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Compile Data Set for Download or QSAR

Found 466 hits of ec50 data for polymerid = 50006630   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313179
PNG
(US10166249, Example 697 | US10166249, Example 698)
Show SMILES COc1ccccc1CCC1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C25H34NO5P/c1-30-24-5-3-2-4-19(24)8-6-18-7-9-21-15-22(11-10-20(21)14-18)23-12-13-25(26,16-23)17-31-32(27,28)29/h2-5,10-11,15,18,23H,6-9,12-14,16-17,26H2,1H3,(H2,27,28,29)/t18?,23-,25+/m0/s1
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n/an/an/an/a 0.600n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313184
PNG
(US10166249, Example 696)
Show SMILES CCOCCCC1CCc2cc(ccc2C1)[C@H]1CC[C@@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C21H34NO5P/c1-2-26-11-3-4-16-5-6-18-13-19(8-7-17(18)12-16)20-9-10-21(22,14-20)15-27-28(23,24)25/h7-8,13,16,20H,2-6,9-12,14-15,22H2,1H3,(H2,23,24,25)/t16?,20-,21-/m0/s1
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n/an/an/an/a 1.20n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313176
PNG
(US10166249, Example 692)
Show SMILES COCCCCCC1CCc2cc(ccc2C1)[C@@H]1CC[C@@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H36NO5P/c1-27-12-4-2-3-5-17-6-7-19-14-20(9-8-18(19)13-17)21-10-11-22(23,15-21)16-28-29(24,25)26/h8-9,14,17,21H,2-7,10-13,15-16,23H2,1H3,(H2,24,25,26)/t17?,21-,22+/m1/s1
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n/an/an/an/a 4.40n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313174
PNG
(US10166249, Example 689)
Show SMILES COCCCCCC1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H36NO5P/c1-27-12-4-2-3-5-17-6-7-19-14-20(9-8-18(19)13-17)21-10-11-22(23,15-21)16-28-29(24,25)26/h8-9,14,17,21H,2-7,10-13,15-16,23H2,1H3,(H2,24,25,26)/t17?,21-,22+/m0/s1
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n/an/an/an/a 5.70n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313179
PNG
(US10166249, Example 697 | US10166249, Example 698)
Show SMILES COc1ccccc1CCC1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C25H34NO5P/c1-30-24-5-3-2-4-19(24)8-6-18-7-9-21-15-22(11-10-20(21)14-18)23-12-13-25(26,16-23)17-31-32(27,28)29/h2-5,10-11,15,18,23H,6-9,12-14,16-17,26H2,1H3,(H2,27,28,29)/t18?,23-,25+/m0/s1
PDB

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n/an/an/an/a 8.90n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65303
PNG
(US10166249, Example 620 | US9522888, 620)
Show SMILES CCCCCC[C@H]1CCc2cc([C@H]3CC[C@](N)(COP(O)(O)=O)C3)c(I)cc2C1
Show InChI InChI=1S/C22H35INO4P/c1-2-3-4-5-6-16-7-8-17-12-20(21(23)13-19(17)11-16)18-9-10-22(24,14-18)15-28-29(25,26)27/h12-13,16,18H,2-11,14-15,24H2,1H3,(H2,25,26,27)/t16-,18-,22+/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65304
PNG
(US10166249, Example 622 | US9522888, 622)
Show SMILES CCCCCC[C@H]1CCc2cc([C@H]3CC[C@](N)(COP(O)(O)=O)C3)c(C)cc2C1
Show InChI InChI=1S/C23H38NO4P/c1-3-4-5-6-7-18-8-9-19-14-22(17(2)12-21(19)13-18)20-10-11-23(24,15-20)16-28-29(25,26)27/h12,14,18,20H,3-11,13,15-16,24H2,1-2H3,(H2,25,26,27)/t18-,20-,23+/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65306
PNG
(US10166249, Example 623 | US9522888, 623)
Show SMILES CCCCCC(=O)OC1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO6P/c1-2-3-4-5-21(24)29-20-9-8-16-12-17(6-7-18(16)13-20)19-10-11-22(23,14-19)15-28-30(25,26)27/h6-7,12,19-20H,2-5,8-11,13-15,23H2,1H3,(H2,25,26,27)/t19-,20?,22+/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313384
PNG
(US10166249, Example 624)
Show SMILES CCCCC(C)(C)C(=O)OC1CCc2cc(ccc2C1)[C@H]1CC[C@@](N)(CO)C1
Show InChI InChI=1S/C24H37NO3/c1-4-5-11-23(2,3)22(27)28-21-9-8-17-13-18(6-7-19(17)14-21)20-10-12-24(25,15-20)16-26/h6-7,13,20-21,26H,4-5,8-12,14-16,25H2,1-3H3/t20-,21?,24-/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313386
PNG
(US10166249, Example 626)
Show SMILES CCCCCCNC(=O)OC1CCc2cc(ccc2C1)[C@H]1CC[C@@](N)(CO)C1
Show InChI InChI=1S/C23H36N2O3/c1-2-3-4-5-12-25-22(27)28-21-9-8-17-13-18(6-7-19(17)14-21)20-10-11-23(24,15-20)16-26/h6-7,13,20-21,26H,2-5,8-12,14-16,24H2,1H3,(H,25,27)/t20-,21?,23-/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65311
PNG
(US10166249, Example 628 | US9522888, 628)
Show SMILES CCCCN(C)C(=O)OC1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H35N2O6P/c1-3-4-11-24(2)21(25)30-20-8-7-16-12-17(5-6-18(16)13-20)19-9-10-22(23,14-19)15-29-31(26,27)28/h5-6,12,19-20H,3-4,7-11,13-15,23H2,1-2H3,(H2,26,27,28)/t19-,20?,22+/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65311
PNG
(US10166249, Example 628 | US9522888, 628)
Show SMILES CCCCN(C)C(=O)OC1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H35N2O6P/c1-3-4-11-24(2)21(25)30-20-8-7-16-12-17(5-6-18(16)13-20)19-9-10-22(23,14-19)15-29-31(26,27)28/h5-6,12,19-20H,3-4,7-11,13-15,23H2,1-2H3,(H2,26,27,28)/t19-,20?,22+/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65314
PNG
(US10166249, Example 629 | US9522888, 629)
Show SMILES CCCCCC(=O)NC1CCc2cc(ccc2C1)[C@H]1CC[C@@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H35N2O5P/c1-2-3-4-5-21(25)24-20-9-8-16-12-17(6-7-18(16)13-20)19-10-11-22(23,14-19)15-29-30(26,27)28/h6-7,12,19-20H,2-5,8-11,13-15,23H2,1H3,(H,24,25)(H2,26,27,28)/t19-,20?,22-/m0/s1
PDB

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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65316
PNG
(US10166249, Example 633 | US9522888, 630)
Show SMILES CCCCC1CCCC2(CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)O1
Show InChI InChI=1S/C24H38NO5P/c1-2-3-5-22-6-4-11-24(30-22)13-10-19-14-18(7-8-20(19)16-24)21-9-12-23(25,15-21)17-29-31(26,27)28/h7-8,14,21-22H,2-6,9-13,15-17,25H2,1H3,(H2,26,27,28)/t21-,22?,23+,24?/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65316
PNG
(US10166249, Example 633 | US9522888, 630)
Show SMILES CCCCC1CCCC2(CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)O1
Show InChI InChI=1S/C24H38NO5P/c1-2-3-5-22-6-4-11-24(30-22)13-10-19-14-18(7-8-20(19)16-24)21-9-12-23(25,15-21)17-29-31(26,27)28/h7-8,14,21-22H,2-6,9-13,15-17,25H2,1H3,(H2,26,27,28)/t21-,22?,23+,24?/m0/s1
PDB

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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65320
PNG
(US10166249, Example 635 | US9522888, 635)
Show SMILES CCCCC1CCc2cc(ccc2C1=O)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C20H30NO5P/c1-2-3-4-14-5-6-16-11-15(7-8-18(16)19(14)22)17-9-10-20(21,12-17)13-26-27(23,24)25/h7-8,11,14,17H,2-6,9-10,12-13,21H2,1H3,(H2,23,24,25)/t14?,17-,20+/m0/s1
PDB

