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Found 1187 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase Lyn'
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM50545405(CP-26,154 | CP-26154 | Mlr-1023 | Tolimidone)
Affinity DataEC50:  63nMAssay Description:Inhibition of Lyn (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340095((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340188((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340189((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340196((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340095((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme (Millipore catalog #14-510), is diluted to 250 mU/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340187((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme (Millipore catalog #14-510), is diluted to 250 mU/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340188((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme (Millipore catalog #14-510), is diluted to 250 mU/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340189((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme (Millipore catalog #14-510), is diluted to 250 mU/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340196((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme (Millipore catalog #14-510), is diluted to 250 mU/mL in KR buffer (10 mM Tris-HCl, 10 mM MgCl2, 0.01% Tween-20, 0.05% NaN3, 1 mM DTT, 2 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340187((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340188((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340189((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340196((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340095((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340095((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340187((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50:  550nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340184((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)piper...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340185((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340186((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340119(US10239883, Example 3 | US10934296, Example 3 | US...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340191((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)pyrro...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340192((S)-4-(8-amino-3-(1-(2- chloropyrimidine-4- carbon...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340193((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340194((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340195((S)-4-(8-amino-3-(1-but-2- ynoylpyrrolidin-2-yl)im...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340091(4-(8-amino-3-((S)-1-(2- chloropyrimidine-4- carbon...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340092((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)pyrro...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340093((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)pyrro...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340094((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)but-2- en...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340159((S)-4-(3-(1-acryloylpiperidin-2-yl)-8- aminoimidaz...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340160((S)-4-(3-(1-acryloylpyrrolidin-2-yl)- 8-aminoimida...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340161((S)-4-(8-amino-3-(1-but-2- ynoylpiperidin-2-yl)imi...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340162((S)-4-(8-amino-3-(1-but-2- ynoylpiperidin-2-yl)imi...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340163((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)but-2- en...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340164(4-(8-amino-3-((S)-1- (vinylsulfonyl)piperidin-2- y...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340165((S)-4-(8-amino-3-(1-but-2- ynoylpiperidin-2-yl)imi...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340068(4-(3-((S)-1-acryloylpiperidin-2-yl)-8- aminoimidaz...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340096((E)-4-(8-amino-3-((4-(dimethyl amino)but-2-enamido...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340097((S)-4-(8-amino-3-(1-(2-chloro pyrimidine-4-carbony...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340098((S)-4-(8-amino-3-(1-(2-chloro pyrimidine-4-carbony...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340069((S,E)-4-(8-amino-3-(1-(4- methoxybut-2-enoyl)piper...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340099((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)but-2- en...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340070((S)-4-(8-amino-3-(1-(2- chloropyrimidine-4- carbon...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340166((S,E)-4-(8-amino-3-(1-(4-methoxy- N-methylbut-2- e...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340167((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)-N-methyl...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340168((S,E)-4-(8-amino-3-(1-(4- (pyrrolidin-1-yl)but-2- ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340169((S,E)-4-(8-amino-3-(1-(4- (dimethylamino)but-2- en...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340170((S)-4-(8-amino-3-(1-(2- chloropyrimidine-4- carbon...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Melior Discovery

Curated by ChEMBL
LigandPNGBDBM340100((S)-4-(8-amino-3-(1-(2- chloropyrimidine-4- carbon...)
Affinity DataEC50: >1.00E+3nMAssay Description:Lyn enzyme activity is measured using the IMAP (immobilized metal ion affinity-based fluorescence polarization) assay as outlined below.Lyn enzyme (M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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