Affinity DataEC50: 0.210nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.280nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.360nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.370nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.390nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.440nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 77nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 115nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at LPA3 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 127nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 164nMAssay Description:Activity at LPA3 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 194nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 204nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 263nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 265nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:Agonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as increase in intracellular calcium level measured every 3...More data for this Ligand-Target Pair
Affinity DataEC50: 546nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 580nMAssay Description:Agonist activity at human LPA3 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 639nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 692nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 830nMAssay Description:Agonist activity at human LPA3 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 3 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
Affinity DataEC50: >7.03E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Rattus norvegicus)
University Of Tennessee Health Science Center
Curated by ChEMBL
University Of Tennessee Health Science Center
Curated by ChEMBL
Affinity DataEC50: 7.59E+3nMAssay Description:Activity at LPA3 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity as increased intracellular calcium level by human LPA3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.18E+4nMAssay Description:Agonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair