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Found 69 Enz. Inhib. hit(s) with Target = 'Myelin-associated glycoprotein'
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354062(CHEMBL1836190)
Affinity DataKd:  15nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354056(CHEMBL1836336)
Affinity DataKd:  130nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354061(CHEMBL1836340)
Affinity DataKd:  480nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354046(CHEMBL1836312)
Affinity DataKd:  500nMAssay Description:Binding affinity to MAGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327099(CHEMBL1253679 | sodium2R,4S,5R,6R)-6-((1R,2R)-3-(4...)
Affinity DataKd:  500nMAssay Description:Binding affinity to mouse MAGd1-3Fc domain expressed in CHO-Lec1 cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327099(CHEMBL1253679 | sodium2R,4S,5R,6R)-6-((1R,2R)-3-(4...)
Affinity DataKd:  500nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354055(CHEMBL1836335)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354054(CHEMBL1836334)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354058(CHEMBL1836337)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354060(CHEMBL1836339)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378605(CHEMBL590756)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354059(CHEMBL1836338)
Affinity DataKd:  1.76E+3nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354053(CHEMBL1836313)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378604(CHEMBL590929)
Affinity DataKd:  2.10E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378607(CHEMBL590980)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378603(CHEMBL600189)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50292878((Sodium 5-Acetamido-9-(4-chlorobenzamido)-3,5,9-tr...)
Affinity DataKd:  2.83E+3nMAssay Description:Binding affinity to human IgG Fc-domain tagged MAG N-terminal domain expressed in CHO cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378610(CHEMBL590917)
Affinity DataKd:  2.83E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378608(CHEMBL601721)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378602(CHEMBL600188)
Affinity DataKd:  4.30E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378611(CHEMBL590827)
Affinity DataKd:  4.44E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50292879((Sodium 5-Acetamido-9-benzamido-3,5,9-trideoxy-D-g...)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to human IgG Fc-domain tagged MAG N-terminal domain expressed in CHO cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378609(CHEMBL601722)
Affinity DataKd:  5.80E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378600(CHEMBL590978)
Affinity DataKd:  6.10E+3nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378601(CHEMBL590979)
Affinity DataKd:  1.16E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378613(CHEMBL598744)
Affinity DataKd:  1.17E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354057(CHEMBL1833997)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to wild type MAG at 400 uM by Isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378599(CHEMBL603912)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  1.49E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under NaCl condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378598(CHEMBL600994)
Affinity DataKd:  1.50E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378597(CHEMBL239255)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378606(CHEMBL601720)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  1.76E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under HEPES condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  1.78E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under carboxymethyl-dextran sodium salt condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378612(CHEMBL394182)
Affinity DataKd:  1.92E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under HBS-EP condition by CM4 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  2.18E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells under HBS-EP condition by CM5 chip SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  2.60E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc domain expressed in CHO-Lec1 cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327098(CHEMBL1254099 | sodium(2R,4S,5R,6R)-5-acetamido-6-...)
Affinity DataKd:  2.60E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50556307(CHEMBL4788433)
Affinity DataKd:  3.07E+4nMAssay Description:Binding affinity to human MAG by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354047(CHEMBL1836311)
Affinity DataKd:  3.20E+4nMAssay Description:Binding affinity to MAGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50292880(2-(Trimethylsilyl)ethyl (Sodium 5-Acetamido-9-benz...)
Affinity DataKd:  3.26E+4nMAssay Description:Binding affinity to human IgG Fc-domain tagged MAG N-terminal domain expressed in CHO cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378614(CHEMBL391051)
Affinity DataKd:  3.39E+4nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50556306(CHEMBL4780037)
Affinity DataKd:  5.64E+4nMAssay Description:Binding affinity to human MAG by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378596(CHEMBL609756)
Affinity DataKd:  1.37E+5nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by biocoreMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50378596(CHEMBL609756)
Affinity DataKd:  1.37E+5nMAssay Description:Binding affinity to mouse MAGd1-3Fc expressed in CHO-Lec 3.2.8.1 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354045(CHEMBL1836305)
Affinity DataKd:  1.80E+5nMAssay Description:Binding affinity to MAGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354048(CHEMBL1836307)
Affinity DataKd:  1.80E+5nMAssay Description:Binding affinity to MAGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Mus musculus)
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50327100(CHEMBL1254194 | sodium(1R,3R,4R,5S)-5-acetamido-1-...)
Affinity DataKd: >8.00E+5nMAssay Description:Binding affinity to mouse MAGd1-3Fc domain expressed in CHO-Lec1 cells by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354058(CHEMBL1836337)
Affinity DataIC50:  640nMAssay Description:Inhibition of MAG -Fc chimera expressed in CHO cells using NeuAc alpha2-3Galbeta1-4GlcNAc-R coupled biotinylated polyacrylamide after 30 mins by ELIS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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