Affinity DataKi: 18.4nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in diabetic human liver microsomes assessed as reduction in enzyme-mediated mycophenolic acid phenolic 7...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in diabetic human kidney microsomes assessed as reduction in enzyme-mediated mycophenolic acid phenolic ...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in non-diabetic human liver microsomes assessed as reduction in enzyme-mediated mycophenolic acid phenol...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in non-diabetic human kidney microsomes assessed as reduction in enzyme-mediated mycophenolic acid pheno...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in diabetic human kidney microsomes assessed as reduction in enzyme-mediated mycophenolic acid acyl gluc...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in non-diabetic human kidney microsomes assessed as reduction in enzyme-mediated mycophenolic acid acyl ...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in diabetic human liver microsomes assessed as reduction in enzyme-mediated mycophenolic acid acyl glucu...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in non-diabetic human liver microsomes assessed as reduction in enzyme-mediated mycophenolic acid acyl g...More data for this Ligand-Target Pair
Affinity DataKi: 1.01E+5nMAssay Description:Competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+5nMAssay Description:Competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+5nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in diabetic human kidney microsomes assessed as reduction in enzyme-mediated zidovudine glucuronide form...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+5nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in non-diabetic human kidney microsomes assessed as reduction in enzyme-mediated zidovudine glucuronide ...More data for this Ligand-Target Pair
Affinity DataKi: 1.62E+5nMAssay Description:Inhibition of recombinant human C-terminal His-tagged UGT2B7 after 15 to 60 mins by Michaelis-Menten equation analysis in presence of UDPGAMore data for this Ligand-Target Pair
Affinity DataKi: 1.92E+5nMAssay Description:Non competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+5nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in diabetic human liver microsomes assessed as reduction in enzyme-mediated zidovudine glucuronide forma...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+5nMAssay Description:Uncompetitive substrate inhibition of UGT2B7 in non-diabetic human liver microsomes assessed as reduction in enzyme-mediated zidovudine glucuronide f...More data for this Ligand-Target Pair
Affinity DataKi: 2.58E+5nMAssay Description:Non competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 3.01E+5nMAssay Description:Competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+5nMAssay Description:Drug metabolism assessed as recombinant human UGT2B7 assessed as O-glucuronidation measured as inhibition constant at 10 to 400 uM incubated for 60 m...More data for this Ligand-Target Pair
Affinity DataKi: 6.24E+5nMAssay Description:Non competitive inhibition of UGT2B7-catalyzed scopoletin glucuronidationMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+6nMAssay Description:Inhibition of AZT glucuronidation by human recombinant UGT2B7More data for this Ligand-Target Pair