Affinity DataKd: 0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
Affinity DataKd: 0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
Affinity DataKd: 0.00000100nMAssay Description:In vivo inihibition of Beta-1 adrenergic receptor in guinea pig right atria after 40 minMore data for this Ligand-Target Pair
Affinity DataKd: 0.00000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
Affinity DataKd: 0.0000100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
Affinity DataKd: 0.0000100nMAssay Description:In vivo inihibition of Beta-1 adrenergic receptor in guinea pig right atria after 40 minMore data for this Ligand-Target Pair
Affinity DataKd: 0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
Affinity DataKd: 0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 minMore data for this Ligand-Target Pair
Affinity DataKd: 0.00100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
Affinity DataKd: 0.100nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3hMore data for this Ligand-Target Pair
Affinity DataKd: 0.363nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 0.851nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 0.851nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 0.891nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 1.90nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:In vitro ability to block beta-1 adrenergic receptor in guinea pig right atria.More data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Antagonism of the isoprenaline-induced positive chronotropic effect on the atria of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 2.40nMAssay Description:Beta-1 adrenergic receptor blocking activity in atria of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 2.5nMAssay Description:In vitro ability to block beta-1 adrenergic receptor in guinea pig right atria.More data for this Ligand-Target Pair
Affinity DataKd: 3.10nMAssay Description:Compound was evaluated for competitive antagonism of beta-1 adrenergic receptor in guinea pig atria measured as pA2 (-log KB)More data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:In vitro ability to block beta-1 adrenergic receptor in guinea pig right atria.More data for this Ligand-Target Pair
Affinity DataKd: 3.20nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 4.40nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:The compound was tested in vitro for its ability to block Beta-1 adrenergic receptor in guinea pig right atriaMore data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Beta-1 adrenergic receptor blocking activity in atria of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 5.40nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 5.5nMAssay Description:Antagonism of the isoprenaline-induced positive chronotropic effect on the atria of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 5.80nMAssay Description:Compound was evaluated for competitive antagonism of beta-1 adrenergic receptor in guinea pig atria measured as pA2 (-log KB)More data for this Ligand-Target Pair
Affinity DataKd: 6nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 6.20nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 6.30nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 8.5nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKd: 8.70nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
Affinity DataKd: 9.10nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 9.80nMAssay Description:Beta-1 adrenergic receptor blocking activity in atria of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Beta-1 adrenergic receptor blocking activity in atria of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:In vitro ability to block beta-1 adrenergic receptor in guinea pig right atria.More data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:The compound was tested in vitro for its ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair