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Compile Data Set for Download or QSAR

Found 354 hits of ic50 data for polymerid = 50001330   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271230
PNG
(US10059720, Example 45)
Show SMILES CS(=O)(=O)c1ccc(cc1)-c1ccc(cc1)[C@H](N)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C28H32N2O6S/c1-37(34,35)25-13-11-20(12-14-25)19-7-9-21(10-8-19)26(29)28(33,27(31)32)18-22-17-24(15-16-30-22)36-23-5-3-2-4-6-23/h7-17,23,26,33H,2-6,18,29H2,1H3,(H,31,32)/t26-,28+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271257
PNG
(US10059720, Example 72)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OCCC(C)(C)C)c(C)cn1)C(O)=O
Show InChI InChI=1/C20H34N2O4/c1-13(2)9-17(21)20(25,18(23)24)11-15-10-16(14(3)12-22-15)26-8-7-19(4,5)6/h10,12-13,17,25H,7-9,11,21H2,1-6H3,(H,23,24)/t17-,20+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271275
PNG
(US10059720, Example 90)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(ccn1)N1CCC(C)(C)CC1)C(O)=O
Show InChI InChI=1/C20H33N3O3/c1-14(2)11-17(21)20(26,18(24)25)13-15-12-16(5-8-22-15)23-9-6-19(3,4)7-10-23/h5,8,12,14,17,26H,6-7,9-11,13,21H2,1-4H3,(H,24,25)/t17-,20+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271198
PNG
(US10059720, Example 13)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(ccn1)N1CCCCC1)C(O)=O
Show InChI InChI=1/C18H29N3O3/c1-13(2)10-16(19)18(24,17(22)23)12-14-11-15(6-7-20-14)21-8-4-3-5-9-21/h6-7,11,13,16,24H,3-5,8-10,12,19H2,1-2H3,(H,22,23)/t16-,18+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271277
PNG
(US10059720, Example 92)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(O[C@H](C)Cc2ccccc2)ccn1)C(O)=O
Show InChI InChI=1/C22H30N2O4/c1-15(2)11-20(23)22(27,21(25)26)14-18-13-19(9-10-24-18)28-16(3)12-17-7-5-4-6-8-17/h4-10,13,15-16,20,27H,11-12,14,23H2,1-3H3,(H,25,26)/t16-,20+,22-/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271272
PNG
(US10059720, Example 87)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OC2CCN(CC2)C(=O)OCc2ccccc2)ccn1)C(O)=O
Show InChI InChI=1/C26H35N3O6/c1-18(2)14-23(27)26(33,24(30)31)16-20-15-22(8-11-28-20)35-21-9-12-29(13-10-21)25(32)34-17-19-6-4-3-5-7-19/h3-8,11,15,18,21,23,33H,9-10,12-14,16-17,27H2,1-2H3,(H,30,31)/t23-,26+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271190
PNG
(US10059720, Example 6)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(O[C@H]2CC[C@H](C)CC2)ccn1)C(O)=O
Show InChI InChI=1/C20H32N2O4/c1-13(2)10-18(21)20(25,19(23)24)12-15-11-17(8-9-22-15)26-16-6-4-14(3)5-7-16/h8-9,11,13-14,16,18,25H,4-7,10,12,21H2,1-3H3,(H,23,24)/t14-,16-,18-,20+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271330
PNG
(US10059720, Example 145)
Show SMILES CCCSC[C@H](N)[C@](O)(Cc1cc(O[C@H]2CC[C@H](C)CC2)ccn1)C(O)=O
Show InChI InChI=1/C20H32N2O4S/c1-3-10-27-13-18(21)20(25,19(23)24)12-15-11-17(8-9-22-15)26-16-6-4-14(2)5-7-16/h8-9,11,14,16,18,25H,3-7,10,12-13,21H2,1-2H3,(H,23,24)/t14-,16-,18-,20+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271288
PNG
(US10059720, Example 103)
Show SMILES CSC[C@H](N)[C@](O)(Cc1cc(O[C@H]2CC[C@H](C)CC2)ccn1)C(O)=O
Show InChI InChI=1/C18H28N2O4S/c1-12-3-5-14(6-4-12)24-15-7-8-20-13(9-15)10-18(23,17(21)22)16(19)11-25-2/h7-9,12,14,16,23H,3-6,10-11,19H2,1-2H3,(H,21,22)/t12-,14-,16-,18+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271218
PNG
(US10059720, Example 33)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc2n(CCC3CCCCC3)cnc2cn1)C(O)=O
Show InChI InChI=1/C22H34N4O3/c1-15(2)10-20(23)22(29,21(27)28)12-17-11-19-18(13-24-17)25-14-26(19)9-8-16-6-4-3-5-7-16/h11,13-16,20,29H,3-10,12,23H2,1-2H3,(H,27,28)/t20-,22+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271280
PNG
(US10059720, Example 95)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OCCc2ccsc2)ccn1)C(O)=O
Show InChI InChI=1/C19H26N2O4S/c1-13(2)9-17(20)19(24,18(22)23)11-15-10-16(3-6-21-15)25-7-4-14-5-8-26-12-14/h3,5-6,8,10,12-13,17,24H,4,7,9,11,20H2,1-2H3,(H,22,23)/t17-,19+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271232
PNG
(US10059720, Example 47)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OC2CC3CCC2C3)ccn1)C(O)=O
Show InChI InChI=1/C20H30N2O4/c1-12(2)7-18(21)20(25,19(23)24)11-15-10-16(5-6-22-15)26-17-9-13-3-4-14(17)8-13/h5-6,10,12-14,17-18,25H,3-4,7-9,11,21H2,1-2H3,(H,23,24)/t13?,14?,17?,18-,20+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271258
PNG
(US10059720, Example 73)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(O[C@H]2CC[C@H](C)CC2)c(C)cn1)C(O)=O
Show InChI InChI=1/C21H34N2O4/c1-13(2)9-19(22)21(26,20(24)25)11-16-10-18(15(4)12-23-16)27-17-7-5-14(3)6-8-17/h10,12-14,17,19,26H,5-9,11,22H2,1-4H3,(H,24,25)/t14-,17-,19-,21+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401355
PNG
(US10005762, Example 35)
Show SMILES CSC[C@H](N)[C@](O)(Cc1cc(CCCCC2CC2)c(C)cn1)C(O)=O
Show InChI InChI=1S/C19H30N2O3S/c1-13-11-21-16(9-15(13)6-4-3-5-14-7-8-14)10-19(24,18(22)23)17(20)12-25-2/h9,11,14,17,24H,3-8,10,12,20H2,1-2H3,(H,22,23)/t17-,19+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271245
PNG
(US10059720, Example 60)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OC2CC(C)(C)OC(C)(C)C2)ccn1)C(O)=O
Show InChI InChI=1/C22H36N2O5/c1-14(2)9-18(23)22(27,19(25)26)11-15-10-16(7-8-24-15)28-17-12-20(3,4)29-21(5,6)13-17/h7-8,10,14,17-18,27H,9,11-13,23H2,1-6H3,(H,25,26)/t18-,22+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271233
PNG
(US10059720, Example 48)
Show SMILES N[C@@H](c1ccc(cc1)N1CCOCC1)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C25H33N3O5/c26-23(18-6-8-20(9-7-18)28-12-14-32-15-13-28)25(31,24(29)30)17-19-16-22(10-11-27-19)33-21-4-2-1-3-5-21/h6-11,16,21,23,31H,1-5,12-15,17,26H2,(H,29,30)/t23-,25+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271229
PNG
(US10059720, Example 44)
Show SMILES N[C@@H](c1ccc(cc1)-c1cccnc1)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C26H29N3O4/c27-24(19-10-8-18(9-11-19)20-5-4-13-28-17-20)26(32,25(30)31)16-21-15-23(12-14-29-21)33-22-6-2-1-3-7-22/h4-5,8-15,17,22,24,32H,1-3,6-7,16,27H2,(H,30,31)/t24-,26+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401368
PNG
(US10005762, Example 48)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(\C=C\c2ccccc2)c(C)cn1)C(O)=O
Show InChI InChI=1S/C22H28N2O3/c1-15(2)11-20(23)22(27,21(25)26)13-19-12-18(16(3)14-24-19)10-9-17-7-5-4-6-8-17/h4-10,12,14-15,20,27H,11,13,23H2,1-3H3,(H,25,26)/b10-9+/t20-,22+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271210
PNG
(US10059720, Example 25)
Show SMILES CCCCCCn1ccc2cnc(C[C@@](O)([C@@H](N)CC(C)C)C(O)=O)cc12
Show InChI InChI=1/C21H33N3O3/c1-4-5-6-7-9-24-10-8-16-14-23-17(12-18(16)24)13-21(27,20(25)26)19(22)11-15(2)3/h8,10,12,14-15,19,27H,4-7,9,11,13,22H2,1-3H3,(H,25,26)/t19-,21+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271252
PNG
(US10059720, Example 67)
Show SMILES N[C@@H](C=C1CCOCC1)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C21H30N2O5/c22-19(12-15-7-10-27-11-8-15)21(26,20(24)25)14-16-13-18(6-9-23-16)28-17-4-2-1-3-5-17/h6,9,12-13,17,19,26H,1-5,7-8,10-11,14,22H2,(H,24,25)/t19-,21+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271246
PNG
(US10059720, Example 61)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(O[C@H]2CC[C@]3(CCCO3)CC2)ccn1)C(O)=O
Show InChI InChI=1/C22H34N2O5/c1-15(2)12-19(23)22(27,20(25)26)14-16-13-18(6-10-24-16)29-17-4-8-21(9-5-17)7-3-11-28-21/h6,10,13,15,17,19,27H,3-5,7-9,11-12,14,23H2,1-2H3,(H,25,26)/t17-,19-,21+,22+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271290
PNG
(US10059720, Example 105)
Show SMILES CCSC[C@H](N)[C@](O)(Cc1cc(O[C@H]2CC[C@H](C)CC2)ccn1)C(O)=O
Show InChI InChI=1/C19H30N2O4S/c1-3-26-12-17(20)19(24,18(22)23)11-14-10-16(8-9-21-14)25-15-6-4-13(2)5-7-15/h8-10,13,15,17,24H,3-7,11-12,20H2,1-2H3,(H,22,23)/t13-,15-,17-,19+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271211
PNG
(US10059720, Example 26)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(O[C@@H]2C[C@@H]3C[C@@H]3C2)ccn1)C(O)=O
Show InChI InChI=1/C19H28N2O4/c1-11(2)5-17(20)19(24,18(22)23)10-14-9-15(3-4-21-14)25-16-7-12-6-13(12)8-16/h3-4,9,11-13,16-17,24H,5-8,10,20H2,1-2H3,(H,22,23)/t12-,13+,16+,17-,19+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271241
PNG
(US10059720, Example 56)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(O[C@@H]2CC[C@H](C)CC2)ccn1)C(O)=O
Show InChI InChI=1/C20H32N2O4/c1-13(2)10-18(21)20(25,19(23)24)12-15-11-17(8-9-22-15)26-16-6-4-14(3)5-7-16/h8-9,11,13-14,16,18,25H,4-7,10,12,21H2,1-3H3,(H,23,24)/t14-,16+,18-,20+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM50245396
PNG
(CHEMBL4101200)
Show SMILES N[C@@H](CCc1ccccc1)P(O)(=O)C[C@@H](CC#C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
Show InChI InChI=1/C24H30N3O4P/c1-2-9-20(17-32(30,31)22(25)15-14-18-10-5-3-6-11-18)24(29)27-21(23(26)28)16-19-12-7-4-8-13-19/h1,3-8,10-13,20-22H,9,14-17,25H2,(H2,26,28)(H,27,29)(H,30,31)/t20-,21+,22-/s2
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National and Kapodistrian University of Athens

Curated by ChEMBL


Assay Description
Inhibition of IRAP (unknown origin) expressed in HEK 293S GnTI(-) cells by in vitro fluorimetric assay


J Med Chem 59: 9107-9123 (2016)


Article DOI: 10.1021/acs.jmedchem.6b01031
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401389
PNG
(US10005762, Example 69)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1nccc2CC(CC3(C)CC3)Cc12)C(O)=O
Show InChI InChI=1S/C21H32N2O3/c1-13(2)8-18(22)21(26,19(24)25)12-17-16-10-14(11-20(3)5-6-20)9-15(16)4-7-23-17/h4,7,13-14,18,26H,5-6,8-12,22H2,1-3H3,(H,24,25)/t14?,18-,21+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271240
PNG
(US10059720, Example 55)
Show SMILES CCCC[C@@H](C)Oc1ccnc(C[C@@](O)([C@@H](N)CC(C)C)C(O)=O)c1
Show InChI InChI=1/C19H32N2O4/c1-5-6-7-14(4)25-16-8-9-21-15(11-16)12-19(24,18(22)23)17(20)10-13(2)3/h8-9,11,13-14,17,24H,5-7,10,12,20H2,1-4H3,(H,22,23)/t14-,17+,19-/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401393
PNG
(US10005762, Example 73)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(CCCCC2CC2)c(C)cn1)C(O)=O
Show InChI InChI=1S/C21H34N2O3/c1-14(2)10-19(22)21(26,20(24)25)12-18-11-17(15(3)13-23-18)7-5-4-6-16-8-9-16/h11,13-14,16,19,26H,4-10,12,22H2,1-3H3,(H,24,25)/t19-,21+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271251
PNG
(US10059720, Example 66)
Show SMILES CC(C)CC[C@H](N)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C20H32N2O4/c1-14(2)8-9-18(21)20(25,19(23)24)13-15-12-17(10-11-22-15)26-16-6-4-3-5-7-16/h10-12,14,16,18,25H,3-9,13,21H2,1-2H3,(H,23,24)/t18-,20+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271260
PNG
(US10059720, Example 75)
Show SMILES COCCCCC[C@H](N)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C21H34N2O5/c1-27-13-7-3-6-10-19(22)21(26,20(24)25)15-16-14-18(11-12-23-16)28-17-8-4-2-5-9-17/h11-12,14,17,19,26H,2-10,13,15,22H2,1H3,(H,24,25)/t19-,21+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401320
PNG
(US10005762, Example 4(1))
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(CCCC2CC2)c(C)cn1)C(O)=O
Show InChI InChI=1S/C20H32N2O3/c1-13(2)9-18(21)20(25,19(23)24)11-17-10-16(14(3)12-22-17)6-4-5-15-7-8-15/h10,12-13,15,18,25H,4-9,11,21H2,1-3H3,(H,23,24)/t18-,20+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271188
PNG
(US10059720, Example 4)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OC2CCC3(CC3)CC2)ccn1)C(O)=O
Show InChI InChI=1/C21H32N2O4/c1-14(2)11-18(22)21(26,19(24)25)13-15-12-17(5-10-23-15)27-16-3-6-20(7-4-16)8-9-20/h5,10,12,14,16,18,26H,3-4,6-9,11,13,22H2,1-2H3,(H,24,25)/t18-,21+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401319
PNG
(US10005762, Example 3)
Show SMILES Cc1cnc(C[C@@](O)([C@@H](N)CCC2CC2)C(O)=O)cc1CCCC1CC1
Show InChI InChI=1S/C21H32N2O3/c1-14-13-23-18(11-17(14)4-2-3-15-5-6-15)12-21(26,20(24)25)19(22)10-9-16-7-8-16/h11,13,15-16,19,26H,2-10,12,22H2,1H3,(H,24,25)/t19-,21+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM284929
PNG
(US10023583, Example 2)
Show SMILES CSC[C@H](N)[C@](O)(Cc1nccc2oc(CCC3CC3)cc12)C(O)=O
Show InChI InChI=1/C18H24N2O4S/c1-25-10-16(19)18(23,17(21)22)9-14-13-8-12(5-4-11-2-3-11)24-15(13)6-7-20-14/h6-8,11,16,23H,2-5,9-10,19H2,1H3,(H,21,22)/t16-,18+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10023583 (2018)


Article DOI: 10.1038/nm1003
BindingDB Entry DOI: 10.7270/Q29Z96X2
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271187
PNG
(US10059720, Example 3)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C19H30N2O4/c1-13(2)10-17(20)19(24,18(22)23)12-14-11-16(8-9-21-14)25-15-6-4-3-5-7-15/h8-9,11,13,15,17,24H,3-7,10,12,20H2,1-2H3,(H,22,23)/t17-,19+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401394
PNG
(US10005762, Example 74)
Show SMILES CCCCCc1cc(C[C@@](O)([C@@H](N)CC(C)C)C(O)=O)ncc1C
Show InChI InChI=1S/C19H32N2O3/c1-5-6-7-8-15-10-16(21-12-14(15)4)11-19(24,18(22)23)17(20)9-13(2)3/h10,12-13,17,24H,5-9,11,20H2,1-4H3,(H,22,23)/t17-,19+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271221
PNG
(US10059720, Example 36)
Show SMILES N[C@@H](c1ccc(cc1)-c1ccccc1)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C27H30N2O4/c28-25(21-13-11-20(12-14-21)19-7-3-1-4-8-19)27(32,26(30)31)18-22-17-24(15-16-29-22)33-23-9-5-2-6-10-23/h1,3-4,7-8,11-17,23,25,32H,2,5-6,9-10,18,28H2,(H,30,31)/t25-,27+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271262
PNG
(US10059720, Example 77)
Show SMILES Cc1ccc(OC[C@H](N)[C@](O)(Cc2cc(OC3CCCCC3)ccn2)C(O)=O)nc1
Show InChI InChI=1/C22H29N3O5/c1-15-7-8-20(25-13-15)29-14-19(23)22(28,21(26)27)12-16-11-18(9-10-24-16)30-17-5-3-2-4-6-17/h7-11,13,17,19,28H,2-6,12,14,23H2,1H3,(H,26,27)/t19-,22+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401322
PNG
(US10005762, Example 4(3))
Show SMILES CCC(O)CCCc1cc(C[C@@](O)([C@@H](N)CC(C)C)C(O)=O)ncc1C
Show InChI InChI=1S/C20H34N2O4/c1-5-17(23)8-6-7-15-10-16(22-12-14(15)4)11-20(26,19(24)25)18(21)9-13(2)3/h10,12-13,17-18,23,26H,5-9,11,21H2,1-4H3,(H,24,25)/t17?,18-,20+/m0/s1
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Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271215
PNG
(US10059720, Example 30)
Show SMILES COCc1ccc(OC[C@H](N)[C@](O)(Cc2cc(OC3CCCCC3)ccn2)C(O)=O)cc1
Show InChI InChI=1/C24H32N2O6/c1-30-15-17-7-9-19(10-8-17)31-16-22(25)24(29,23(27)28)14-18-13-21(11-12-26-18)32-20-5-3-2-4-6-20/h7-13,20,22,29H,2-6,14-16,25H2,1H3,(H,27,28)/t22-,24+/s2
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n/an/a 2.70n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271228
PNG
(US10059720, Example 43)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OC2C3CC4CC(C3)CC2C4)ccn1)C(O)=O
Show InChI InChI=1/C23H34N2O4/c1-13(2)5-20(24)23(28,22(26)27)12-18-11-19(3-4-25-18)29-21-16-7-14-6-15(9-16)10-17(21)8-14/h3-4,11,13-17,20-21,28H,5-10,12,24H2,1-2H3,(H,26,27)/t14?,15?,16?,17?,20-,21?,23+/s2
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n/an/a 2.80n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271309
PNG
(US10059720, Example 124)
Show SMILES C[C@H]1CC[C@@H](CC1)Oc1ccnc(C[C@@](O)([C@@H](N)CC(C)(C)C)C(O)=O)c1
Show InChI InChI=1/C21H34N2O4/c1-14-5-7-16(8-6-14)27-17-9-10-23-15(11-17)12-21(26,19(24)25)18(22)13-20(2,3)4/h9-11,14,16,18,26H,5-8,12-13,22H2,1-4H3,(H,24,25)/t14-,16-,18-,21+/s2
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n/an/a 2.90n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271213
PNG
(US10059720, Example 28)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OCCC2(C)CC2)ccn1)C(O)=O
Show InChI InChI=1/C19H30N2O4/c1-13(2)10-16(20)19(24,17(22)23)12-14-11-15(4-8-21-14)25-9-7-18(3)5-6-18/h4,8,11,13,16,24H,5-7,9-10,12,20H2,1-3H3,(H,22,23)/t16-,19+/s2
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n/an/a 2.90n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271234
PNG
(US10059720, Example 49)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OC2Cc3ccccc3C2)ccn1)C(O)=O
Show InChI InChI=1/C22H28N2O4/c1-14(2)9-20(23)22(27,21(25)26)13-17-12-18(7-8-24-17)28-19-10-15-5-3-4-6-16(15)11-19/h3-8,12,14,19-20,27H,9-11,13,23H2,1-2H3,(H,25,26)/t20-,22+/s2
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n/an/a 2.90n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271285
PNG
(US10059720, Example 100)
Show SMILES CCCCCCOc1ccnc(C[C@@](O)([C@@H](N)CC(C)C)C(O)=O)c1
Show InChI InChI=1/C19H32N2O4/c1-4-5-6-7-10-25-16-8-9-21-15(12-16)13-19(24,18(22)23)17(20)11-14(2)3/h8-9,12,14,17,24H,4-7,10-11,13,20H2,1-3H3,(H,22,23)/t17-,19+/s2
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n/an/a 3n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271225
PNG
(US10059720, Example 40)
Show SMILES N[C@@H](\C=C\c1ccccc1)[C@](O)(Cc1cc(OC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C23H28N2O4/c24-21(12-11-17-7-3-1-4-8-17)23(28,22(26)27)16-18-15-20(13-14-25-18)29-19-9-5-2-6-10-19/h1,3-4,7-8,11-15,19,21,28H,2,5-6,9-10,16,24H2,(H,26,27)/b12-11+/t21-,23+/s2
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n/an/a 3n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271282
PNG
(US10059720, Example 97)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OCCOC2CCCCC2)ccn1)C(O)=O
Show InChI InChI=1/C21H34N2O5/c1-15(2)12-19(22)21(26,20(24)25)14-16-13-18(8-9-23-16)28-11-10-27-17-6-4-3-5-7-17/h8-9,13,15,17,19,26H,3-7,10-12,14,22H2,1-2H3,(H,24,25)/t19-,21+/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271243
PNG
(US10059720, Example 58)
Show SMILES CC(C)C[C@@H](C)Oc1ccnc(C[C@@](O)([C@@H](N)CC(C)C)C(O)=O)c1
Show InChI InChI=1/C19H32N2O4/c1-12(2)8-14(5)25-16-6-7-21-15(10-16)11-19(24,18(22)23)17(20)9-13(3)4/h6-7,10,12-14,17,24H,8-9,11,20H2,1-5H3,(H,22,23)/t14-,17+,19-/s2
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Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
Aminopeptidase


