Compile Data Set for Download or QSAR
maximum 50k data
Found 23 of ec50 data for polymerid = 8604
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437028(CHEMBL2403079)
Affinity DataEC50:  1.04E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437028(CHEMBL2403079)
Affinity DataEC50:  1.06E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437029(CHEMBL2403077)
Affinity DataEC50:  1.39E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437026(CHEMBL2403056)
Affinity DataEC50:  1.51E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437022(CHEMBL2403060)
Affinity DataEC50:  2.35E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437027(CHEMBL2403080)
Affinity DataEC50:  3.59E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437038(CHEMBL2403067)
Affinity DataEC50:  3.78E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437021(CHEMBL2403061)
Affinity DataEC50:  3.79E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437025(CHEMBL2403057)
Affinity DataEC50:  4.72E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50424538(CHEMBL2312140)
Affinity DataEC50:  4.73E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437020(CHEMBL2403062)
Affinity DataEC50:  6.64E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437039(CHEMBL2403066)
Affinity DataEC50:  7.99E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437037(CHEMBL2403068)
Affinity DataEC50:  9.14E+3nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437035(CHEMBL2403070)
Affinity DataEC50:  1.09E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437023(CHEMBL2403059)
Affinity DataEC50:  1.24E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437036(CHEMBL2403069)
Affinity DataEC50:  1.68E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437040(CHEMBL2403065)
Affinity DataEC50:  1.76E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437030(CHEMBL2403075)
Affinity DataEC50:  2.13E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437034(CHEMBL2403071)
Affinity DataEC50:  2.77E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437024(CHEMBL2403058)
Affinity DataEC50:  3.95E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437031(CHEMBL2403074)
Affinity DataEC50:  3.96E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437032(CHEMBL2403073)
Affinity DataEC50:  5.01E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50437033(CHEMBL2403072)
Affinity DataEC50:  6.13E+4nMAssay Description:Inhibition of PAK1 in human OVCAR3 cells assessed as MEK phosphorylation by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed