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Found 856 hits Enz. Inhib. hit(s) with Target = 'Angiotensin II receptor (AT-1) type-1'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213779
PNG
(CHEMBL313598)
Show SMILES CCCc1nc(SC)c(C(=O)C[S+]([O-])c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1cccs1
Show InChI InChI=1S/C34H34N4O5S4/c1-3-10-31-36-33(44-2)32(29(39)23-46(41)27-12-5-4-6-13-27)38(31)22-24-16-18-25(19-17-24)28-14-7-8-15-30(28)47(42,43)37-34(40)35-21-26-11-9-20-45-26/h4-9,11-20H,3,10,21-23H2,1-2H3,(H2,35,37,40)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213551
PNG
(CHEMBL90618)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)CCc1cccs1
Show InChI InChI=1S/C28H27F2N3O5S3/c1-2-6-23-31-26(40-28(29)30)25(27(35)36)33(23)17-18-10-12-19(13-11-18)21-8-3-4-9-22(21)41(37,38)32-24(34)15-14-20-7-5-16-39-20/h3-5,7-13,16,28H,2,6,14-15,17H2,1H3,(H,32,34)(H,35,36)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213687
PNG
(CHEMBL87244)
Show SMILES CCCc1nc(SC)c(C(=O)C[S+]([O-])c2ccc(C)cc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C37H38N4O5S3/c1-4-10-34-39-36(47-3)35(32(42)25-48(44)30-21-15-26(2)16-22-30)41(34)24-28-17-19-29(20-18-28)31-13-8-9-14-33(31)49(45,46)40-37(43)38-23-27-11-6-5-7-12-27/h5-9,11-22H,4,10,23-25H2,1-3H3,(H2,38,40,43)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213695
PNG
(CHEMBL89032)
Show SMILES CCCCc1nc(SC)c(C(=O)C[S+]([O-])c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C37H38N4O5S3/c1-3-4-19-34-39-36(47-2)35(32(42)26-48(44)30-15-9-6-10-16-30)41(34)25-28-20-22-29(23-21-28)31-17-11-12-18-33(31)49(45,46)40-37(43)38-24-27-13-7-5-8-14-27/h5-18,20-23H,3-4,19,24-26H2,1-2H3,(H2,38,40,43)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213592
PNG
(CHEMBL315236)
Show SMILES CCCCc1nc(SC)c(C(=O)CS(=O)(=O)c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C37H38N4O6S3/c1-3-4-19-34-39-36(48-2)35(32(42)26-49(44,45)30-15-9-6-10-16-30)41(34)25-28-20-22-29(23-21-28)31-17-11-12-18-33(31)50(46,47)40-37(43)38-24-27-13-7-5-8-14-27/h5-18,20-23H,3-4,19,24-26H2,1-2H3,(H2,38,40,43)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213685
PNG
(CHEMBL431853)
Show SMILES CCCCc1nc(SC)c(C(=O)CS(=O)(=O)c2ccc(F)cc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C37H37FN4O6S3/c1-3-4-14-34-40-36(49-2)35(32(43)25-50(45,46)30-21-19-29(38)20-22-30)42(34)24-27-15-17-28(18-16-27)31-12-8-9-13-33(31)51(47,48)41-37(44)39-23-26-10-6-5-7-11-26/h5-13,15-22H,3-4,14,23-25H2,1-2H3,(H2,39,41,44)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213505
PNG
(CHEMBL314975)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)CC1CCCCC1
Show InChI InChI=1S/C29H33F2N3O5S2/c1-2-8-24-32-27(40-29(30)31)26(28(36)37)34(24)18-20-13-15-21(16-14-20)22-11-6-7-12-23(22)41(38,39)33-25(35)17-19-9-4-3-5-10-19/h6-7,11-16,19,29H,2-5,8-10,17-18H2,1H3,(H,33,35)(H,36,37)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213687
PNG
(CHEMBL87244)
Show SMILES CCCc1nc(SC)c(C(=O)C[S+]([O-])c2ccc(C)cc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C37H38N4O5S3/c1-4-10-34-39-36(47-3)35(32(42)25-48(44)30-21-15-26(2)16-22-30)41(34)24-28-17-19-29(20-18-28)31-13-8-9-14-33(31)49(45,46)40-37(43)38-23-27-11-6-5-7-12-27/h5-9,11-22H,4,10,23-25H2,1-3H3,(H2,38,40,43)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213561
PNG
(CHEMBL312937)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)Cc1cccs1
Show InChI InChI=1S/C27H25F2N3O5S3/c1-2-6-22-30-25(39-27(28)29)24(26(34)35)32(22)16-17-10-12-18(13-11-17)20-8-3-4-9-21(20)40(36,37)31-23(33)15-19-7-5-14-38-19/h3-5,7-14,27H,2,6,15-16H2,1H3,(H,31,33)(H,34,35)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213697
PNG
(CHEMBL84908)
Show SMILES CCc1nc(SC)c(C(=O)C[S+]([O-])c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C35H34N4O5S3/c1-3-32-37-34(45-2)33(30(40)24-46(42)28-14-8-5-9-15-28)39(32)23-26-18-20-27(21-19-26)29-16-10-11-17-31(29)47(43,44)38-35(41)36-22-25-12-6-4-7-13-25/h4-21H,3,22-24H2,1-2H3,(H2,36,38,41)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213688
PNG
(CHEMBL86538)
Show SMILES CCCc1nc(SC)c(C(C)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C30H32N4O4S2/c1-4-10-27-32-29(39-3)28(21(2)35)34(27)20-23-15-17-24(18-16-23)25-13-8-9-14-26(25)40(37,38)33-30(36)31-19-22-11-6-5-7-12-22/h5-9,11-18H,4,10,19-20H2,1-3H3,(H2,31,33,36)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213782
PNG
(CHEMBL264304)
Show SMILES CCCc1nc(SC)c(C(=O)C[S+]([O-])c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C36H36N4O5S3/c1-3-12-33-38-35(46-2)34(31(41)25-47(43)29-15-8-5-9-16-29)40(33)24-27-19-21-28(22-20-27)30-17-10-11-18-32(30)48(44,45)39-36(42)37-23-26-13-6-4-7-14-26/h4-11,13-22H,3,12,23-25H2,1-2H3,(H2,37,39,42)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213593
PNG
(CHEMBL91046)
Show SMILES CCCCc1nc(SC)c(C(=O)CS(C)(=O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C32H36N4O6S3/c1-4-5-15-29-34-31(43-2)30(27(37)22-44(3,39)40)36(29)21-24-16-18-25(19-17-24)26-13-9-10-14-28(26)45(41,42)35-32(38)33-20-23-11-7-6-8-12-23/h6-14,16-19H,4-5,15,20-22H2,1-3H3,(H2,33,35,38)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213680
PNG
(CHEMBL87091)
Show SMILES CCCCc1nc(SC)c(C(=O)CC(=O)OCC)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C34H38N4O6S2/c1-4-6-16-30-36-33(45-3)32(28(39)21-31(40)44-5-2)38(30)23-25-17-19-26(20-18-25)27-14-10-11-15-29(27)46(42,43)37-34(41)35-22-24-12-8-7-9-13-24/h7-15,17-20H,4-6,16,21-23H2,1-3H3,(H2,35,37,41)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213681
PNG
(CHEMBL433010)
Show SMILES CCCc1nc(SC)c(C(=O)CS(=O)(=O)c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C36H36N4O6S3/c1-3-12-33-38-35(47-2)34(31(41)25-48(43,44)29-15-8-5-9-16-29)40(33)24-27-19-21-28(22-20-27)30-17-10-11-18-32(30)49(45,46)39-36(42)37-23-26-13-6-4-7-14-26/h4-11,13-22H,3,12,23-25H2,1-2H3,(H2,37,39,42)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213458
PNG
(CHEMBL90672)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)Cc1ccc(F)cc1
Show InChI InChI=1S/C29H26F3N3O5S2/c1-2-5-24-33-27(41-29(31)32)26(28(37)38)35(24)17-19-8-12-20(13-9-19)22-6-3-4-7-23(22)42(39,40)34-25(36)16-18-10-14-21(30)15-11-18/h3-4,6-15,29H,2,5,16-17H2,1H3,(H,34,36)(H,37,38)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213591
PNG
(CHEMBL84795)
Show SMILES CCCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C30H32N4O5S2/c1-3-4-14-26-32-28(40-2)27(29(35)36)34(26)20-22-15-17-23(18-16-22)24-12-8-9-13-25(24)41(38,39)33-30(37)31-19-21-10-6-5-7-11-21/h5-13,15-18H,3-4,14,19-20H2,1-2H3,(H,35,36)(H2,31,33,37)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213460
PNG
(CHEMBL85081)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)Cc1ccc2ccccc2c1
Show InChI InChI=1S/C33H29F2N3O5S2/c1-2-7-28-36-31(44-33(34)35)30(32(40)41)38(28)20-21-12-16-24(17-13-21)26-10-5-6-11-27(26)45(42,43)37-29(39)19-22-14-15-23-8-3-4-9-25(23)18-22/h3-6,8-18,33H,2,7,19-20H2,1H3,(H,37,39)(H,40,41)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213567
PNG
(CHEMBL315983)
Show SMILES CCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCC1CCCCC1
Show InChI InChI=1S/C29H36N4O5S2/c1-3-9-25-31-27(39-2)26(28(34)35)33(25)19-21-14-16-22(17-15-21)23-12-7-8-13-24(23)40(37,38)32-29(36)30-18-20-10-5-4-6-11-20/h7-8,12-17,20H,3-6,9-11,18-19H2,1-2H3,(H,34,35)(H2,30,32,36)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213552
PNG
(CHEMBL328302)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)CCc1ccccc1
Show InChI InChI=1S/C30H29F2N3O5S2/c1-2-8-25-33-28(41-30(31)32)27(29(37)38)35(25)19-21-13-16-22(17-14-21)23-11-6-7-12-24(23)42(39,40)34-26(36)18-15-20-9-4-3-5-10-20/h3-7,9-14,16-17,30H,2,8,15,18-19H2,1H3,(H,34,36)(H,37,38)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213456
PNG
(CHEMBL315000)
Show SMILES CCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCC1CCCC1
Show InChI InChI=1S/C28H34N4O5S2/c1-3-8-24-30-26(38-2)25(27(33)34)32(24)18-20-13-15-21(16-14-20)22-11-6-7-12-23(22)39(36,37)31-28(35)29-17-19-9-4-5-10-19/h6-7,11-16,19H,3-5,8-10,17-18H2,1-2H3,(H,33,34)(H2,29,31,35)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213500
PNG
(CHEMBL86337)
Show SMILES CCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1cccs1
Show InChI InChI=1S/C27H28N4O5S3/c1-3-7-23-29-25(37-2)24(26(32)33)31(23)17-18-11-13-19(14-12-18)21-9-4-5-10-22(21)39(35,36)30-27(34)28-16-20-8-6-15-38-20/h4-6,8-15H,3,7,16-17H2,1-2H3,(H,32,33)(H2,28,30,34)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213457
PNG
(CHEMBL84686)
Show SMILES CCCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCC1CCCCC1
Show InChI InChI=1S/C30H38N4O5S2/c1-3-4-14-26-32-28(40-2)27(29(35)36)34(26)20-22-15-17-23(18-16-22)24-12-8-9-13-25(24)41(38,39)33-30(37)31-19-21-10-6-5-7-11-21/h8-9,12-13,15-18,21H,3-7,10-11,14,19-20H2,1-2H3,(H,35,36)(H2,31,33,37)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213504
PNG
(CHEMBL89369)
Show SMILES CCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C28H28N4O5S2/c1-3-24-30-26(38-2)25(27(33)34)32(24)18-20-13-15-21(16-14-20)22-11-7-8-12-23(22)39(36,37)31-28(35)29-17-19-9-5-4-6-10-19/h4-16H,3,17-18H2,1-2H3,(H,33,34)(H2,29,31,35)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213783
PNG
(CHEMBL328985)
Show SMILES CCCc1nc(SC)c(C(=O)CS(=O)(=O)c2ccc(OC)cc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C37H38N4O7S3/c1-4-10-34-39-36(49-3)35(32(42)25-50(44,45)30-21-19-29(48-2)20-22-30)41(34)24-27-15-17-28(18-16-27)31-13-8-9-14-33(31)51(46,47)40-37(43)38-23-26-11-6-5-7-12-26/h5-9,11-22H,4,10,23-25H2,1-3H3,(H2,38,40,43)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213591
PNG
(CHEMBL84795)
Show SMILES CCCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C30H32N4O5S2/c1-3-4-14-26-32-28(40-2)27(29(35)36)34(26)20-22-15-17-23(18-16-22)24-12-8-9-13-25(24)41(38,39)33-30(37)31-19-21-10-6-5-7-11-21/h5-13,15-18H,3-4,14,19-20H2,1-2H3,(H,35,36)(H2,31,33,37)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283305
PNG
(3'-Fluoro-4'-[6-(3-isopropyl-ureido)-4-oxo-2-propy...)
Show SMILES CCCc1nc2ccc(NC(=O)NC(C)C)cc2c(=O)n1Cc1ccc(cc1F)-c1ccccc1S(=O)(=O)NC(=O)c1ccc(CC)cc1F
Show InChI InChI=1S/C37H37F2N5O5S/c1-5-9-34-42-32-17-15-26(41-37(47)40-22(3)4)20-29(32)36(46)44(34)21-25-14-13-24(19-30(25)38)27-10-7-8-11-33(27)50(48,49)43-35(45)28-16-12-23(6-2)18-31(28)39/h7-8,10-20,22H,5-6,9,21H2,1-4H3,(H,43,45)(H2,40,41,47)
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n/an/a 0.110n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283317
PNG
(2-Propyl-3-(3-fluoro-2'-(3-methylbutyloxycarbonyla...)
Show SMILES CCCc1nc2ccc(NC(=O)N3CCOCC3)cc2c(=O)n1Cc1ccc(cc1F)-c1ccccc1S(=O)(=O)NC(=O)OCCC(C)C
Show InChI InChI=1S/C35H40FN5O7S/c1-4-7-32-38-30-13-12-26(37-34(43)40-15-18-47-19-16-40)21-28(30)33(42)41(32)22-25-11-10-24(20-29(25)36)27-8-5-6-9-31(27)49(45,46)39-35(44)48-17-14-23(2)3/h5-6,8-13,20-21,23H,4,7,14-19,22H2,1-3H3,(H,37,43)(H,39,44)
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n/an/a 0.130n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283312
PNG
(4'-[2-Ethyl-6-(3-isopropyl-ureido)-4-oxo-4H-quinaz...)
Show SMILES CCc1ccc(C(=O)NS(=O)(=O)c2ccccc2-c2ccc(Cn3c(CC)nc4ccc(NC(=O)NC(C)C)cc4c3=O)c(F)c2)c(F)c1
Show InChI InChI=1S/C36H35F2N5O5S/c1-5-22-11-15-27(30(38)17-22)34(44)42-49(47,48)32-10-8-7-9-26(32)23-12-13-24(29(37)18-23)20-43-33(6-2)41-31-16-14-25(19-28(31)35(43)45)40-36(46)39-21(3)4/h7-19,21H,5-6,20H2,1-4H3,(H,42,44)(H2,39,40,46)
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n/an/a 0.140n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration of the compound against AT2 receptor of rat adrenal membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283300
PNG
(2-Butyl-3-(3-fluoro-2'-(3-methylbutyloxycarbonylam...)
Show SMILES CCCCc1nc2ccc(NC(=O)N(C)C(C)C)cc2c(=O)n1Cc1ccc(cc1F)-c1ccccc1S(=O)(=O)NC(=O)OCCC(C)C
Show InChI InChI=1S/C36H44FN5O6S/c1-7-8-13-33-39-31-17-16-27(38-35(44)41(6)24(4)5)21-29(31)34(43)42(33)22-26-15-14-25(20-30(26)37)28-11-9-10-12-32(28)49(46,47)40-36(45)48-19-18-23(2)3/h9-12,14-17,20-21,23-24H,7-8,13,18-19,22H2,1-6H3,(H,38,44)(H,40,45)
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n/an/a 0.140n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283310
PNG
(4'-[2-Ethyl-6-(3-isopropyl-3-methyl-ureido)-4-oxo-...)
Show SMILES CCc1ccc(cc1)C(=O)NS(=O)(=O)c1ccccc1-c1ccc(Cn2c(CC)nc3ccc(NC(=O)N(C)C(C)C)cc3c2=O)c(F)c1
Show InChI InChI=1S/C37H38FN5O5S/c1-6-24-12-14-25(15-13-24)35(44)41-49(47,48)33-11-9-8-10-29(33)26-16-17-27(31(38)20-26)22-43-34(7-2)40-32-19-18-28(21-30(32)36(43)45)39-37(46)42(5)23(3)4/h8-21,23H,6-7,22H2,1-5H3,(H,39,46)(H,41,44)
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TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213499
PNG
(CHEMBL88653)
Show SMILES CCCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)Cc1ccccc1
Show InChI InChI=1S/C30H29F2N3O5S2/c1-2-3-13-25-33-28(41-30(31)32)27(29(37)38)35(25)19-21-14-16-22(17-15-21)23-11-7-8-12-24(23)42(39,40)34-26(36)18-20-9-5-4-6-10-20/h4-12,14-17,30H,2-3,13,18-19H2,1H3,(H,34,36)(H,37,38)
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n/an/a 0.150n/an/an/an/an/an/a


TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II AT1B


(RAT)
BDBM50282363
PNG
(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Show SMILES CCCCc1ncc(\C=C(/Cc2cccs2)C(O)=O)n1Cc1ccc(C(O)=O)c(Cl)c1Cl
Show InChI InChI=1S/C23H22Cl2N2O4S/c1-2-3-6-19-26-12-16(10-15(22(28)29)11-17-5-4-9-32-17)27(19)13-14-7-8-18(23(30)31)21(25)20(14)24/h4-5,7-10,12H,2-3,6,11,13H2,1H3,(H,28,29)(H,30,31)/b15-10+
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n/an/a 0.160n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50


Bioorg Med Chem Lett 4: 23-28 (1994)


Article DOI: 10.1016/S0960-894X(01)81116-1
BindingDB Entry DOI: 10.7270/Q29G5MRF
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283316
PNG
(3'-Fluoro-4'-[6-(3-isopropyl-ureido)-4-oxo-2-propy...)
Show SMILES CCCc1nc2ccc(NC(=O)NC(C)C)cc2c(=O)n1Cc1ccc(cc1F)-c1ccccc1S(=O)(=O)NC(=O)COCC(C)C
Show InChI InChI=1S/C34H40FN5O6S/c1-6-9-31-38-29-15-14-25(37-34(43)36-22(4)5)17-27(29)33(42)40(31)18-24-13-12-23(16-28(24)35)26-10-7-8-11-30(26)47(44,45)39-32(41)20-46-19-21(2)3/h7-8,10-17,21-22H,6,9,18-20H2,1-5H3,(H,39,41)(H2,36,37,43)
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n/an/a 0.170n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213550
PNG
(CHEMBL87847)
Show SMILES CCCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)CC1CCCCC1
Show InChI InChI=1S/C30H35F2N3O5S2/c1-2-3-13-25-33-28(41-30(31)32)27(29(37)38)35(25)19-21-14-16-22(17-15-21)23-11-7-8-12-24(23)42(39,40)34-26(36)18-20-9-5-4-6-10-20/h7-8,11-12,14-17,20,30H,2-6,9-10,13,18-19H2,1H3,(H,34,36)(H,37,38)
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n/an/a 0.200n/an/an/an/an/an/a


TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213557
PNG
(CHEMBL309602)
Show SMILES CCCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCC
Show InChI InChI=1S/C25H30N4O5S2/c1-4-6-11-21-27-23(35-3)22(24(30)31)29(21)16-17-12-14-18(15-13-17)19-9-7-8-10-20(19)36(33,34)28-25(32)26-5-2/h7-10,12-15H,4-6,11,16H2,1-3H3,(H,30,31)(H2,26,28,32)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213554
PNG
(CHEMBL314527)
Show SMILES CCCc1nc(SC)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C29H30N4O5S2/c1-3-9-25-31-27(39-2)26(28(34)35)33(25)19-21-14-16-22(17-15-21)23-12-7-8-13-24(23)40(37,38)32-29(36)30-18-20-10-5-4-6-11-20/h4-8,10-17H,3,9,18-19H2,1-2H3,(H,34,35)(H2,30,32,36)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213564
PNG
(CHEMBL316234)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)Cc1ccccc1
Show InChI InChI=1S/C29H27F2N3O5S2/c1-2-8-24-32-27(40-29(30)31)26(28(36)37)34(24)18-20-13-15-21(16-14-20)22-11-6-7-12-23(22)41(38,39)33-25(35)17-19-9-4-3-5-10-19/h3-7,9-16,29H,2,8,17-18H2,1H3,(H,33,35)(H,36,37)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213679
PNG
(5-Beta-Ketosulfoxide Imidazolyl Biphenyl Sulfonylu...)
Show SMILES CCCc1nc(SC)c(C(=O)CSc2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C36H36N4O4S3/c1-3-12-33-38-35(45-2)34(31(41)25-46-29-15-8-5-9-16-29)40(33)24-27-19-21-28(22-20-27)30-17-10-11-18-32(30)47(43,44)39-36(42)37-23-26-13-6-4-7-14-26/h4-11,13-22H,3,12,23-25H2,1-2H3,(H2,37,39,42)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213569
PNG
(CHEMBL78866)
Show SMILES CCCCNC(=O)NS(=O)(=O)c1ccccc1-c1ccc(Cn2c(CCCC)nc(SC)c2C(O)=O)cc1
Show InChI InChI=1S/C27H34N4O5S2/c1-4-6-12-23-29-25(37-3)24(26(32)33)31(23)18-19-13-15-20(16-14-19)21-10-8-9-11-22(21)38(35,36)30-27(34)28-17-7-5-2/h8-11,13-16H,4-7,12,17-18H2,1-3H3,(H,32,33)(H2,28,30,34)
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n/an/a 0.200n/an/an/an/an/an/a


TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50285769
PNG
(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Show SMILES CCCCc1nc(SC)c(C(=O)n2cnnn2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C31H32N8O4S2/c1-3-4-14-27-34-29(44-2)28(30(40)39-21-33-36-37-39)38(27)20-23-15-17-24(18-16-23)25-12-8-9-13-26(25)45(42,43)35-31(41)32-19-22-10-6-5-7-11-22/h5-13,15-18,21H,3-4,14,19-20H2,1-2H3,(H2,32,35,41)
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n/an/a 0.200n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.


Bioorg Med Chem Lett 5: 2611-2616 (1995)


Article DOI: 10.1016/0960-894X(95)00479-D
BindingDB Entry DOI: 10.7270/Q2GT5N57
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50285760
PNG
(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Show SMILES CCCCc1nc(SC)c(C(O)CC(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C32H36N4O6S2/c1-3-4-14-28-34-31(43-2)30(26(37)19-29(38)39)36(28)21-23-15-17-24(18-16-23)25-12-8-9-13-27(25)44(41,42)35-32(40)33-20-22-10-6-5-7-11-22/h5-13,15-18,26,37H,3-4,14,19-21H2,1-2H3,(H,38,39)(H2,33,35,40)
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n/an/a 0.200n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.


Bioorg Med Chem Lett 5: 2611-2616 (1995)


Article DOI: 10.1016/0960-894X(95)00479-D
BindingDB Entry DOI: 10.7270/Q2GT5N57
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213781
PNG
(CHEMBL327927)
Show SMILES CCCCc1nc(SC)c(C(=O)CC(=O)c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C38H38N4O5S2/c1-3-4-19-35-40-37(48-2)36(33(44)24-32(43)30-15-9-6-10-16-30)42(35)26-28-20-22-29(23-21-28)31-17-11-12-18-34(31)49(46,47)41-38(45)39-25-27-13-7-5-8-14-27/h5-18,20-23H,3-4,19,24-26H2,1-2H3,(H2,39,41,45)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50285761
PNG
(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Show SMILES CCCCc1nc(SC)c(C(=O)C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCc1ccccc1
Show InChI InChI=1S/C31H32N4O6S2/c1-3-4-14-26-33-29(42-2)27(28(36)30(37)38)35(26)20-22-15-17-23(18-16-22)24-12-8-9-13-25(24)43(40,41)34-31(39)32-19-21-10-6-5-7-11-21/h5-13,15-18H,3-4,14,19-20H2,1-2H3,(H,37,38)(H2,32,34,39)
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n/an/a 0.200n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.


Bioorg Med Chem Lett 5: 2611-2616 (1995)


Article DOI: 10.1016/0960-894X(95)00479-D
BindingDB Entry DOI: 10.7270/Q2GT5N57
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283319
PNG
(2-Butyl-3-(3-fluoro-2'-(2-cyclopropylethyloxycarbo...)
Show SMILES CCCCc1nc2ccc(NC(=O)N(C)C(C)C)cc2c(=O)n1Cc1ccc(cc1F)-c1ccccc1S(=O)(=O)NC(=O)OCCC1CC1
Show InChI InChI=1S/C36H42FN5O6S/c1-5-6-11-33-39-31-17-16-27(38-35(44)41(4)23(2)3)21-29(31)34(43)42(33)22-26-15-14-25(20-30(26)37)28-9-7-8-10-32(28)49(46,47)40-36(45)48-19-18-24-12-13-24/h7-10,14-17,20-21,23-24H,5-6,11-13,18-19,22H2,1-4H3,(H,38,44)(H,40,45)
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n/an/a 0.230n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283318
PNG
(2-Butyl-3-(3-fluoro-2'-(butyloxycarbonylaminosulph...)
Show SMILES CCCCOC(=O)NS(=O)(=O)c1ccccc1-c1ccc(Cn2c(CCCC)nc3ccc(NC(=O)N(C)C(C)C)cc3c2=O)c(F)c1
Show InChI InChI=1S/C35H42FN5O6S/c1-6-8-14-32-38-30-18-17-26(37-34(43)40(5)23(3)4)21-28(30)33(42)41(32)22-25-16-15-24(20-29(25)36)27-12-10-11-13-31(27)48(45,46)39-35(44)47-19-9-7-2/h10-13,15-18,20-21,23H,6-9,14,19,22H2,1-5H3,(H,37,43)(H,39,44)
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n/an/a 0.25n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213778
PNG
(CHEMBL312990)
Show SMILES CCCc1nc(SC)c(C(=O)C[S+]([O-])c2ccccc2)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)NCC1CCCCC1
Show InChI InChI=1S/C36H42N4O5S3/c1-3-12-33-38-35(46-2)34(31(41)25-47(43)29-15-8-5-9-16-29)40(33)24-27-19-21-28(22-20-27)30-17-10-11-18-32(30)48(44,45)39-36(42)37-23-26-13-6-4-7-14-26/h5,8-11,15-22,26H,3-4,6-7,12-14,23-25H2,1-2H3,(H2,37,39,42)
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TBA

Assay Description
Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50283302
PNG
(2-ethyl-3-(3-fluoro-2'-(3-methyl-butyloxycarbonyla...)
Show SMILES CCc1nc2ccc(NC(=O)N(C)C(C)C)cc2c(=O)n1Cc1ccc(cc1F)-c1ccccc1S(=O)(=O)NC(=O)OCCC(C)C
Show InChI InChI=1S/C34H40FN5O6S/c1-7-31-37-29-15-14-25(36-33(42)39(6)22(4)5)19-27(29)32(41)40(31)20-24-13-12-23(18-28(24)35)26-10-8-9-11-30(26)47(44,45)38-34(43)46-17-16-21(2)3/h8-15,18-19,21-22H,7,16-17,20H2,1-6H3,(H,36,42)(H,38,43)
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n/an/a 0.300n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membrane


Bioorg Med Chem Lett 4: 2337-2342 (1994)


Article DOI: 10.1016/0960-894X(94)85036-4
BindingDB Entry DOI: 10.7270/Q2X066Z9
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213461
PNG
(CHEMBL407824)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)Cc1ccc2OCOc2c1
Show InChI InChI=1S/C30H27F2N3O7S2/c1-2-5-25-33-28(43-30(31)32)27(29(37)38)35(25)16-18-8-11-20(12-9-18)21-6-3-4-7-24(21)44(39,40)34-26(36)15-19-10-13-22-23(14-19)42-17-41-22/h3-4,6-14,30H,2,5,15-17H2,1H3,(H,34,36)(H,37,38)
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n/an/a 0.300n/an/an/an/an/an/a


TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
Angiotensin II receptor (AT-1) type-1


(RAT)
BDBM50213562
PNG
(CHEMBL327455)
Show SMILES CCCc1nc(SC(F)F)c(C(O)=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)C(C)c1ccccc1
Show InChI InChI=1S/C30H29F2N3O5S2/c1-3-9-25-33-28(41-30(31)32)26(29(37)38)35(25)18-20-14-16-22(17-15-20)23-12-7-8-13-24(23)42(39,40)34-27(36)19(2)21-10-5-4-6-11-21/h4-8,10-17,19,30H,3,9,18H2,1-2H3,(H,34,36)(H,37,38)
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TBA

Assay Description
In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparation


Citation and Details
More data for this
Ligand-Target Pair
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