TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.00370nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.00850nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.0150nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.0770nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.720nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.800nM ΔG°: -51.4kJ/mole IC50: 2.40nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Noncompetitive inhibition of Torpedo californica AChE using ATCh as substrate preincubated for 90 mins followed by substrate addition by potentiometr...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Competitive inhibition of Torpedo californica AChE using ATCh as substrate preincubated for 90 mins followed by substrate addition by potentiometric ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Tested for the ability to inhibit Acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Binding affinity tested against acetylcholinesterase in Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.5nM ΔG°: -47.2kJ/mole IC50: 16nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 17.5nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity tested against acetylcholinesterase in Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 37.6nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 175nM ΔG°: -38.2kJ/mole IC50: 414nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 175nM ΔG°: -38.6kJ/molepH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 190nM ΔG°: -39.0kJ/moleT: 2°CAssay Description:AChE and BChE inhibitory activities were measured in vitro by a modified spectrophotometric method. all the inhibition studies were performed using ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 230nM ΔG°: -38.5kJ/moleT: 2°CAssay Description:AChE and BChE inhibitory activities were measured in vitro by a modified spectrophotometric method. all the inhibition studies were performed using ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 334nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 334nM ΔG°: -37.0kJ/molepH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 700nM ΔG°: -35.1kJ/molepH: 7.5 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Compound was evaluated for the inhibition of acetylcholinesterase (AChE) in bovine brainMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Compound was evaluated for competitive inhibition constant of acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Compound was evaluated for competitive inhibition constant of acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 2.65E+3nMAssay Description:In vitro binding affinity was determined against acetylcholinesterase from torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 3.03E+3nMAssay Description:In vitro binding affinity was determined against acetylcholinesterase from torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Compound was evaluated for competitive inhibition constant of acetylcholinesterase (AChE) from Torpedo californicaMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition of Torpedo californica AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 4.10E+3nMAssay Description:In vitro binding affinity was determined against acetylcholinesterase from torpedo californicaMore data for this Ligand-Target Pair