Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with Target = 'Toll-like receptor 3'
TargetToll-like receptor 3(Homo sapiens)
University Of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50239681(CHEMBL4074408)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at human TLR3 expressed in HEK293 cells assessed as induction of NF-kB activation-mediated SEAP production after 24 hrs by HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 3(Homo sapiens)
University Of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50239682(CHEMBL4105063)
Affinity DataEC50:  2.23E+4nMAssay Description:Agonist activity at human TLR3 expressed in HEK293 cells assessed as induction of NF-kB activation-mediated SEAP production after 24 hrs by HTS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 3(Homo sapiens)
University Of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50239680(CHEMBL4064228)
Affinity DataEC50:  4.25E+4nMAssay Description:Inhibitory activity against Herpes simplex virus type-I specific thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 3(Homo sapiens)
University Of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50563780(CHEMBL4795714)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human TLR3 stably expressed in HEK293 cells cotransfected with secreted alkaline phosphatase assessed as assessed as inhibition of poly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 3(Homo sapiens)
University Of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50543466(CHEMBL4647818)
Affinity DataIC50:  2.16E+3nMAssay Description:Antagonist activity at human TLR3 overexpressed in HEK-Blue cells assessed as inhibition of Poly IC-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 3(Homo sapiens)
University Of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM21958(2-(2,6-dimethylpyridin-4-yl)-3-isopropyl-5-(piperi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at Poly C stimulated human TRL3 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated w...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetToll-like receptor 3(Homo sapiens)
University Of Colorado Boulder

Curated by ChEMBL
LigandPNGBDBM50543465(CHEMBL4636498)
Affinity DataIC50:  5.44E+3nMAssay Description:Antagonist activity at human TLR3 overexpressed in HEK-Blue cells assessed as inhibition of Poly IC-induced NFkappaB and AP-1 activation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed