Affinity DataKd: 0.220nMAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
Affinity DataKd: 0.220nMpH: 7.4 T: 2°CAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
Affinity DataKd: 0.240nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.1 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.260nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 0.05 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.270nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.1 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.280nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 0.05 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.310nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 100 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.320nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.330nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.340nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.360nMAssay Description:Inhibition of NKA-induced airway contraction of isolated hamster trachea (ht) was used as a measure of NK2-receptor antagonist activity.More data for this Ligand-Target Pair
Affinity DataKd: 0.360nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.360nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor(AR) at 5 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.370nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.370nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 5 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Inhibitory concentration against [3H]-DPCPX binding to Adenosine A1 recepto from DDT1 MF2 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.400nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.460nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
Affinity DataKd: 0.530nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.530nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.530nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.530nMAssay Description:Equilibrium dissociation constant for [3H]-DPCPX binding to Adenosine A1 receptor from DDT1 MF2 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 0.690nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.690nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.700nMAssay Description:Displacement of 2-[2-(4-amino-3-[125I]iodophenyl)ethylamino]adenosine from human recombinant adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.710nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 100 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.710nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.730nMAssay Description:Binding of [3H]-CPX to A1 adenosine receptor of DDT1 MF-2 (DDT) cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.740nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.75nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
Affinity DataKd: 0.790nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.810nMAssay Description:Dissociation constant of [3H]-DPCPX binding to adenosine A1 receptor (AR) at 200 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.820nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.860nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKd: 1.10nMAssay Description:Specific binding of [3H]-CPX to the A1-adenosine receptorMore data for this Ligand-Target Pair