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Found 524 Enz. Inhib. hit(s) with Target = 'Tubulin beta chain'
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485036(CHEMBL2024544)
Affinity DataKd:  200nMAssay Description:Binding affinity to porcine tubulin after 1 hr by spectrofluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485035(CHEMBL2024561)
Affinity DataKd:  620nMAssay Description:Binding affinity to porcine tubulin after 1 hr by spectrofluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030765(NPI-2358 | Plinabulin)
Affinity DataKd:  1.06E+3nMAssay Description:Binding affinity to porcine tubulin after 1 hr by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030765(NPI-2358 | Plinabulin)
Affinity DataKd:  1.06E+3nMAssay Description:Binding affinity to pig tubulin after 1 hr by fluorescence quenching analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030765(NPI-2358 | Plinabulin)
Affinity DataKd:  1.06E+3nMAssay Description:Binding affinity to porcine tubulin after 1 hr by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030766(CHEMBL3342339)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to porcine tubulin incubated for 1 hr by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50520178(CHEMBL4468642)
Affinity DataKd:  2.66E+3nMAssay Description:Binding affinity to porcine brain tubulin polymerization by surface plasmon analysis analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKd:  3.70E+3nMAssay Description:Binding affinity to porcine tubulin after 1 hr by spectrofluorometric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50482143(CHEMBL1077255 | KPU-244-B2)
Affinity DataKd:  9.74E+3nMAssay Description:Binding affinity to pig tubulin after 1 hr by fluorescence quenching analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKd:  1.13E+4nMAssay Description:Binding affinity to porcine brain tubulin polymerization by surface plasmon analysis analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50483308(CHEMBL1643852)
Affinity DataKd:  1.79E+4nMAssay Description:Binding affinity to porcine tubulin after 1 hr by spectrofluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50482142(CHEMBL1096312 | KPU-244-B3)
Affinity DataKd:  2.52E+4nMAssay Description:Binding affinity to pig tubulin after 1 hr by fluorescence quenching analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Homo sapiens)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50501218(CHEMBL3917601)
Affinity DataKd:  6.54E+5nMAssay Description:Binding affinity to human recombinant tubulin alpha 1A/tubulin beta chain after 30 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Homo sapiens)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50501217(CHEMBL4298925)
Affinity DataKd:  1.06E+6nMAssay Description:Binding affinity to human recombinant tubulin alpha 1A/tubulin beta chain after 30 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485941(CHEMBL2181004)
Affinity DataKi:  0.0460nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485945(CHEMBL2181003)
Affinity DataKi:  0.0585nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485942(CHEMBL2181002)
Affinity DataKi:  0.0637nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485950(CHEMBL2181009)
Affinity DataKi:  0.122nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485944(CHEMBL2181006)
Affinity DataKi:  0.127nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485943(CHEMBL2181001)
Affinity DataKi:  0.131nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485946(CHEMBL2181000)
Affinity DataKi:  0.143nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485947(CHEMBL2181008)
Affinity DataKi:  0.183nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485949(CHEMBL2180999)
Affinity DataKi:  0.198nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485948(CHEMBL2181007)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50485940(CHEMBL2181005)
Affinity DataKi:  0.367nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataKi:  2.18E+3nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKi:  5.75E+3nMAssay Description:Binding affinity against tubulin usingf [3H]-colchicine as radioligandMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50146019(steganacin)
Affinity DataKi:  1.05E+4nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50146021(CHEMBL152714)
Affinity DataKi:  3.20E+4nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50146017(CHEMBL152476)
Affinity DataKi:  1.00E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50146018(CHEMBL3349041)
Affinity DataKi:  1.78E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50146022(CHEMBL346865)
Affinity DataKi:  1.85E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50146018(CHEMBL3349041)
Affinity DataKi:  1.85E+5nMAssay Description:Binding affinity against tubulin usingf [3H]-colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50146016(CHEMBL149525)
Affinity DataKi:  2.01E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030765(NPI-2358 | Plinabulin)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of porcine tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030766(CHEMBL3342339)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of porcine tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160798(4,4''-Dimethoxy-9,10-dihydro-[1,1'']biphenanthreny...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160799(8-(4-Hydroxy-benzyl)-7-methoxy-9,10-dihydro-phenan...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160800(1,3-Bis-(4-hydroxy-benzyl)-4-methoxy-9,10-dihydro-...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160801(4-(4-Hydroxy-benzyl)-3-[2-(3-hydroxy-phenyl)-ethyl...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160802(2,4-Bis-(4-hydroxy-benzyl)-3-[2-(3-hydroxy-phenyl)...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160803(4,4''-Dimethoxy-9,10,9'',10''-tetrahydro-[1,3'']bi...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160804(4,4''-Dimethoxy-[1,1'']biphenanthrenyl-2,7,2'',7''...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50160805(1-(4-Hydroxy-benzyl)-4,8-dimethoxy-phenanthrene-2,...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of tubulin polymerization interacting at the colchicine binding site.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50156479(5-((S)-2-Oxo-4-phenyl-imidazolidine-1-sulfonyl)-2,...)
Affinity DataIC50:  3.00E+4nMAssay Description:Compound was tested for inhibition of tubulin polymerisationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50156480((S)-4-Phenyl-1-[1-(2-phenylamino-acetyl)-2,3-dihyd...)
Affinity DataIC50:  3.50E+3nMAssay Description:Compound was tested for inhibition of tubulin polymerisationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50156482(4-Amino-N-[2-chloro-4-((S)-2-oxo-4-phenyl-imidazol...)
Affinity DataIC50:  5.50E+3nMAssay Description:Compound was tested for inhibition of tubulin polymerisationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain [1-43](Leishmania donovani)
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50156484((S)-1-[1-(5-Nitro-furan-2-carbonyl)-2,3-dihydro-1H...)
Affinity DataIC50:  4.00E+4nMAssay Description:Compound was tested for inhibition of tubulin polymerisationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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