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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65324
PNG
(US10166249, Example 638 | US9522888, 638)
Show SMILES COCCC\C=C\[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO5P/c1-27-12-4-2-3-5-17-6-7-19-14-20(9-8-18(19)13-17)21-10-11-22(23,15-21)16-28-29(24,25)26/h3,5,8-9,14,17,21H,2,4,6-7,10-13,15-16,23H2,1H3,(H2,24,25,26)/b5-3+/t17-,21-,22+/m0/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65327
PNG
(US10166249, Example 640 | US9522888, 640)
Show SMILES COCCC\C=C\[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO5P/c1-27-12-4-2-3-5-17-6-7-19-14-20(9-8-18(19)13-17)21-10-11-22(23,15-21)16-28-29(24,25)26/h3,5,8-9,14,17,21H,2,4,6-7,10-13,15-16,23H2,1H3,(H2,24,25,26)/b5-3+/t17-,21+,22-/m1/s1
PDB

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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65327
PNG
(US10166249, Example 640 | US9522888, 640)
Show SMILES COCCC\C=C\[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO5P/c1-27-12-4-2-3-5-17-6-7-19-14-20(9-8-18(19)13-17)21-10-11-22(23,15-21)16-28-29(24,25)26/h3,5,8-9,14,17,21H,2,4,6-7,10-13,15-16,23H2,1H3,(H2,24,25,26)/b5-3+/t17-,21+,22-/m1/s1
PDB

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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65332
PNG
(US10166249, Example 642 | US9522888, 642)
Show SMILES N[C@]1(COP(O)(O)=O)CC[C@@H](C1)c1ccc2C[C@@H](CCc2c1)\C=C\C1CCOCC1
Show InChI InChI=1S/C23H34NO5P/c24-23(16-29-30(25,26)27)10-7-22(15-23)21-6-5-19-13-18(3-4-20(19)14-21)2-1-17-8-11-28-12-9-17/h1-2,5-6,14,17-18,22H,3-4,7-13,15-16,24H2,(H2,25,26,27)/b2-1+/t18-,22+,23-/m1/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65332
PNG
(US10166249, Example 642 | US9522888, 642)
Show SMILES N[C@]1(COP(O)(O)=O)CC[C@@H](C1)c1ccc2C[C@@H](CCc2c1)\C=C\C1CCOCC1
Show InChI InChI=1S/C23H34NO5P/c24-23(16-29-30(25,26)27)10-7-22(15-23)21-6-5-19-13-18(3-4-20(19)14-21)2-1-17-8-11-28-12-9-17/h1-2,5-6,14,17-18,22H,3-4,7-13,15-16,24H2,(H2,25,26,27)/b2-1+/t18-,22+,23-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65344
PNG
(US10166249, Example 653 | US9522888, 652)
Show SMILES CCC\C=C\C[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO4P/c1-2-3-4-5-6-17-7-8-19-14-20(10-9-18(19)13-17)21-11-12-22(23,15-21)16-27-28(24,25)26/h4-5,9-10,14,17,21H,2-3,6-8,11-13,15-16,23H2,1H3,(H2,24,25,26)/b5-4+/t17-,21+,22-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65344
PNG
(US10166249, Example 653 | US9522888, 652)
Show SMILES CCC\C=C\C[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO4P/c1-2-3-4-5-6-17-7-8-19-14-20(10-9-18(19)13-17)21-11-12-22(23,15-21)16-27-28(24,25)26/h4-5,9-10,14,17,21H,2-3,6-8,11-13,15-16,23H2,1H3,(H2,24,25,26)/b5-4+/t17-,21+,22-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65346
PNG
(US10166249, Example 654 | US9522888, 654)
Show SMILES CCC\C=C\C[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO4P/c1-2-3-4-5-6-17-7-8-19-14-20(10-9-18(19)13-17)21-11-12-22(23,15-21)16-27-28(24,25)26/h4-5,9-10,14,17,21H,2-3,6-8,11-13,15-16,23H2,1H3,(H2,24,25,26)/b5-4+/t17-,21-,22+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65346
PNG
(US10166249, Example 654 | US9522888, 654)
Show SMILES CCC\C=C\C[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO4P/c1-2-3-4-5-6-17-7-8-19-14-20(10-9-18(19)13-17)21-11-12-22(23,15-21)16-27-28(24,25)26/h4-5,9-10,14,17,21H,2-3,6-8,11-13,15-16,23H2,1H3,(H2,24,25,26)/b5-4+/t17-,21-,22+/m0/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65350
PNG
(US10166249, Example 658 | US9522888, 658)
Show SMILES CC\C=C\CC[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO4P/c1-2-3-4-5-6-17-7-8-19-14-20(10-9-18(19)13-17)21-11-12-22(23,15-21)16-27-28(24,25)26/h3-4,9-10,14,17,21H,2,5-8,11-13,15-16,23H2,1H3,(H2,24,25,26)/b4-3+/t17-,21-,22+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65350
PNG
(US10166249, Example 658 | US9522888, 658)
Show SMILES CC\C=C\CC[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H34NO4P/c1-2-3-4-5-6-17-7-8-19-14-20(10-9-18(19)13-17)21-11-12-22(23,15-21)16-27-28(24,25)26/h3-4,9-10,14,17,21H,2,5-8,11-13,15-16,23H2,1H3,(H2,24,25,26)/b4-3+/t17-,21-,22+/m0/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65351
PNG
(US10166249, Example 659 | US9522888, 659)
Show SMILES C\C=C\CCCC[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C23H36NO4P/c1-2-3-4-5-6-7-18-8-9-20-15-21(11-10-19(20)14-18)22-12-13-23(24,16-22)17-28-29(25,26)27/h2-3,10-11,15,18,22H,4-9,12-14,16-17,24H2,1H3,(H2,25,26,27)/b3-2+/t18-,22-,23+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65352
PNG
(US10166249, Example 660 | US9522888, 660)
Show SMILES C\C=C/CCCC[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C23H36NO4P/c1-2-3-4-5-6-7-18-8-9-20-15-21(11-10-19(20)14-18)22-12-13-23(24,16-22)17-28-29(25,26)27/h2-3,10-11,15,18,22H,4-9,12-14,16-17,24H2,1H3,(H2,25,26,27)/b3-2-/t18-,22-,23+/m0/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65354
PNG
(US10166249, Example 661 | US9522888, 661)
Show SMILES C\C=C/CCCC[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C23H36NO4P/c1-2-3-4-5-6-7-18-8-9-20-15-21(11-10-19(20)14-18)22-12-13-23(24,16-22)17-28-29(25,26)27/h2-3,10-11,15,18,22H,4-9,12-14,16-17,24H2,1H3,(H2,25,26,27)/b3-2-/t18-,22+,23-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65354
PNG
(US10166249, Example 661 | US9522888, 661)
Show SMILES C\C=C/CCCC[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C23H36NO4P/c1-2-3-4-5-6-7-18-8-9-20-15-21(11-10-19(20)14-18)22-12-13-23(24,16-22)17-28-29(25,26)27/h2-3,10-11,15,18,22H,4-9,12-14,16-17,24H2,1H3,(H2,25,26,27)/b3-2-/t18-,22+,23-/m1/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65355
PNG
(US10166249, Example 664 | US9522888, 664)
Show SMILES C\C(=N/OCc1ccccc1)[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C25H33N2O5P/c1-18(27-31-16-19-5-3-2-4-6-19)20-7-8-22-14-23(10-9-21(22)13-20)24-11-12-25(26,15-24)17-32-33(28,29)30/h2-6,9-10,14,20,24H,7-8,11-13,15-17,26H2,1H3,(H2,28,29,30)/b27-18+/t20-,24+,25-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65355
PNG
(US10166249, Example 664 | US9522888, 664)
Show SMILES C\C(=N/OCc1ccccc1)[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C25H33N2O5P/c1-18(27-31-16-19-5-3-2-4-6-19)20-7-8-22-14-23(10-9-21(22)13-20)24-11-12-25(26,15-24)17-32-33(28,29)30/h2-6,9-10,14,20,24H,7-8,11-13,15-17,26H2,1H3,(H2,28,29,30)/b27-18+/t20-,24+,25-/m1/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65356
PNG
(US10166249, Example 665 | US9522888, 665)
Show SMILES CCCCO\N=C(/C)[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H35N2O5P/c1-3-4-11-28-24-16(2)17-5-6-19-13-20(8-7-18(19)12-17)21-9-10-22(23,14-21)15-29-30(25,26)27/h7-8,13,17,21H,3-6,9-12,14-15,23H2,1-2H3,(H2,25,26,27)/b24-16+/t17-,21+,22-/m1/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65360
PNG
(US10166249, Example 668 | US9522888, 668)
Show SMILES CCCCS(=O)C[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C21H34NO5PS/c1-2-3-10-29(26)14-16-4-5-18-12-19(7-6-17(18)11-16)20-8-9-21(22,13-20)15-27-28(23,24)25/h6-7,12,16,20H,2-5,8-11,13-15,22H2,1H3,(H2,23,24,25)/t16-,20+,21-,29?/m1/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65198
PNG
(US10166249, Example 539 | US9522888, 539)
Show SMILES CC(C)CSCC[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H36NO4PS/c1-16(2)14-29-10-8-17-3-4-19-12-20(6-5-18(19)11-17)21-7-9-22(23,13-21)15-27-28(24,25)26/h5-6,12,16-17,21H,3-4,7-11,13-15,23H2,1-2H3,(H2,24,25,26)/t17-,21+,22-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313306
PNG
(US10166249, Example 540)
Show SMILES COCCC1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C19H30NO5P/c1-24-9-7-14-2-3-16-11-17(5-4-15(16)10-14)18-6-8-19(20,12-18)13-25-26(21,22)23/h4-5,11,14,18H,2-3,6-10,12-13,20H2,1H3,(H2,21,22,23)/t14?,18-,19+/m0/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65200
PNG
(US10166249, Example 541 | US9522888, 541)
Show SMILES CCOCC[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C20H32NO5P/c1-2-25-10-8-15-3-4-17-12-18(6-5-16(17)11-15)19-7-9-20(21,13-19)14-26-27(22,23)24/h5-6,12,15,19H,2-4,7-11,13-14,21H2,1H3,(H2,22,23,24)/t15-,19-,20+/m0/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65201
PNG
(US10166249, Example 542 | US9522888, 542)
Show SMILES CC(C)COCC[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H36NO5P/c1-16(2)14-27-10-8-17-3-4-19-12-20(6-5-18(19)11-17)21-7-9-22(23,13-21)15-28-29(24,25)26/h5-6,12,16-17,21H,3-4,7-11,13-15,23H2,1-2H3,(H2,24,25,26)/t17-,21-,22+/m0/s1
PDB

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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65201
PNG
(US10166249, Example 542 | US9522888, 542)
Show SMILES CC(C)COCC[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H36NO5P/c1-16(2)14-27-10-8-17-3-4-19-12-20(6-5-18(19)11-17)21-7-9-22(23,13-21)15-28-29(24,25)26/h5-6,12,16-17,21H,3-4,7-11,13-15,23H2,1-2H3,(H2,24,25,26)/t17-,21-,22+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65202
PNG
(US10166249, Example 543 | US9522888, 543)
Show SMILES CC(C)COCC[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H36NO5P/c1-16(2)14-27-10-8-17-3-4-19-12-20(6-5-18(19)11-17)21-7-9-22(23,13-21)15-28-29(24,25)26/h5-6,12,16-17,21H,3-4,7-11,13-15,23H2,1-2H3,(H2,24,25,26)/t17-,21+,22-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65202
PNG
(US10166249, Example 543 | US9522888, 543)
Show SMILES CC(C)COCC[C@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C22H36NO5P/c1-16(2)14-27-10-8-17-3-4-19-12-20(6-5-18(19)11-17)21-7-9-22(23,13-21)15-28-29(24,25)26/h5-6,12,16-17,21H,3-4,7-11,13-15,23H2,1-2H3,(H2,24,25,26)/t17-,21+,22-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313310
PNG
(US10166249, Example 544 | US10166249, Example 545)
Show SMILES COc1cccc(OCCC2CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)c1
Show InChI InChI=1S/C25H34NO6P/c1-30-23-3-2-4-24(15-23)31-12-10-18-5-6-20-14-21(8-7-19(20)13-18)22-9-11-25(26,16-22)17-32-33(27,28)29/h2-4,7-8,14-15,18,22H,5-6,9-13,16-17,26H2,1H3,(H2,27,28,29)/t18?,22-,25+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM313310
PNG
(US10166249, Example 544 | US10166249, Example 545)
Show SMILES COc1cccc(OCCC2CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)c1
Show InChI InChI=1S/C25H34NO6P/c1-30-23-3-2-4-24(15-23)31-12-10-18-5-6-20-14-21(8-7-19(20)13-18)22-9-11-25(26,16-22)17-32-33(27,28)29/h2-4,7-8,14-15,18,22H,5-6,9-13,16-17,26H2,1H3,(H2,27,28,29)/t18?,22-,25+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65209
PNG
(US10166249, Example 548 | US9522888, 548)
Show SMILES CCOc1cccc(C[C@H]2CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)c1
Show InChI InChI=1S/C25H34NO5P/c1-2-30-24-5-3-4-18(14-24)12-19-6-7-21-15-22(9-8-20(21)13-19)23-10-11-25(26,16-23)17-31-32(27,28)29/h3-5,8-9,14-15,19,23H,2,6-7,10-13,16-17,26H2,1H3,(H2,27,28,29)/t19-,23+,25-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65212
PNG
(US10166249, Example 549 | US9522888, 549)
Show SMILES CCOc1ccc(C[C@@H]2CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)cc1
Show InChI InChI=1S/C25H34NO5P/c1-2-30-24-9-4-18(5-10-24)13-19-3-6-21-15-22(8-7-20(21)14-19)23-11-12-25(26,16-23)17-31-32(27,28)29/h4-5,7-10,15,19,23H,2-3,6,11-14,16-17,26H2,1H3,(H2,27,28,29)/t19-,23-,25+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65215
PNG
(US10166249, Example 550 | US9522888, 550)
Show SMILES COCc1ccc(C[C@@H]2CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)cc1
Show InChI InChI=1S/C25H34NO5P/c1-30-16-19-4-2-18(3-5-19)12-20-6-7-22-14-23(9-8-21(22)13-20)24-10-11-25(26,15-24)17-31-32(27,28)29/h2-5,8-9,14,20,24H,6-7,10-13,15-17,26H2,1H3,(H2,27,28,29)/t20-,24-,25+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65221
PNG
(US10166249, Example 553 | US9522888, 553)
Show SMILES COc1ccc(C[C@@H]2CCc3cc(ccc3C2)[C@H]2CC[C@](N)(COP(O)(O)=O)C2)cc1OC
Show InChI InChI=1S/C25H34NO6P/c1-30-23-8-4-18(13-24(23)31-2)11-17-3-5-20-14-21(7-6-19(20)12-17)22-9-10-25(26,15-22)16-32-33(27,28)29/h4,6-8,13-14,17,22H,3,5,9-12,15-16,26H2,1-2H3,(H2,27,28,29)/t17-,22-,25+/m0/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65224
PNG
(US10166249, Example 556 | US9522888, 556)
Show SMILES CC(C)=CCCC[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C23H36NO4P/c1-17(2)5-3-4-6-18-7-8-20-14-21(10-9-19(20)13-18)22-11-12-23(24,15-22)16-28-29(25,26)27/h5,9-10,14,18,22H,3-4,6-8,11-13,15-16,24H2,1-2H3,(H2,25,26,27)/t18-,22+,23-/m1/s1
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Bristol-Myers Squibb Company

US Patent


Assay Description
Compounds were loaded in a 384 Falcon v-bottom plate (0.5 l/well in a 11 point, 3-fold dilution). Membranes prepared from S1P1/CHO cells or EDG3-Gal5...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
Sphingosine-1-phosphate lyase 1


(Homo sapiens)
BDBM65224
PNG
(US10166249, Example 556 | US9522888, 556)
Show SMILES CC(C)=CCCC[C@@H]1CCc2cc(ccc2C1)[C@H]1CC[C@](N)(COP(O)(O)=O)C1
Show InChI InChI=1S/C23H36NO4P/c1-17(2)5-3-4-6-18-7-8-20-14-21(10-9-19(20)13-18)22-11-12-23(24,15-22)16-28-29(25,26)27/h5,9-10,14,18,22H,3-4,6-8,11-13,15-16,24H2,1-2H3,(H2,25,26,27)/t18-,22+,23-/m1/s1
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n/an/an/an/a<10n/an/an/an/a



Bristol-Myers Squibb Company

US Patent


Assay Description
hS1P1/CHO cells were plated into BD Amine 384-well plates the day before the assay. On the day of the assay, growth medium was removed and replaced w...


US Patent US10166249 (2019)

More data for this
Ligand-Target Pair
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