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Found 82 hits Enz. Inhib. hit(s) with Target = 'NADPH-dependent enoyl-ACP reductase (FabI)'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM231620
PNG
(CG400549 | US10071965, Compound CG400549)
Show SMILES Cc1c(N)cccc1Cn1ccc(OCCc2cccs2)cc1=O
Show InChI InChI=1S/C19H20N2O2S/c1-14-15(4-2-6-18(14)20)13-21-9-7-16(12-19(21)22)23-10-8-17-5-3-11-24-17/h2-7,9,11-12H,8,10,13,20H2,1H3
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1.30n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM190654
PNG
(PT173)
Show SMILES CCCCCCc1ccn(Cc2cccc(N)c2C)c(=O)c1
Show InChI InChI=1S/C19H26N2O/c1-3-4-5-6-8-16-11-12-21(19(22)13-16)14-17-9-7-10-18(20)15(17)2/h7,9-13H,3-6,8,14,20H2,1-2H3
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2n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM190661
PNG
(PT166)
Show SMILES CCCCCCc1cc(=O)c(Oc2ccccc2C)cn1C
Show InChI InChI=1S/C19H25NO2/c1-4-5-6-7-11-16-13-17(21)19(14-20(16)3)22-18-12-9-8-10-15(18)2/h8-10,12-14H,4-7,11H2,1-3H3
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2.70n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM231623
PNG
(PT159)
Show SMILES CCCCCCc1cc(=O)c(Cc2ccccc2C#N)cn1C
Show InChI InChI=1S/C20H24N2O/c1-3-4-5-6-11-19-13-20(23)18(15-22(19)2)12-16-9-7-8-10-17(16)14-21/h7-10,13,15H,3-6,11-12H2,1-2H3
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11n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM190653
PNG
(PT172)
Show SMILES CCCCCCc1ccn(Cc2ccccc2Cl)c(=O)c1
Show InChI InChI=1S/C18H22ClNO/c1-2-3-4-5-8-15-11-12-20(18(21)13-15)14-16-9-6-7-10-17(16)19/h6-7,9-13H,2-5,8,14H2,1H3
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11n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM190652
PNG
(LOX inhibitor, 13 | PT171)
Show SMILES CCCCCCc1ccn(Cc2ccccc2C)c(=O)c1
Show InChI InChI=1S/C23H24ClN3O2/c1-17(28)26-11-13-27(14-12-26)21-7-5-20(6-8-21)25-16-22-9-10-23(29-22)18-3-2-4-19(24)15-18/h2-10,15,25H,11-14,16H2,1H3
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11.9n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM190655
PNG
(PT179)
Show SMILES CCCCCCc1ccn(Cc2ccccc2)c(=O)c1
Show InChI InChI=1S/C18H23NO/c1-2-3-4-6-9-16-12-13-19(18(20)14-16)15-17-10-7-5-8-11-17/h5,7-8,10-14H,2-4,6,9,15H2,1H3
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19n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM231621
PNG
(PT420)
Show SMILES CCCCCc1ccn(Cc2ccccc2C#N)c(=O)c1
Show InChI InChI=1S/C18H20N2O/c1-2-3-4-7-15-10-11-20(18(21)12-15)14-17-9-6-5-8-16(17)13-19/h5-6,8-12H,2-4,7,14H2,1H3
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29.6n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM231624
PNG
(PT191)
Show SMILES CCCCCCc1ccc(Oc2ccccc2)c(=O)[nH]1
Show InChI InChI=1S/C17H21NO2/c1-2-3-4-6-9-14-12-13-16(17(19)18-14)20-15-10-7-5-8-11-15/h5,7-8,10-13H,2-4,6,9H2,1H3,(H,18,19)
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197n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM231622
PNG
(PT170 | US10071965, Compound PT170)
Show SMILES Cc1ccn(Cc2ccccc2Cl)c(=O)c1
Show InChI InChI=1S/C13H12ClNO/c1-10-6-7-15(13(16)8-10)9-11-4-2-3-5-12(11)14/h2-8H,9H2,1H3
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229n/an/an/an/an/an/a7.5n/a



University of Wuerzburg



Assay Description
Kinetics were performed on a Cary 100 spectrophotometer (Varian) at 20 C. Reaction velocities were measured by monitoring the oxidation of NAD(P)H t...


J Biol Chem 289: 15987-6005 (2014)


Article DOI: 10.1074/jbc.M113.532804
BindingDB Entry DOI: 10.7270/Q2H41Q89
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133668
PNG
(US8846711, 12 | US9051321, 12)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CC(C1)OCc1cccs1
Show InChI InChI=1S/C19H19N3O3S/c23-17-5-4-14-8-13(9-20-19(14)21-17)3-6-18(24)22-10-15(11-22)25-12-16-2-1-7-26-16/h1-3,6-9,15H,4-5,10-12H2,(H,20,21,23)/b6-3+
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n/an/a 13n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM50399404
PNG
(CHEMBL2178287 | US8623865, 1)
Show SMILES CCc1cc(O)c(Oc2ccc(cc2F)C(=O)N2CCNC(=O)C2)cc1F
Show InChI InChI=1S/C19H18F2N2O4/c1-2-11-8-15(24)17(9-13(11)20)27-16-4-3-12(7-14(16)21)19(26)23-6-5-22-18(25)10-23/h3-4,7-9,24H,2,5-6,10H2,1H3,(H,22,25)
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n/an/a 16n/an/an/an/a6.5n/a



Fab Pharma S.A.S.

US Patent


Assay Description
The assay buffer AB contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 mM...


US Patent US8623865 (2014)


BindingDB Entry DOI: 10.7270/Q21R6P6R
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133671
PNG
(US8846711, 15 | US9051321, 15)
Show SMILES CCCCCOC1CN(C1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C19H25N3O3/c1-2-3-4-9-25-16-12-22(13-16)18(24)8-5-14-10-15-6-7-17(23)21-19(15)20-11-14/h5,8,10-11,16H,2-4,6-7,9,12-13H2,1H3,(H,20,21,23)/b8-5+
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n/an/a 25n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM50399405
PNG
(CHEMBL2178286 | US8623865, 2)
Show SMILES CCc1ccc(Oc2ccc(cc2F)C(=O)N2CCNC(=O)C2)c(O)c1
Show InChI InChI=1S/C19H19FN2O4/c1-2-12-3-5-17(15(23)9-12)26-16-6-4-13(10-14(16)20)19(25)22-8-7-21-18(24)11-22/h3-6,9-10,23H,2,7-8,11H2,1H3,(H,21,24)
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n/an/a 29n/an/an/an/a6.5n/a



Fab Pharma S.A.S.

US Patent


Assay Description
The assay buffer AB contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 mM...


US Patent US8623865 (2014)


