Affinity DataKd: 0.340nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 0.340nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 0.340nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding affinity to Fc-tagged EphB4 (unknown origin) assessed as reduction in ephrin-B2 binding by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 9.20nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 12nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 520nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 520nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 520nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 560nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 560nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 560nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 570nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 730nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 750nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Average Binding Constant for EPHB4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Average Binding Constant for EPHB4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to recombinant N-terminal His-FLAG-GST-tagged EPHB4 (unknown origin) (577 to 987 residues) expressed in baculovirus infected Sf9 ins...More data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to EPHB4More data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.10E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+3nMAssay Description:Average Binding Constant for EPHB4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.60E+3nMAssay Description:Average Binding Constant for EPHB4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 2.70E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.80E+3nMpH: 7.4 T: 2°CAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 2.80E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.90E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.10E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.90E+3nMAssay Description:Average Binding Constant for EPHB4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 5.00E+3nMAssay Description:Average Binding Constant for EPHB4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 6.90E+3nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for EPHB4 kinase domainMore data for this Ligand-Target Pair