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Found 70 Enz. Inhib. hit(s) with Target = 'tRNA (guanine-N(1)-)-methyltransferase'
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataKd:  1.60nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  91nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataKd:  190nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surfac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataKd:  3.10E+3nMAssay Description:Binding affinity to full length Staphylococcus aureus tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surface pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to full length Staphylococcus aureus tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surface pla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKd:  5.90E+3nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | CHEMBL418052 | S-(5'-adenosyl)-L-homocyst...)
Affinity DataKd:  1.01E+4nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surfac...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  1.04E+4nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surfac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  2.75E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surface pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225672(GTC000444A)
Affinity DataIC50:  3.16E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225673(GTC000445A)
Affinity DataIC50:  2.51E+4nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM50391357(CHEMBL69810 | GTC000446A)
Affinity DataIC50:  1.58E+5nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225674(GTC000447A)
Affinity DataIC50:  3.16E+5nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225675(GTC000448A)
Affinity DataIC50:  3.98E+4nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225676(GTC000449A)
Affinity DataIC50:  5.01nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225677(GTC000450A)
Affinity DataIC50:  5.01nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225678(GTC000451A)
Affinity DataIC50:  158nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225679(GTC000452A)
Affinity DataIC50:  2.00E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225680(GTC000453A)
Affinity DataIC50:  3.98E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225681(GTC000454A)
Affinity DataIC50:  794nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225682(GTC000455A)
Affinity DataIC50:  6.31E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225683(GTC000456A)
Affinity DataIC50:  7.94E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225684(GTC000457A)
Affinity DataIC50:  200nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225685(GTC000458A)
Affinity DataIC50:  501nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225686(GTC000459A)
Affinity DataIC50:  1.26E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225687(GTC000460A)
Affinity DataIC50:  200nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225688(GTC000461A)
Affinity DataIC50:  7.94E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225689(GTC000462A)
Affinity DataIC50:  2.00E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225690(GTC000463A)
Affinity DataIC50:  1.58E+4nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225691(GTC000464A)
Affinity DataIC50:  631nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225692(GTC000465A)
Affinity DataIC50:  2.00E+4nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225693(GTC000466A)
Affinity DataIC50:  1.58E+4nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225694(GTC000467A)
Affinity DataIC50:  631nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225695(GTC000468A)
Affinity DataIC50:  1.59E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225696(GTC000469A)
Affinity DataIC50:  501nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225697(GTC000470A)
Affinity DataIC50:  2.00E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225698(GTC000471A)
Affinity DataIC50:  794nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225699(GTC000472A)
Affinity DataIC50:  1.00E+5nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225700(GTC000473A)
Affinity DataIC50:  2.51E+3nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225701(GTC000474A)
Affinity DataIC50:  794nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519346(CHEMBL4580116)
Affinity DataIC50:  130nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519347(CHEMBL4555967)
Affinity DataIC50:  110nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataIC50:  60nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519350(CHEMBL4585250)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519351(CHEMBL4541348)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataIC50:  24nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519352(CHEMBL4458857)
Affinity DataIC50:  370nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519353(CHEMBL4564647)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology

Curated by ChEMBL
LigandPNGBDBM50519354(CHEMBL4469887)
Affinity DataIC50:  150nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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