Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibitory activity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Inhibitory activity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.40E+4nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.60E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.10E+4nMAssay Description:Tested for inhibitory activity of the compound against gamma-aminobutyric acid aminotransferase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMAssay Description:Reversible inhibition of pig brain GABA-AT using GABA as substrateMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.20E+4nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.30E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.90E+4nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.90E+5nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.90E+5nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.95E+5nMpH: 8.5Assay Description:Compound was tested for inhibitory constant of Gamma-amino-N-butyrate transaminase in pig brain at pH of 8.5 and 25 degree CMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.00E+5nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.30E+5nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.00E+5nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.00E+6nMAssay Description:Binding affinity against Gamma-amino-N-butyrate transaminase in pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.20E+6nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.30E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.35E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.40E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.59E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.60E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 1.64E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.00E+6nMpH: 6.5Assay Description:Compound was tested for inhibitory constant of Gamma-amino-N-butyrate transaminase in pig brain at pH of 6.5More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.14E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.27E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.40E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.49E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.70E+6nMAssay Description:Compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase (GABA-AT)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.80E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 2.86E+6nMAssay Description:Competitive inhibition of pig GABA aminotransferase using alpha-ketoglutarate as substrate by SSADH-coupled assayMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.14E+6nMAssay Description:Compound was evaluated for the kinetic constant for the inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.20E+6nMAssay Description:Tested for inhibitory activity of the compound against gamma-aminobutyric acid aminotransferase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 3.60E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.11E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.20E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.20E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 4.70E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.70E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 5.90E+6nMAssay Description:Compound was evaluated for the competitive inhibition of of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.01E+6nMAssay Description:Binding affinity pig brain GABA-AT assessed as inactivation constant using GABA as substrate in presence of NADP+ and alpha-ketoglutarate by SSDH cou...More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.30E+6nMAssay Description:Competitive inhibition of pig brain GABA aminotransferase by Dixon/Cornish-Bowden plot analysis in presence of GABAMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.30E+6nMAssay Description:The compound was tested for the inhibition of Gamma-amino-N-butyrate transaminase from pig brainMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.50E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 6.80E+6nMAssay Description:Apparent dissociation constants for inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Sus scrofa)
Northwestern University
Curated by ChEMBL
Northwestern University
Curated by ChEMBL
Affinity DataKi: 7.74E+6nMAssay Description:Inhibition of pig brain GABA-AT in presence of beta-mercaptoethanolMore data for this Ligand-Target Pair