BindingDB Entry DOI: 10.7270/Q21R6P6R
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133664
PNG
(US8846711, 8 | US9051321, 8)
Show SMILES CCCC1CCN(CC1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C19H25N3O2/c1-2-3-14-8-10-22(11-9-14)18(24)7-4-15-12-16-5-6-17(23)21-19(16)20-13-15/h4,7,12-14H,2-3,5-6,8-11H2,1H3,(H,20,21,23)/b7-4+
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n/an/a 41n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133673
PNG
(US8846711, 17 | US9051321, 17)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CC(C1)OCc1ccccc1
Show InChI InChI=1S/C21H21N3O3/c25-19-8-7-17-10-16(11-22-21(17)23-19)6-9-20(26)24-12-18(13-24)27-14-15-4-2-1-3-5-15/h1-6,9-11,18H,7-8,12-14H2,(H,22,23,25)/b9-6+
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n/an/a 50n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133676
PNG
(US8846711, 20 | US9051321, 20)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CC(C1)OCc1nccs1
Show InChI InChI=1S/C18H18N4O3S/c23-15-3-2-13-7-12(8-20-18(13)21-15)1-4-17(24)22-9-14(10-22)25-11-16-19-5-6-26-16/h1,4-8,14H,2-3,9-11H2,(H,20,21,23)/b4-1+
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n/an/a 57n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133681
PNG
(US8846711, 25 | US8846711, 26 | US9051321, 25)
Show SMILES COC(=O)C1Cc2cc(\C=C\C(=O)N3CCC(COc4ccc(F)cc4)CC3)cnc2NC1=O
Show InChI InChI=1S/C25H26FN3O5/c1-33-25(32)21-13-18-12-17(14-27-23(18)28-24(21)31)2-7-22(30)29-10-8-16(9-11-29)15-34-20-5-3-19(26)4-6-20/h2-7,12,14,16,21H,8-11,13,15H2,1H3,(H,27,28,31)/b7-2+
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n/an/a 60n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM9913
PNG
(US8846711, 26 | US9051321, 27)
Show SMILES NC(=O)C1Cc2cc(\C=C\C(=O)N3CCC(COc4ccc(F)cc4)CC3)cnc2NC1=O
Show InChI InChI=1S/C24H25FN4O4/c25-18-2-4-19(5-3-18)33-14-15-7-9-29(10-8-15)21(30)6-1-16-11-17-12-20(22(26)31)24(32)28-23(17)27-13-16/h1-6,11,13,15,20H,7-10,12,14H2,(H2,26,31)(H,27,28,32)/b6-1+
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n/an/a 78n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133683
PNG
(US8846711, 28 | US9051321, 28)
Show SMILES OCC1Cc2cc(\C=C\C(=O)N3CCC(COc4ccc(F)cc4)CC3)cnc2NC1=O
Show InChI InChI=1S/C24H26FN3O4/c25-20-2-4-21(5-3-20)32-15-16-7-9-28(10-8-16)22(30)6-1-17-11-18-12-19(14-29)24(31)27-23(18)26-13-17/h1-6,11,13,16,19,29H,7-10,12,14-15H2,(H,26,27,31)/b6-1+
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n/an/a 81n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133666
PNG
(US8846711, 10 | US9051321, 10)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(C1)Oc1ccccc1
Show InChI InChI=1S/C21H21N3O3/c25-19-8-7-16-12-15(13-22-21(16)23-19)6-9-20(26)24-11-10-18(14-24)27-17-4-2-1-3-5-17/h1-6,9,12-13,18H,7-8,10-11,14H2,(H,22,23,25)/b9-6+
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n/an/a 120n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM162339
PNG
(US9051321, 11)
Show SMILES Cc1nc(no1)C1CN(C1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C17H17N5O3/c1-10-19-17(21-25-10)13-8-22(9-13)15(24)5-2-11-6-12-3-4-14(23)20-16(12)18-7-11/h2,5-7,13H,3-4,8-9H2,1H3,(H,18,20,23)/b5-2+
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n/an/a 150n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133675
PNG
(US8846711, 19 | US9051321, 19)
Show SMILES CC(=C)COC1CN(C1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C18H21N3O3/c1-12(2)11-24-15-9-21(10-15)17(23)6-3-13-7-14-4-5-16(22)20-18(14)19-8-13/h3,6-8,15H,1,4-5,9-11H2,2H3,(H,19,20,22)/b6-3+
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n/an/a 170n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133661
PNG
(US8846711, 5 | US9051321, 5)
Show SMILES CC(C)(C)OC(=O)N1CCC(COc2ccc(F)cc2)CC1
Show InChI InChI=1S/C17H24FNO3/c1-17(2,3)22-16(20)19-10-8-13(9-11-19)12-21-15-6-4-14(18)5-7-15/h4-7,13H,8-12H2,1-3H3
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n/an/a 250n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133680
PNG
(US8846711, 24 | US9051321, 24)
Show SMILES CC(=O)Nc1ccc(\C=C\C(=O)N2CC(C2)OCc2ccncc2)cn1
Show InChI InChI=1S/C19H20N4O3/c1-14(24)22-18-4-2-15(10-21-18)3-5-19(25)23-11-17(12-23)26-13-16-6-8-20-9-7-16/h2-10,17H,11-13H2,1H3,(H,21,22,24)/b5-3+
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n/an/a 260n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133670
PNG
(US8846711, 14 | US9051321, 14)
Show SMILES OC1(CCN(CC1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1)c1ccccc1
Show InChI InChI=1S/C22H23N3O3/c26-19-8-7-17-14-16(15-23-21(17)24-19)6-9-20(27)25-12-10-22(28,11-13-25)18-4-2-1-3-5-18/h1-6,9,14-15,28H,7-8,10-13H2,(H,23,24,26)/b9-6+
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n/an/a 340n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM9913
PNG
(US8846711, 26 | US9051321, 27)
Show SMILES NC(=O)C1Cc2cc(\C=C\C(=O)N3CCC(COc4ccc(F)cc4)CC3)cnc2NC1=O
Show InChI InChI=1S/C24H25FN4O4/c25-18-2-4-19(5-3-18)33-14-15-7-9-29(10-8-15)21(30)6-1-16-11-17-12-20(22(26)31)24(32)28-23(17)27-13-16/h1-6,11,13,15,20H,7-10,12,14H2,(H2,26,31)(H,27,28,32)/b6-1+
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n/an/a 550n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302048
PNG
(US9598407, Compound 4)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(CC1)c1ccccc1
Show InChI InChI=1S/C22H23N3O2/c26-20-8-7-19-14-16(15-23-22(19)24-20)6-9-21(27)25-12-10-18(11-13-25)17-4-2-1-3-5-17/h1-6,9,14-15,18H,7-8,10-13H2,(H,23,24,26)/b9-6+
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n/an/a 802n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302046
PNG
(US9598407, Compound 2)
Show SMILES COc1ccccc1C1=CCN(CC1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C23H23N3O3/c1-29-20-5-3-2-4-19(20)17-10-12-26(13-11-17)22(28)9-6-16-14-18-7-8-21(27)25-23(18)24-15-16/h2-6,9-10,14-15H,7-8,11-13H2,1H3,(H,24,25,27)/b9-6+
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n/an/a 821n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302056
PNG
(US9598407, Compound 12)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(Cc2ccccc2)CC1
Show InChI InChI=1S/C23H25N3O2/c27-21-8-7-20-15-19(16-24-23(20)25-21)6-9-22(28)26-12-10-18(11-13-26)14-17-4-2-1-3-5-17/h1-6,9,15-16,18H,7-8,10-14H2,(H,24,25,27)/b9-6+
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Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133677
PNG
(US8846711, 21 | US9051321, 21)
Show SMILES C\C(Cc1ncccn1)=N/OC1CN(C1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C21H22N6O3/c1-14(9-18-22-7-2-8-23-18)26-30-17-12-27(13-17)20(29)6-3-15-10-16-4-5-19(28)25-21(16)24-11-15/h2-3,6-8,10-11,17H,4-5,9,12-13H2,1H3,(H,24,25,28)/b6-3+,26-14+
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n/an/a 870n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302049
PNG
(US9598407, Compound 5)
Show SMILES Oc1cccc(c1)C1CCN(CC1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C22H23N3O3/c26-19-3-1-2-17(13-19)16-8-10-25(11-9-16)21(28)7-4-15-12-18-5-6-20(27)24-22(18)23-14-15/h1-4,7,12-14,16,26H,5-6,8-11H2,(H,23,24,27)/b7-4+
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Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133672
PNG
(US8846711, 16 | US9051321, 16)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(C1)Oc1cccnc1
Show InChI InChI=1S/C20H20N4O3/c25-18-5-4-15-10-14(11-22-20(15)23-18)3-6-19(26)24-9-7-17(13-24)27-16-2-1-8-21-12-16/h1-3,6,8,10-12,17H,4-5,7,9,13H2,(H,22,23,25)/b6-3+
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FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302053
PNG
(US9598407, Compound 9)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(=CC1)c1ccco1
Show InChI InChI=1S/C20H19N3O3/c24-18-5-4-16-12-14(13-21-20(16)22-18)3-6-19(25)23-9-7-15(8-10-23)17-2-1-11-26-17/h1-3,6-7,11-13H,4-5,8-10H2,(H,21,22,24)/b6-3+
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n/an/a 973n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM162329
PNG
(US9051321, 6)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CC(C1)Oc1ccccc1
Show InChI InChI=1S/C20H19N3O3/c24-18-8-7-15-10-14(11-21-20(15)22-18)6-9-19(25)23-12-17(13-23)26-16-4-2-1-3-5-16/h1-6,9-11,17H,7-8,12-13H2,(H,21,22,24)/b9-6+
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FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302051
PNG
(US9598407, Compound 7)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(=CC1)c1ccccc1
Show InChI InChI=1S/C22H21N3O2/c26-20-8-7-19-14-16(15-23-22(19)24-20)6-9-21(27)25-12-10-18(11-13-25)17-4-2-1-3-5-17/h1-6,9-10,14-15H,7-8,11-13H2,(H,23,24,26)/b9-6+
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n/an/a 1.14E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302077
PNG
(US9598407, Compound 34)
Show SMILES Fc1ccc(OCC2CCN(CC2)C(=O)\C=C\c2cnc3NC(=O)CCc3c2)cc1
Show InChI InChI=1S/C23H24FN3O3/c24-19-3-5-20(6-4-19)30-15-16-9-11-27(12-10-16)22(29)8-1-17-13-18-2-7-21(28)26-23(18)25-14-17/h1,3-6,8,13-14,16H,2,7,9-12,15H2,(H,25,26,28)/b8-1+
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Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302078
PNG
(US9598407, Compound 35)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(Cc2ccccn2)CC1
Show InChI InChI=1S/C22H24N4O2/c27-20-6-5-18-13-17(15-24-22(18)25-20)4-7-21(28)26-11-8-16(9-12-26)14-19-3-1-2-10-23-19/h1-4,7,10,13,15-16H,5-6,8-9,11-12,14H2,(H,24,25,27)/b7-4+
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n/an/a 1.27E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM162330
PNG
(US9051321, 9)
Show SMILES Fc1ccc(OCC2CCCN(C2)C(=O)\C=C\c2cnc3NC(=O)CCc3c2)cc1
Show InChI InChI=1S/C23H24FN3O3/c24-19-5-7-20(8-6-19)30-15-17-2-1-11-27(14-17)22(29)10-3-16-12-18-4-9-21(28)26-23(18)25-13-16/h3,5-8,10,12-13,17H,1-2,4,9,11,14-15H2,(H,25,26,28)/b10-3+
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n/an/a 1.30E+3n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302080
PNG
(US9598407, Compound 37)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(Cc2cccs2)CC1
Show InChI InChI=1S/C21H23N3O2S/c25-19-5-4-17-12-16(14-22-21(17)23-19)3-6-20(26)24-9-7-15(8-10-24)13-18-2-1-11-27-18/h1-3,6,11-12,14-15H,4-5,7-10,13H2,(H,22,23,25)/b6-3+
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n/an/a 1.31E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302052
PNG
(US9598407, Compound 8)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(=CC1)c1ccc2OCOc2c1
Show InChI InChI=1S/C23H21N3O4/c27-21-5-3-18-11-15(13-24-23(18)25-21)1-6-22(28)26-9-7-16(8-10-26)17-2-4-19-20(12-17)30-14-29-19/h1-2,4,6-7,11-13H,3,5,8-10,14H2,(H,24,25,27)/b6-1+
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US Patent
n/an/a 1.31E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302057
PNG
(US9598407, Compound 13)
Show SMILES COc1ccccc1C1CCN(CC1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C23H25N3O3/c1-29-20-5-3-2-4-19(20)17-10-12-26(13-11-17)22(28)9-6-16-14-18-7-8-21(27)25-23(18)24-15-16/h2-6,9,14-15,17H,7-8,10-13H2,1H3,(H,24,25,27)/b9-6+
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n/an/a 1.35E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302054
PNG
(US9598407, Compound 10)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(=CC1)c1ccoc1
Show InChI InChI=1S/C20H19N3O3/c24-18-3-2-16-11-14(12-21-20(16)22-18)1-4-19(25)23-8-5-15(6-9-23)17-7-10-26-13-17/h1,4-5,7,10-13H,2-3,6,8-9H2,(H,21,22,24)/b4-1+
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n/an/a 1.37E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302047
PNG
(US9598407, Compound 3)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCc2ccccc2C1
Show InChI InChI=1S/C20H19N3O2/c24-18-7-6-16-11-14(12-21-20(16)22-18)5-8-19(25)23-10-9-15-3-1-2-4-17(15)13-23/h1-5,8,11-12H,6-7,9-10,13H2,(H,21,22,24)/b8-5+
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n/an/a 1.43E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302060
PNG
(US9598407, Compound 16)
Show SMILES Clc1ccccc1C1=CCN(CC1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C22H20ClN3O2/c23-19-4-2-1-3-18(19)16-9-11-26(12-10-16)21(28)8-5-15-13-17-6-7-20(27)25-22(17)24-14-15/h1-5,8-9,13-14H,6-7,10-12H2,(H,24,25,27)/b8-5+
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n/an/a 1.47E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302071
PNG
(US9598407, Compound 27)
Show SMILES CC1CN(CC=C1c1ccccc1)C(=O)\C=C\c1cnc2NC(=O)CCc2c1
Show InChI InChI=1S/C23H23N3O2/c1-16-15-26(12-11-20(16)18-5-3-2-4-6-18)22(28)10-7-17-13-19-8-9-21(27)25-23(19)24-14-17/h2-7,10-11,13-14,16H,8-9,12,15H2,1H3,(H,24,25,27)/b10-7+
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n/an/a 1.52E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302079
PNG
(US9598407, Compound 36)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCC(CC2CCCS2)CC1
Show InChI InChI=1S/C21H27N3O2S/c25-19-5-4-17-12-16(14-22-21(17)23-19)3-6-20(26)24-9-7-15(8-10-24)13-18-2-1-11-27-18/h3,6,12,14-15,18H,1-2,4-5,7-11,13H2,(H,22,23,25)/b6-3+
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n/an/a 1.58E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133674
PNG
(US8846711, 18 | US9051321, 18)
Show SMILES O=C(\C=C\c1cnc2NC(=O)CCc2c1)N1CCCC[C@@H]1c1nc2ccccc2o1
Show InChI InChI=1S/C23H22N4O3/c28-20-10-9-16-13-15(14-24-22(16)26-20)8-11-21(29)27-12-4-3-6-18(27)23-25-17-5-1-2-7-19(17)30-23/h1-2,5,7-8,11,13-14,18H,3-4,6,9-10,12H2,(H,24,26,28)/b11-8+/t18-/m1/s1
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n/an/a 1.80E+3n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM133679
PNG
(US8846711, 23 | US9051321, 23)
Show SMILES Nc1ccc(\C=C\C(=O)N2CC(C2)OCc2ccncc2)cn1
Show InChI InChI=1S/C17H18N4O2/c18-16-3-1-13(9-20-16)2-4-17(22)21-10-15(11-21)23-12-14-5-7-19-8-6-14/h1-9,15H,10-12H2,(H2,18,20)/b4-2+
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Similars

US Patent
n/an/a 1.80E+3n/an/an/an/a6.525



FAB PHARMA S.A.S.

US Patent


Assay Description
The assay buffer "AB" contained 50 mM ADA (N-(2-acetamido)iminodiacetic acid monosodium salt) pH 6.5, 1 mM dithiothreitol, 0.006% Triton-X100 and 50 ...


US Patent US9051321 (2015)


BindingDB Entry DOI: 10.7270/Q2WW7GDG
More data for this
Ligand-Target Pair
NADPH-dependent enoyl-ACP reductase (FabI)


(Staphylococcus aureus)
BDBM302075
PNG
(US9598407, Compound 31)
Show SMILES Fc1ccc2c(CC3CCN(CC3)C(=O)\C=C\c3cnc4NC(=O)CCc4c3)coc2c1
Show InChI InChI=1S/C25H24FN3O3/c26-20-3-4-21-19(15-32-22(21)13-20)11-16-7-9-29(10-8-16)24(31)6-1-17-12-18-2-5-23(30)28-25(18)27-14-17/h1,3-4,6,12-16H,2,5,7-11H2,(H,27,28,30)/b6-1+
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n/an/a 1.82E+3n/an/an/an/an/an/a



Janssen Sciences Ireland UC

US Patent


Assay Description
FabI enzyme inhibition assays were carried out in half-area, 384-well microtitre plates. Compounds were evaluated in 40-μl assay mixtures contai...


US Patent US9598407 (2017)

More data for this
Ligand-Target Pair
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