Compile Data Set for Download or QSAR
maximum 50k data
Found 151 of ki data for polymerid = 50000613
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060055(4-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060016(4-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  22nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060047(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-(4-phen...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060022(4-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  28nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060029(3-[(R)-3-(4-Acetyl-piperazin-1-yl)-2-(naphthalene-...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060026(3-[3-(4-Butyryl-piperazin-1-yl)-2-(naphthalene-2-s...)
Affinity DataKi:  49nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060041(3-[3-(4-Hexanoyl-piperazin-1-yl)-2-(naphthalene-2-...)
Affinity DataKi:  64nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060017(3-[(R)-3-(4-Methanesulfonyl-piperazin-1-yl)-2-(nap...)
Affinity DataKi:  67nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060021(3-[3-(4-Cyclohexanecarbonyl-piperazin-1-yl)-2-(nap...)
Affinity DataKi:  72nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060023(3-[(R)-3-(4-Formyl-piperazin-1-yl)-2-(naphthalene-...)
Affinity DataKi:  73nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50080479(CHEMBL117156 | N-(3-Carbamimidoyl-benzyl)-2-(napht...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against bovine pancreatic trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060035(4-[(R)-3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2...)
Affinity DataKi:  97nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082194(4-[3-(3-Carbamimidoyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  110nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)
Affinity DataKi:  120nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060051(3-[3-(4-Acetyl-piperazin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060018(3-[3-(4-Benzoyl-piperazin-1-yl)-2-(naphthalene-2-s...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060033(3-[3-(4-Methyl-piperidin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  140nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060027(3-[2-(4-tert-Butyl-benzenesulfonylamino)-3-(4-meth...)
Affinity DataKi:  160nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060056(4-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060044(3-[3-[4-(Butane-1-sulfonyl)-piperazin-1-yl]-2-(nap...)
Affinity DataKi:  180nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060042(3-[3-[4-(Naphthalene-2-carbonyl)-piperazin-1-yl]-2...)
Affinity DataKi:  190nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060037(3-[3-(4-Ethanesulfonyl-piperazin-1-yl)-2-(naphthal...)
Affinity DataKi:  190nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060014(3-[3-(4-Methanesulfonyl-piperazin-1-yl)-2-(naphtha...)
Affinity DataKi:  190nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082175(3-[3-Morpholin-4-yl-2-(naphthalene-2-sulfonylamino...)
Affinity DataKi:  210nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060034(3-{2-(Naphthalene-2-sulfonylamino)-3-oxo-3-[4-(pro...)
Affinity DataKi:  210nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060053(4-[3-(3-Carbamimidoyl-phenyl)-2-(naphthalene-2-sul...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060043(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperaz...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060046(3-[(R)-2-[2-(7,7-Dimethyl-2-oxo-bicyclo[2.2.1]hept...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060025(3-{2-(Naphthalene-2-sulfonylamino)-3-oxo-3-[4-(tol...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060043(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperaz...)
Affinity DataKi:  220nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060054(3-[2-[2-(7,7-Dimethyl-2-oxo-bicyclo[2.2.1]hept-1-y...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060032(3-[3-(4-Formyl-piperazin-1-yl)-2-(naphthalene-2-su...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082193(3-[3-(4-Acetyl-piperazin-1-yl)-3-oxo-2-(2,4,6-trii...)
Affinity DataKi:  220nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082190(1-[3-(3-Carbamimidoyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  270nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060048(3-[3-(4-Methanesulfonyl-piperazin-1-yl)-2-(naphtha...)
Affinity DataKi:  320nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060019(3-[(R)-3-(4-Methanesulfonyl-piperazin-1-yl)-3-oxo-...)
Affinity DataKi:  320nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060049(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperid...)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060040(3-[3-(4-Benzenesulfonyl-piperazin-1-yl)-2-(naphtha...)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060049(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-piperid...)
Affinity DataKi:  330nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082174(1-[3-(3-Carbamimidoyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  360nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082192(1-[3-(3-Carbamimidoyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  360nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060057(3-{2-(Naphthalene-2-sulfonylamino)-3-[4-(naphthale...)
Affinity DataKi:  400nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082182(3-[2-(Naphthalene-2-sulfonylamino)-3-oxo-3-pyrroli...)
Affinity DataKi:  440nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060054(3-[2-[2-(7,7-Dimethyl-2-oxo-bicyclo[2.2.1]hept-1-y...)
Affinity DataKi:  440nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060031(3-[(R)-3-(4-Methyl-piperazin-1-yl)-2-(naphthalene-...)
Affinity DataKi:  470nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082183(3-[3-Morpholin-4-yl-3-oxo-2-(2,4,6-triisopropyl-be...)
Affinity DataKi:  490nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50082179(1-[3-(3-Carbamimidoyl-phenyl)-2-(2,4,6-triisopropy...)
Affinity DataKi:  500nMAssay Description:Tested for inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50080482(4-[(S)-3-(7-Methoxy-naphthalene-2-sulfonylamino)-2...)
Affinity DataKi:  500nMAssay Description:Inhibitory activity against bovine pancreatic trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM13279(4-{[(3S)-3-[(7-methoxynaphthalene-2-)(methyl)sulfo...)
Affinity DataKi:  530nMAssay Description:Inhibitory activity against bovine pancreatic trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnionic trypsin(Bos taurus)
Klinikum Der Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50060024(3-[(R)-3-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-2-(n...)
Affinity DataKi:  600nMAssay Description:Inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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