(Homo sapiens (Human))
BDBM401395
PNG
(US10005762, Example 75)
Show SMILES CCCCCCc1cc(C[C@@](O)([C@@H](N)CC(C)C)C(O)=O)ncc1C
Show InChI InChI=1S/C20H34N2O3/c1-5-6-7-8-9-16-11-17(22-13-15(16)4)12-20(25,19(23)24)18(21)10-14(2)3/h11,13-14,18,25H,5-10,12,21H2,1-4H3,(H,23,24)/t18-,20+/m0/s1
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n/an/a 3.10n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
The inventors have assumed that inhibition of nocturnal activity of placental leucine aminopeptidase (P-LAP), i.e. aminopeptidase that cleaves AVP, w...


US Patent US10005762 (2018)

More data for this
Ligand-Target Pair
Leucyl-cystinyl aminopeptidase


(Homo sapiens (Human))
BDBM271199
PNG
(US10059720, Example 14)
Show SMILES CC(C)C[C@H](N)[C@](O)(Cc1cc(OCc2cccc3ccccc23)ccn1)C(O)=O
Show InChI InChI=1/C24H28N2O4/c1-16(2)12-22(25)24(29,23(27)28)14-19-13-20(10-11-26-19)30-15-18-8-5-7-17-6-3-4-9-21(17)18/h3-11,13,16,22,29H,12,14-15,25H2,1-2H3,(H,27,28)/t22-,24+/s2
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n/an/a 3.10n/an/an/an/an/an/a



Astellas Pharma Inc

US Patent


Assay Description
HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...


US Patent US10059720 (2018)


Article DOI: 10.1021/jm970124v
BindingDB Entry DOI: 10.7270/Q2XD13Q5
More data for this
Ligand-Target Pair
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