Affinity DataEC50: 1.60nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY5 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 7.89nMAssay Description:Agonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y5 receptorsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 7.90nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 8.20nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 112nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 172nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 187nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 410nMAssay Description:Agonist activity at NPY5R (unknown origin) by CRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: >500nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: >500nMAssay Description:Agonist activity at human NPYY5 receptor expressed in HEK293 cells assessed as decrease in isoproterenol-induced cAMP level measured every 30 secs fo...More data for this Ligand-Target Pair
Affinity DataEC50: 500nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 790nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 790nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Activation of human Y5R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair