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Found 67 Enz. Inhib. hit(s) with Target = 'Carnitine O-palmitoyltransferase 1, muscle isoform'
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50:  30nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403029(CHEMBL2216792)
Affinity DataIC50:  40nMAssay Description:Inhibition of rat CPT1B expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403040(CHEMBL2216779)
Affinity DataIC50:  55nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403037(CHEMBL2216774)
Affinity DataIC50:  130nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403041(CHEMBL2216776)
Affinity DataIC50:  150nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403031(CHEMBL2216771)
Affinity DataIC50:  160nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50:  180nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403028(CHEMBL2216769)
Affinity DataIC50:  360nMAssay Description:Inhibition of CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260111(CHEBI:15531 | MALONYL-COENZYME A)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM80613(1-(2,3,4-Trimethoxy-benzyl)-piperazine | 1-(2,3,4-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of CPT1A in rat myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839(CHEMBL106227 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataIC50:  1.45E+3nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101594(CHEMBL80493 | [3-Carboxy-2-(decane-1-sulfonylamino...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403039(CHEMBL2216778)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101604(CHEMBL309568 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403038(CHEMBL2216777)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101589(CHEMBL77174 | [3-Carboxy-2-(nonylaminosulphonyl-am...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839(CHEMBL106227 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101591(CHEMBL308869 | R-[3-Carboxy-2-(undecane-1-sulfamoy...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101591(CHEMBL308869 | R-[3-Carboxy-2-(undecane-1-sulfamoy...)
Affinity DataIC50:  5.80E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403043(CHEMBL2216780)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101600(CHEMBL305897 | [3-Carboxy-2-(undecane-1-sulfamoyla...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101600(CHEMBL305897 | [3-Carboxy-2-(undecane-1-sulfamoyla...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101604(CHEMBL309568 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101598(CHEMBL307495 | [3-Carboxy-2-(dodecane-1-sulfonylam...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260115(CHEMBL4097976)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM61402((Z)-2-butenedioic acid;2-(2,2-dicyclohexylethyl)pi...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50118093((4-Hydroxy-phenyl)-oxo-acetic acid | CHEMBL129918)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of CPT1B in heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260105(CHEMBL1592481)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260109(CHEMBL4077250)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403033(CHEMBL1231507)
Affinity DataIC50:  2.17E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403034(CHEMBL2114397)
Affinity DataIC50:  2.73E+4nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260108(CHEMBL4082420)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122839(CHEMBL106227 | [3-Carboxy-2-(3-tetradecyl-ureido)-...)
Affinity DataIC50:  4.34E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260104(CHEMBL4081530)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122827(CHEMBL105330 | [3-Carboxy-2-(3-nonyl-ureido)-propy...)
Affinity DataIC50:  4.62E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403030(CHEMBL2216768)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50118093((4-Hydroxy-phenyl)-oxo-acetic acid | CHEMBL129918)
Affinity DataIC50:  6.03E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260105(CHEMBL1592481)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50122833((3-Carboxy-2-octyloxycarbonylamino-propyl)-trimeth...)
Affinity DataIC50:  8.01E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50101590(CHEMBL78921 | [3-Carboxy-2-(3-nonyl-ureido)-propyl...)
Affinity DataIC50:  8.32E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403032(CHEMBL2216785)
Affinity DataIC50:  8.53E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50260112(CHEMBL4068222)
Affinity DataIC50:  8.80E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403034(CHEMBL2114397)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403035(OXFENICINE)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM18957((2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2,6-di...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM61402((Z)-2-butenedioic acid;2-(2,2-dicyclohexylethyl)pi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM80613(1-(2,3,4-Trimethoxy-benzyl)-piperazine | 1-(2,3,4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403042(CHEMBL2216775)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50403037(CHEMBL2216774)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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