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Compile Data Set for Download or QSAR

Found 25 hits of ic50 data for polymerid = 5332   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM50022815
PNG
((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Show SMILES CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C
Show InChI InChI=1/C62H111N11O12/c1-25-27-28-40(15)52(75)51-56(79)65-43(26-2)58(81)67(18)33-48(74)68(19)44(29-34(3)4)55(78)66-49(38(11)12)61(84)69(20)45(30-35(5)6)54(77)63-41(16)53(76)64-42(17)57(80)70(21)46(31-36(7)8)59(82)71(22)47(32-37(9)10)60(83)72(23)50(39(13)14)62(85)73(51)24/h25,27,34-47,49-52,75H,26,28-33H2,1-24H3,(H,63,77)(H,64,76)(H,65,79)(H,66,78)/b27-25+/t40-,41+,42-,43+,44+,45+,46+,47+,49+,50+,51+,52-/s2
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n/an/a 3.60n/an/an/an/an/an/a



University of Kansas

Curated by ChEMBL


Assay Description
Inhibition of human recombinant cyclophilin D using Suc-AAPF-MCA as substrate preincubated for 1 hr followed by substrate addition measured per milli...


ACS Med Chem Lett 7: 294-9 (2016)


Article DOI: 10.1021/acsmedchemlett.5b00451
BindingDB Entry DOI: 10.7270/Q24T6M8F
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140005
PNG
(US8901295, F684)
Show SMILES CSc1ccccc1C1CCCN1C(=O)CNC(=O)NCc1ccc(N)cc1
Show InChI InChI=1/C21H26N4O2S/c1-28-19-7-3-2-5-17(19)18-6-4-12-25(18)20(26)14-24-21(27)23-13-15-8-10-16(22)11-9-15/h2-3,5,7-11,18H,4,6,12-14,22H2,1H3,(H2,23,24,27)
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n/an/a 640n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140008
PNG
(US8901295, F716)
Show SMILES CSCCC(NC(=O)NCc1ccc(N)cc1)C(=O)N1CCCC1c1ccccc1SC
Show InChI InChI=1/C24H32N4O2S2/c1-31-15-13-20(27-24(30)26-16-17-9-11-18(25)12-10-17)23(29)28-14-5-7-21(28)19-6-3-4-8-22(19)32-2/h3-4,6,8-12,20-21H,5,7,13-16,25H2,1-2H3,(H2,26,27,30)
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n/an/a 660n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140007
PNG
(US8901295, F714)
Show SMILES CSc1ccccc1C1CCCN1C(=O)C(C)NC(=O)NCc1ccc(N)cc1
Show InChI InChI=1/C22H28N4O2S/c1-15(25-22(28)24-14-16-9-11-17(23)12-10-16)21(27)26-13-5-7-19(26)18-6-3-4-8-20(18)29-2/h3-4,6,8-12,15,19H,5,7,13-14,23H2,1-2H3,(H2,24,25,28)
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n/an/a 1.10E+3n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140004
PNG
(US8901295, F680)
Show SMILES Nc1ccc(CNC(=O)NCC(=O)N2CCCC2c2ccccc2Br)cc1
Show InChI InChI=1/C20H23BrN4O2/c21-17-5-2-1-4-16(17)18-6-3-11-25(18)19(26)13-24-20(27)23-12-14-7-9-15(22)10-8-14/h1-2,4-5,7-10,18H,3,6,11-13,22H2,(H2,23,24,27)
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n/an/a 1.10E+3n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140002
PNG
(US8901295, F671)
Show SMILES Nc1ccc(CNC(=O)NCC(=O)N2CCCC2c2cccc3ccccc23)cc1
Show InChI InChI=1/C24H26N4O2/c25-19-12-10-17(11-13-19)15-26-24(30)27-16-23(29)28-14-4-9-22(28)21-8-3-6-18-5-1-2-7-20(18)21/h1-3,5-8,10-13,22H,4,9,14-16,25H2,(H2,26,27,30)
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n/an/a 1.40E+3n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM50169545
PNG
(CHEMBL3805631)
Show SMILES CC(C)COc1ccc(cc1C#N)-c1nc(C)c(s1)C(=O)Nc1ccc(cc1)S(N)(=O)=O
Show InChI InChI=1S/C22H22N4O4S2/c1-13(2)12-30-19-9-4-15(10-16(19)11-23)22-25-14(3)20(31-22)21(27)26-17-5-7-18(8-6-17)32(24,28)29/h4-10,13H,12H2,1-3H3,(H,26,27)(H2,24,28,29)
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n/an/a 1.49E+3n/an/an/an/an/an/a



University of Kansas

Curated by ChEMBL


Assay Description
Inhibition of human recombinant cyclophilin D using Suc-AAPF-MCA as substrate preincubated for 1 hr followed by substrate addition measured per milli...


ACS Med Chem Lett 7: 294-9 (2016)


Article DOI: 10.1021/acsmedchemlett.5b00451
BindingDB Entry DOI: 10.7270/Q24T6M8F
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140006
PNG
(US8901295, F712)
Show SMILES CSc1ccccc1C1CCCN1C(=O)C(CC(C)C)NC(=O)NCc1ccc(N)cc1
Show InChI InChI=1/C25H34N4O2S/c1-17(2)15-21(28-25(31)27-16-18-10-12-19(26)13-11-18)24(30)29-14-6-8-22(29)20-7-4-5-9-23(20)32-3/h4-5,7,9-13,17,21-22H,6,8,14-16,26H2,1-3H3,(H2,27,28,31)
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n/an/a 3.00E+3n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM139995
PNG
(US8901295, F428)
Show SMILES CCOC(=O)CNC(=O)NCc1ccc(N)cc1
Show InChI InChI=1S/C12H17N3O3/c1-2-18-11(16)8-15-12(17)14-7-9-3-5-10(13)6-4-9/h3-6H,2,7-8,13H2,1H3,(H2,14,15,17)
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n/an/a 6.20E+3n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140003
PNG
(US8901295, F673)
Show SMILES Nc1ccc(CNC(=O)NCC(=O)N2CCCC2c2ccccc2Cl)cc1
Show InChI InChI=1/C20H23ClN4O2/c21-17-5-2-1-4-16(17)18-6-3-11-25(18)19(26)13-24-20(27)23-12-14-7-9-15(22)10-8-14/h1-2,4-5,7-10,18H,3,6,11-13,22H2,(H2,23,24,27)
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n/an/a 6.20E+3n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394270
PNG
(US9975902, Example 1)
Show SMILES O[C@@H]1COC2C[C@H]1Nc1ccc(CNC(=O)CN3C(=O)C4[C@@H]5CCC(C5)[C@H]4C3=O)cc21
Show InChI InChI=1S/C23H27N3O5/c27-17-10-31-18-7-16(17)25-15-4-1-11(5-14(15)18)8-24-19(28)9-26-22(29)20-12-2-3-13(6-12)21(20)23(26)30/h1,4-5,12-13,16-18,20-21,25,27H,2-3,6-10H2,(H,24,28)/t12-,13?,16-,17-,18?,20?,21-/m1/s1
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n/an/a<1.00E+4n/an/an/an/an/an/a



Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394274
PNG
(US9975902, Example 4)
Show SMILES [O-][N+](=O)c1ccc(CNC(=O)CN2C(=O)C3[C@@H]4CCC(C4)[C@@H]3C2=O)cc1
Show InChI InChI=1S/C18H19N3O5/c22-14(19-8-10-1-5-13(6-2-10)21(25)26)9-20-17(23)15-11-3-4-12(7-11)16(15)18(20)24/h1-2,5-6,11-12,15-16H,3-4,7-9H2,(H,19,22)/t11-,12?,15?,16+/m1/s1
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n/an/a<1.00E+4n/an/an/an/an/an/a



Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394273
PNG
(US9975902, Example 3)
Show SMILES O[C@@H]1COC2C[C@H]1Nc1ccc(CNC(=O)CN3C(=O)[C@H]4[C@H]5CC[C@H](C5)[C@H]4C3=O)cc21
Show InChI InChI=1S/C23H27N3O5/c27-17-10-31-18-7-16(17)25-15-4-1-11(5-14(15)18)8-24-19(28)9-26-22(29)20-12-2-3-13(6-12)21(20)23(26)30/h1,4-5,12-13,16-18,20-21,25,27H,2-3,6-10H2,(H,24,28)/t12-,13+,16?,17-,18?,20-,21+/m1/s1
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n/an/a<1.00E+4n/an/an/an/an/an/a



Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394272
PNG
(US9975902, Example 2)
Show SMILES O=C(CN1C(=O)[C@H]2[C@H]3CC[C@H](C3)[C@H]2C1=O)NCc1ccc2NCCCc2c1
Show InChI InChI=1S/C21H25N3O3/c25-17(23-10-12-3-6-16-13(8-12)2-1-7-22-16)11-24-20(26)18-14-4-5-15(9-14)19(18)21(24)27/h3,6,8,14-15,18-19,22H,1-2,4-5,7,9-11H2,(H,23,25)/t14-,15+,18-,19+
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n/an/a<1.00E+4n/an/an/an/an/an/a



Merck Patent GmbH

US Patent


Assay Description
The peptidyl-proline isomerase activity (PPase) was determined by using a PPase-chymotrypsin coupled assay with suc-AAPF-p-NA as substrated and color...


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394272
PNG
(US9975902, Example 2)
Show SMILES O=C(CN1C(=O)[C@H]2[C@H]3CC[C@H](C3)[C@H]2C1=O)NCc1ccc2NCCCc2c1
Show InChI InChI=1S/C21H25N3O3/c25-17(23-10-12-3-6-16-13(8-12)2-1-7-22-16)11-24-20(26)18-14-4-5-15(9-14)19(18)21(24)27/h3,6,8,14-15,18-19,22H,1-2,4-5,7,9-11H2,(H,23,25)/t14-,15+,18-,19+
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM140001
PNG
(US8901295, F609)
Show SMILES COc1ccccc1C1CCCN1C(=O)CNC(=O)NCc1ccc(N)cc1
Show InChI InChI=1/C21H26N4O3/c1-28-19-7-3-2-5-17(19)18-6-4-12-25(18)20(26)14-24-21(27)23-13-15-8-10-16(22)11-9-15/h2-3,5,7-11,18H,4,6,12-14,22H2,1H3,(H2,23,24,27)
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n/an/a 1.14E+4n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Cyclophilin D (CypD)


(Homo sapiens (Human))
BDBM46034
PNG
(US8901295, F607)
Show SMILES CCN(OCc1ccccc1)C(=O)CNC(=O)NCc1ccc(N)cc1
Show InChI InChI=1S/C19H24N4O3/c1-2-23(26-14-16-6-4-3-5-7-16)18(24)13-22-19(25)21-12-15-8-10-17(20)11-9-15/h3-11H,2,12-14,20H2,1H3,(H2,21,22,25)
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n/an/a 3.00E+4n/an/an/an/a7.820



University of Montpellier

US Patent


Assay Description
Cyclophilin PPlase activity was measured at 20 C. by using the standard chymotrypsin coupled assay (Kofron J L, Kuzmic P, Kishore V, Colon-Bonilla E,...


US Patent US8901295 (2014)


BindingDB Entry DOI: 10.7270/Q2R49PGS
More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394274
PNG
(US9975902, Example 4)
Show SMILES [O-][N+](=O)c1ccc(CNC(=O)CN2C(=O)C3[C@@H]4CCC(C4)[C@@H]3C2=O)cc1
Show InChI InChI=1S/C18H19N3O5/c22-14(19-8-10-1-5-13(6-2-10)21(25)26)9-20-17(23)15-11-3-4-12(7-11)16(15)18(20)24/h1-2,5-6,11-12,15-16H,3-4,7-9H2,(H,19,22)/t11-,12?,15?,16+/m1/s1
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n/an/a 1.05E+5n/an/an/an/an/an/a



Merck Patent GmbH

US Patent


Assay Description
The peptidyl-proline isomerase activity (PPase) was determined by using a PPase-chymotrypsin coupled assay with suc-AAPF-p-NA as substrated and color...


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394275
PNG
(US9975902, Example 5)
Show SMILES Nc1ccc(cc1)C1(CC1)NC(=O)CN1C(=O)[C@H]2[C@H]3CC[C@H](C3)[C@H]2C1=O
Show InChI InChI=1S/C20H23N3O3/c21-14-5-3-13(4-6-14)20(7-8-20)22-15(24)10-23-18(25)16-11-1-2-12(9-11)17(16)19(23)26/h3-6,11-12,16-17H,1-2,7-10,21H2,(H,22,24)/t11-,12+,16-,17+
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US Patent
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394278
PNG
(US9975902, Example 8)
Show SMILES Nc1ccc(CNC(=O)CN2C(=O)C3C4CCC(O4)C3C2=O)cc1
Show InChI InChI=1S/C17H19N3O4/c18-10-3-1-9(2-4-10)7-19-13(21)8-20-16(22)14-11-5-6-12(24-11)15(14)17(20)23/h1-4,11-12,14-15H,5-8,18H2,(H,19,21)
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US Patent
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394277
PNG
(US9975902, Example 7)
Show SMILES Nc1ccc(CCNC(=O)CN2C(=O)C3CCCCC3C2=O)cc1
Show InChI InChI=1S/C18H23N3O3/c19-13-7-5-12(6-8-13)9-10-20-16(22)11-21-17(23)14-3-1-2-4-15(14)18(21)24/h5-8,14-15H,1-4,9-11,19H2,(H,20,22)
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US Patent
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394281
PNG
(US9975902, Example 11)
Show SMILES CCC1Oc2cc(ccc2NC1=O)C(C)NC(=O)CN1C(=O)[C@H]2[C@H]3CC[C@H](C3)[C@H]2C1=O
Show InChI InChI=1S/C23H27N3O5/c1-3-16-21(28)25-15-7-6-12(9-17(15)31-16)11(2)24-18(27)10-26-22(29)19-13-4-5-14(8-13)20(19)23(26)30/h6-7,9,11,13-14,16,19-20H,3-5,8,10H2,1-2H3,(H,24,27)(H,25,28)/t11?,13-,14+,16?,19-,20+
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394280
PNG
(US9975902, Example 10)
Show SMILES [O-][N+](=O)c1ccc(CCNC(=O)CN2C(=O)C3[C@@H]4CCC(C4)[C@@H]3C2=O)cc1
Show InChI InChI=1S/C19H21N3O5/c23-15(20-8-7-11-1-5-14(6-2-11)22(26)27)10-21-18(24)16-12-3-4-13(9-12)17(16)19(21)25/h1-2,5-6,12-13,16-17H,3-4,7-10H2,(H,20,23)/t12-,13?,16?,17+/m1/s1
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394279
PNG
(US9975902, Example 9)
Show SMILES O=C(CN1C(=O)[C@H]2[C@H]3CC[C@H](C3)[C@H]2C1=O)NCCc1ccc2NCCCc2c1
Show InChI InChI=1S/C22H27N3O3/c26-18(24-9-7-13-3-6-17-14(10-13)2-1-8-23-17)12-25-21(27)19-15-4-5-16(11-15)20(19)22(25)28/h3,6,10,15-16,19-20,23H,1-2,4-5,7-9,11-12H2,(H,24,26)/t15-,16+,19-,20+
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US Patent
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair
Peptidyl-prolyl cis-trans isomerase D


(Homo sapiens (Human))
BDBM394276
PNG
(US9975902, Example 6)
Show SMILES CCN1Cc2cc(CNC(=O)CN3C(=O)C4[C@@H]5CC[C@@H](C5)[C@H]4C3=O)ccc2NCCC1=O
Show InChI InChI=1S/C24H30N4O4/c1-2-27-12-17-9-14(3-6-18(17)25-8-7-20(27)30)11-26-19(29)13-28-23(31)21-15-4-5-16(10-15)22(21)24(28)32/h3,6,9,15-16,21-22,25H,2,4-5,7-8,10-13H2,1H3,(H,26,29)/t15-,16+,21+,22?/m0/s1
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Merck Patent GmbH

US Patent


Assay Description
The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.


US Patent US9975902 (2018)

More data for this
Ligand-Target Pair