Compile Data Set for Download or QSAR
maximum 50k data
Found 160 of ki data for polymerid = 49000250,49000251,49000255,49000256,50000525,50002638
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50019443(1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol ...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM81885(2-(3-tert-Butylamino-2-hydroxypropylthio)-4-(5-car...)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25764(ALPRENOLOL,(+) | ALPRENOLOL,(-) | Alfeprol | Alphe...)
Affinity DataKi:  0.580nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25768(1-[(7-methyl-2,3-dihydro-1H-inden-4-yl)oxy]-3-(pro...)
Affinity DataKi:  1.78nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM81886(CAS_3506-09-0 | CHEMBL287651 | PROPRANOLOL, dl)
Affinity DataKi:  2.45nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50240370(1-(2-(allyloxy)phenoxy)-3-(isopropylamino)propan-2...)
Affinity DataKi:  9.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM81882(CAS_93633-92-2 | YM-09538)
Affinity DataKi:  13.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  43.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000504(6-Isopropylamino-5,6,7,8-tetrahydro-naphthalene-1,...)
Affinity DataKi:  62nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-2 adrenergic receptor of bovine lungMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25758(2-hydroxy-5-{1-hydroxy-2-[(4-phenylbutan-2-yl)amin...)
Affinity DataKi:  67.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKi:  110nMAssay Description:Tested for binding affinity against beta-2 adrenergic receptor in bovine lung using [3H]DHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKi:  110nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards beta-2 receptor of bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50000503(6-Amino-5,6,7,8-tetrahydro-naphthalene-1,2,5-triol...)
Affinity DataKi:  120nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards beta-2 receptor of bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036835(1-(3,4-Dichloro-phenyl)-2-isopropylamino-ethanol |...)
Affinity DataKi:  140nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50010555(6-[3-(4-Acetylamino-phenoxy)-2-hydroxy-propylamino...)
Affinity DataKi:  146nMAssay Description:Ki value was determined by accumulation of c-AMP in S-49 mouse lymphoma cells (Beta2).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25762(CHEMBL471 | N-{4-[1-hydroxy-2-(propan-2-ylamino)et...)
Affinity DataKi:  339nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM85190(CAS_3055171 | NAD-299 | NSC_3055171)
Affinity DataKi:  340nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50010562(6-[3-(4-Acetylamino-phenoxy)-2-hydroxy-propylamino...)
Affinity DataKi:  390nMAssay Description:Ki value was determined by accumulation of c-AMP in S-49 mouse lymphoma cells (Beta2).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM81887(Butoxamine | CAS_1937-89-9)
Affinity DataKi:  468nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50042999(3,6-Difluoro-4-(1-hydroxy-2-methylamino-ethyl)-ben...)
Affinity DataKi:  710nMAssay Description:Binding affinity against adrenergic beta 2 receptor versus 1 nM [3H]dihydroalprenolol in rat cerebral cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50029050((-)-(R)-epinephrine | (-)-3,4-dihydroxy-alpha-((me...)
Affinity DataKi:  720nMAssay Description:Binding affinity against adrenergic beta 2 receptor versus 1 nM [3H]dihydroalprenolol in rat cerebral cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50010564(6-[3-(4-Acetylamino-phenoxy)-2-hydroxy-propylamino...)
Affinity DataKi:  810nMAssay Description:Ki value was determined by accumulation of c-AMP in S-49 mouse lymphoma cells (Beta2).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036842(3-tert-Butylamino-2-hydroxy-propionaldehyde O-prop...)
Affinity DataKi:  850nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50022784((R)-N-methyl-3-phenyl-3-(o-tolyloxy)propan-1-amine...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM86708(CAS_146714-97-8 | CHEMBL31354 | CHEMBL514874 | CHE...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50094670(1-(4-Dipropylamino-1,3,4,5-tetrahydro-benzo[cd]ind...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50010565(6-[3-(4-Acetylamino-phenoxy)-2-hydroxy-propylamino...)
Affinity DataKi:  1.18E+3nMAssay Description:Ki value was determined by accumulation of c-AMP in S-49 mouse lymphoma cells (Beta2).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036840(CHEMBL38033 | Propionaldehyde O-(3-tert-butylamino...)
Affinity DataKi:  1.26E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036841(3-tert-Butylamino-2-hydroxy-propionaldehyde O-ethy...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50019060((+/-)4-(2-Amino-1-hydroxy-ethyl)-3-fluoro-benzene-...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity against adrenergic beta 2 receptor versus 1 nM [3H]dihydroalprenolol in rat cerebral cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25756((2R,3R)-2,3-dihydroxysuccinic acid;1-(isopropylami...)
Affinity DataKi:  1.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036838(Acetaldehyde O-(3-tert-butylamino-2-hydroxy-propyl...)
Affinity DataKi:  1.98E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25752(Betaxolol | Levobetaxolol | [(2S)-3-{4-[2-(cyclopr...)
Affinity DataKi:  2.04E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50010553(6-[3-(4-Acetylamino-phenoxy)-2-hydroxy-propylamino...)
Affinity DataKi:  2.17E+3nMAssay Description:Ki value was determined by accumulation of c-AMP in S-49 mouse lymphoma cells (Beta2).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM81881(l-Metoprolol)
Affinity DataKi:  2.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50333880(CHEMBL1614664 | Hypericin | Pseudohypericin)
Affinity DataKi:  2.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM25753(2-{4-[2-hydroxy-3-(propan-2-ylamino)propoxy]phenyl...)
Affinity DataKi:  2.82E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50010550(6-[3-(4-Acetylamino-phenoxy)-2-hydroxy-propylamino...)
Affinity DataKi:  2.85E+3nMAssay Description:Ki value was determined by accumulation of c-AMP in S-49 mouse lymphoma cells (Beta2).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  2.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036839(2-Hydroxy-3-isopropylamino-propionaldehyde O-ethyl...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50029051((-)-arterenol | (-)-noradrenaline | (-)-norepineph...)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity against adrenergic beta 2 receptor versus 1 nM [3H]dihydroalprenolol in rat cerebral cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036836(CHEMBL38114 | Propionaldehyde O-(2-hydroxy-3-isopr...)
Affinity DataKi:  4.58E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50041915(1-(Isopropylamino-methyl)-isochroman-6,7-diol | CH...)
Affinity DataKi:  4.90E+3nMAssay Description:Tested for binding affinity against beta-2 adrenergic receptor in bovine lung using [3H]DHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College Of Pharmacy

Curated by PDSP Ki Database
LigandPNGBDBM50042998(5-(2-Amino-1-hydroxy-ethyl)-3-fluoro-benzene-1,2-d...)
Affinity DataKi:  5.50E+3nMAssay Description:Binding affinity against adrenergic beta 2 receptor versus 1 nM [3H]dihydroalprenolol in rat cerebral cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50036837(2-Hydroxy-3-isopropylamino-propionaldehyde O-propy...)
Affinity DataKi:  5.60E+3nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(BOVINE)
Universit£

Curated by ChEMBL
LigandPNGBDBM50029051((-)-arterenol | (-)-noradrenaline | (-)-norepineph...)
Affinity DataKi:  6.00E+3nMAssay Description:Tested for binding affinity against beta-2 adrenergic receptor in bovine lung using [3H]DHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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