TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged BMP2K kinase domain (38 to 345 residues) (unknown origin...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 4.40E+3nMAssay Description:Binding affinity to biotinylated BMP2K (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assa...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: 9.50E+4nMAssay Description:Binding affinity to C-terminal AVI-tagged BMP2K (unknown origin) (38 to 345 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to C-terminal AVI-tagged BMP2K (unknown origin) (38 to 345 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to C-terminal AVI-tagged BMP2K (unknown origin) (38 to 345 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human BIKe using peptide as substrate incubated for 120 mins in presence of [gamma-33ATP] by scintillation counting based r...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human BIKe using peptide as substrate incubated for 120 mins in presence of [gamma-33ATP] by scintillation counting based r...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of wild-type human partial length BIKE (S34 to N329 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 161nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 707nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of NanoLuc-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of BIKE (unknown origin)More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 2.74E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair
TargetBMP-2-inducible protein kinase(Homo sapiens (Human))
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
University Of North Carolina At Chapel Hill (Unc-Ch)
Curated by ChEMBL
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused BMP2K (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by ...More data for this Ligand-Target Pair