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Found 505 Enz. Inhib. hit(s) with Target = 'DNA repair protein RAD51 homolog 1'
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50088343(CHEMBL3427781)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to of humanised RAD51 C-terminal ATPase domain (with deletion of L2 loop residues 288 to 314) from Pyrococcus furiosus expressed in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50088343(CHEMBL3427781)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to RAD51 (unknown origin) by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50088345(CHEMBL3427780)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to RAD51 (unknown origin) by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM48804(3-(phenylmethyl)-2-[(E)-2-(3-pyridinyl)ethenyl]-4-...)
Affinity DataKd:  5.60E+3nMAssay Description:Binding affinity to human RAD51 in absence of ATP by SPR methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50527107(CHEMBL4450955)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to recombinant His-tagged human RAD51 expressed in Escherichia coli Rosetta(DE3) pLysS cells by microscale thermophoresis analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50088346(CHEMBL3427779)
Affinity DataKd:  3.50E+4nMAssay Description:Binding affinity to RAD51 (unknown origin) by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM93044(L-Methyl ester tryptophan, 8)
Affinity DataKd:  5.70E+5nMAssay Description:Binding affinity to RAD51 (unknown origin) by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM93044(L-Methyl ester tryptophan, 8)
Affinity DataKd:  5.70E+5nMAssay Description:Binding affinity to of humanised RAD51 C-terminal ATPase domain (with deletion of L2 loop residues 288 to 314) from Pyrococcus furiosus expressed in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM32212(1H-indol-5-ol | cid_16054)
Affinity DataKd:  2.10E+6nMAssay Description:Binding affinity to RAD51 (unknown origin) by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50416570(CHEMBL1215819)
Affinity DataKi:  750nMAssay Description:Inhibition of human RAD51 assessed as concentration required for half dissociation of protein/single-stranded DNA complex formation by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50416568(CHEMBL1215817)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human RAD51 assessed as concentration required for half dissociation of protein/single-stranded DNA complex formation by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50416569(CHEMBL1215818)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of human RAD51 assessed as concentration required for half dissociation of protein/single-stranded DNA complex formation by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50416566(CHEMBL1215815)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human RAD51 assessed as concentration required for half dissociation of protein/single-stranded DNA complex formation by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50416564(CHEMBL1215813)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human RAD51 assessed as concentration required for half dissociation of protein/single-stranded DNA complex formation by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50416567(CHEMBL1215816)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of human RAD51 assessed as concentration required for half dissociation of protein/single-stranded DNA complex formation by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50055659(2N-(3,3-aminoiminopropyl)-4-[4-(4-formamido-1-meth...)
Affinity DataIC50:  4.70E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51310(6,7,12,15,15-pentamethyl-3,10-diazatetracyclo[10.2...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM44459(1,1,3-Trimethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51311(3-[[8,9-dimethoxy-2-(3-pyridyl)-[1,2,4]triazolo[1,...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51312(3-[(8,9-dimethoxy-2-phenyl-[1,2,4]triazolo[1,5-c]q...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM43826(2-[5-(diethylsulfamoyl)-1-(4-methoxyphenyl)benzimi...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51314((6-chloranyl-2-phenyl-chromen-4-ylidene)-(2,2,6,6-...)
Affinity DataIC50:  3.66E+3nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM48804(3-(phenylmethyl)-2-[(E)-2-(3-pyridinyl)ethenyl]-4-...)
Affinity DataIC50:  4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51315(3-[(2Z)-2-(3-formyl-4-oxo-1-cyclohexa-2,5-dienylid...)
Affinity DataIC50:  4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM32329((2Z)-3-ethyl-2-[(E)-3-(3-ethyl-1,3-benzothiazol-3-...)
Affinity DataIC50:  4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM29673(1,4,10-Trihydroxy-5-hydroxymethyl-8-methyl-3,7-dio...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50056922(1,4-Dihydroxy-10-methoxy-5,8-dimethyl-3,7-dioxo-1,...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)
Affinity DataIC50:  2.68E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM43864(2-chloranyl-N1,N4-bis[4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataIC50:  1.64E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM43865(6-formyl-4,7-dihydroxy-9-keto-5H-phenazine-1-carbo...)
Affinity DataIC50:  4.25E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50056939(4-Formyl-3-hydroxy-8-methoxy-1,9-dimethyl-11-oxo-1...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM43866(2-amino-4,6-dimethyl-3-oxo-1-N,9-N-bis[(3R,6S,7R,1...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51319(2-(7-benzyl-2,6-diketo-3-methyl-8-piperidino-purin...)
Affinity DataIC50:  8.50E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM45326((4E)-4-[2,3-dihydro-1,4-benzodioxin-6-yl(hydroxy)m...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51320(4-[2-(4-methylphenyl)-3,4-dioxo-1-cyclobutenyl]-1-...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51321(2-(2,4-dimethoxyphenyl)-1H-indene-1,3(2H)-dione | ...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM39401(4-[4-(4-methoxyphenyl)piperazin-1-yl]carbonyl-2,9-...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51322(1,4-dioxa-8-azaspiro[4.5]decan-8-yl-[3-(3-methoxyp...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51323(4-(1-propylsulfonylnipecotoyl)piperazine-1-carboxy...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM38621(MLS000050598 | N-(2-ethyl-1,2,3,4-tetrazol-5-yl)-3...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51324(1-bromanylnaphthalen-2-ol | 1-bromo-2-naphthalenol...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM44459(1,1,3-Trimethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-...)
Affinity DataIC50:  1.06E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51311(3-[[8,9-dimethoxy-2-(3-pyridyl)-[1,2,4]triazolo[1,...)
Affinity DataIC50:  4.99E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51312(3-[(8,9-dimethoxy-2-phenyl-[1,2,4]triazolo[1,5-c]q...)
Affinity DataIC50:  2.11E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM33089((3-methyl-4-pyrrolidino-phenyl)amine;hydrochloride...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51325(8-chloranyl-N-(3-methoxyphenyl)-2-pyridin-3-yl-qui...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51326(1-(3,5-dimethylphenyl)-3-(1-phenyltetrazol-5-yl)su...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50230((E)-3-(4-chloranyl-3-nitro-phenyl)-N-(4-pyrrolidin...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetDNA repair protein RAD51 homolog 1(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM51327(MLS000723396 | N-(1-naphthalenyl)hexanamide | N-(1...)
Affinity DataIC50:  5.30E+4nMAssay Description:Project Title: A screen for modulators of human Rad51, a key DNA repair protein Application Number: MH084119 Assay Submitter: Dr. Alex Mazin Submitte...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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