Found 180 Enz. Inhib. hit(s) with Target = 'Calcium/calmodulin-dependent protein kinase type II subunit gamma'
Affinity DataEC50: 7.40nMAssay Description:Inhibition of CaMK2gamma/delta in neonatal rat ventricular myocytes assessed as phospholamban phosphorylation after 4 hrs by Hoechst 33342 fluorescen...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 4.00E+4nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 7.80E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 690nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:The compound of Example 39, 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one, was subjected to a kinase...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:The compound of Example 39, 2-(1H-indol-5-ylamino)-6-(2,4-difluorophenylsulfonyl)-8-methylpyrido[2,3-d]pyrimidin-7(8H)-one, was subjected to a kinase...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 0.5nMAssay Description:Average Binding Constant for CAMK2G; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 470nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 690nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 26nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 26nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of CAMK2gamma (unknown origin) by Millipore kinase analysisMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 760nMAssay Description:Average Binding Constant for CAMK2G; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human CAMK2gamma using [KKLNRTLSFAEPG] as substrateMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 440nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CAMK1GMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 540nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 690nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: 7.80E+3nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit gamma(Homo sapiens (Human))
Macquarie University
Curated by ChEMBL
Macquarie University
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CAMK2G kinase domainMore data for this Ligand-Target Pair