyl-amino)-ethoxy]-ph...)
Affinity DataEC50:  100nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50448025(CHEMBL3115243)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse PPARgamma expressed in CV-1 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50083625(CHEMBL320553 | {3-[2-(4-Methoxy-phenyl)-ethyl]-2-p...)
Affinity DataEC50:  140nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50049239(5-[1-{4-[2-(Benzooxazol-2-yl-methyl-amino)-ethoxy]...)
Affinity DataEC50:  140nMAssay Description:In vitro transcriptional activation of Peroxisome proliferator activated receptor gamma (PPAR) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50075315(5-(2,4-Dioxo-thiazolidin-5-ylmethyl)-2-methoxy-N-(...)
Affinity DataEC50:  140nMAssay Description:Agonist activity for murine PPAR gamma receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50200411((S)-2-(5-(3-((2-(4-ethylphenyl)-5-methylpyrimidin-...)
Affinity DataEC50:  145nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50245945(2-(4-((1-allyl-5-(4-tert-butylphenyl)-1H-pyrazole-...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at mouse PPARgamma receptor by cell based transient transfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50148090((R)-7-{3-[2-Chloro-4-(4-fluoro-phenoxy)-phenoxy]-p...)
Affinity DataEC50:  150nMAssay Description:In vitro transcriptional activation by PPAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50615951(CHEMBL5285352)
Affinity DataEC50:  150nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50200410((S)-2-(5-(3-((2-(4-tert-butylphenyl)-5-methylpyrim...)
Affinity DataEC50:  156nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50322695(4,6-Bis(benzylthio)-2-(methylthio)pyrimidine-5-car...)
Affinity DataEC50:  158nMAssay Description:Partial agonist activity at mouse PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as luciferase activity by transactivation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Rattus norvegicus)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50322695(4,6-Bis(benzylthio)-2-(methylthio)pyrimidine-5-car...)
Affinity DataEC50:  158nMAssay Description:Partial agonist activity at rat PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as luciferase activity by transactivation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50200416((S)-2-(5-(3-((2-(4-ethoxyphenyl)-5-methylpyrimidin...)
Affinity DataEC50:  161nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50049242(5-[1-{4-[2-(Methyl-pyridin-2-yl-amino)-ethoxy]-phe...)
Affinity DataEC50:  190nMAssay Description:In vitro transcriptional activation of Peroxisome proliferator activated receptor gamma (PPAR) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50615948(CHEMBL5281528)
Affinity DataEC50:  200nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50448031(CHEMBL3115239)
Affinity DataEC50:  200nMAssay Description:Agonist activity at mouse PPARgamma expressed in CV-1 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50244350(CHEMBL4091374)
Affinity DataEC50:  202nMAssay Description:Transactivation of mouse GAL4-fused PPARgamma LBD expressed in African green monkey COS7 cells co-expressing 5Gal4 pGL3 TK Luc after overnight incuba...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50615964(CHEMBL5277165)
Affinity DataEC50:  230nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50200415((S)-2-(5-(3-((2-(4-acetylphenyl)-5-methylpyrimidin...)
Affinity DataEC50:  237nMAssay Description:Agonist activity at PPARgamma in mouse 3T3-L1 cells by IRBAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50615954(CHEMBL5290870)
Affinity DataEC50:  240nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50615955(CHEMBL5283926)
Affinity DataEC50:  240nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50448026(CHEMBL3115244)
Affinity DataEC50:  250nMAssay Description:Partial agonist activity at mouse PPARgamma expressed in CV-1 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM50448027(CHEMBL3115245)
Affinity DataEC50:  250nMAssay Description:Agonist activity at mouse PPARgamma expressed in CV-1 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Glaxo Wellcome Research And Development

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  250nMAssay Description:Effective concentration against murine peroxisome proliferator activated receptor gamma in Gal4 transactivation assayMore data for this Ligand-Target Pair
Displayed 1 to 50 (of 151 total ) | Next | Last >>
Jump to: