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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Prokineticin 2 (PK2)'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Prokineticin 2 (PK2)


(Homo sapiens (Human))
BDBM121129
PNG
(A457 | US8722896, (+/-)-1-Benzyl-N-(9-chloro-3,4- ...)
Show SMILES CC(C)CN(Cc1cc(Cl)c2OCCCOc2c1)C(=O)C1CCN(Cc2ccccc2)C1
Show InChI InChI=1S/C26H33ClN2O3/c1-19(2)15-29(17-21-13-23(27)25-24(14-21)31-11-6-12-32-25)26(30)22-9-10-28(18-22)16-20-7-4-3-5-8-20/h3-5,7-8,13-14,19,22H,6,9-12,15-18H2,1-2H3
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 40n/a 7.80n/an/an/an/a



Central South University; Changsha Medical University



Assay Description
Briefly, Chinese hamster ovary cells stably expressing the photoprotein aequorin were transiently transfected with WT or respective mutant PKR2-expre...


J Biol Chem 289: 15518-26 (2014)


Article DOI: 10.1074/jbc.M114.556381
BindingDB Entry DOI: 10.7270/Q2H9943S
More data for this
Ligand-Target Pair