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Found 3457 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A'
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91603(4' | alpha7 agonists 4')
Affinity DataKi:  900nM ΔG°:  -35.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM125052(US8772511, 21 | US9714242, 21)
Affinity DataKi:  1.60E+3nMpH: 7.4Assay Description:Membranes from HEK293 cells which express recombinant human 5-HT3 receptor (RB-HS3, Receptor Biology, Inc., MD, USA) are diluted in accordance with t...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM125049(US8772511, 6 | US9714242, 6)
Affinity DataKi:  1.70E+3nMpH: 7.4Assay Description:Membranes from HEK293 cells which express recombinant human 5-HT3 receptor (RB-HS3, Receptor Biology, Inc., MD, USA) are diluted in accordance with t...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM125051(US8772511, 16 | US9714242, 16)
Affinity DataKi:  2.10E+3nMpH: 7.4Assay Description:Membranes from HEK293 cells which express recombinant human 5-HT3 receptor (RB-HS3, Receptor Biology, Inc., MD, USA) are diluted in accordance with t...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91628(13t | alpha7 agonists 13t)
Affinity DataKi:  5.00E+3nM ΔG°:  -31.5kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM125050(US8772511, 11 | US9714242, 11)
Affinity DataKi:  5.50E+3nMpH: 7.4Assay Description:Membranes from HEK293 cells which express recombinant human 5-HT3 receptor (RB-HS3, Receptor Biology, Inc., MD, USA) are diluted in accordance with t...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM264253(N-[(3R)-1-Azabicyclo[2.2.2]oct-3-yl]-6-({[(3,4,5-t...)
Affinity DataKi:  6.90E+3nMpH: 7.4Assay Description:Membranes from HEK293 cells which express recombinant human 5-HT3 receptor (RB-HS3, Receptor Biology, Inc., MD, USA) are diluted in accordance with t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91617(17q | alpha7 agonists 17q)
Affinity DataKi:  8.00E+3nM ΔG°:  -30.3kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM125048(US8772511, 5 | US9714242, 5)
Affinity DataKi:  1.20E+4nMpH: 7.4Assay Description:Membranes from HEK293 cells which express recombinant human 5-HT3 receptor (RB-HS3, Receptor Biology, Inc., MD, USA) are diluted in accordance with t...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91633(18t | alpha7 agonists 18t)
Affinity DataKi:  1.20E+4nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91637(22t | alpha7 agonists 22t)
Affinity DataKi:  1.20E+4nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91624(alpha7 agonists 4t)
Affinity DataKi:  1.50E+4nM ΔG°:  -28.6kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91619(19q | alpha7 agonists 19q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91620(20q | alpha7 agonists 20q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91621(21q | alpha7 agonists 21q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91622(22q | alpha7 agonists 22q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91623(23q | alpha7 agonists 23q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91625(10t | alpha7 agonists 10t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91626(11t | alpha7 agonists 11t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91627(12t | alpha7 agonists 12t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91629(14t | alpha7 agonists 14t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91631(16t | alpha7 agonists 16t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91632(17t | alpha7 agonists 17t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91634(19t | alpha7 agonists 19t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91635(20t | alpha7 agonists 20t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91636(21t | alpha7 agonists 21t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91638(23t | alpha7 agonists 23t)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91596(alpha7 agonists 1)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91707(alpha7 agonists 1')
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91598(alpha7 agonists 2)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91599(2' | alpha7 agonists 2')
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91600(alpha7 agonists 3)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91601(3' | alpha7 agonists 3')
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91604(alpha7 agonists 5)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91605(5' | alpha7 agonists 5')
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91606(alpha7 agonists 6)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91607(alpha7 agonists 7)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91608(alpha7 agonists 8)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91609(alpha7 agonists 9)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91610(10q | alpha7 agonists 10q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91611(11q | alpha7 agonists 11q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91612(12q | alpha7 agonists 12q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91613(13q | alpha7 agonists 13q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91614(14q | alpha7 agonists 14q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91615(15q | alpha7 agonists 15q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91616(16q | alpha7 agonists 16q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91618(18q | alpha7 agonists 18q)
Affinity DataKi: >3.00E+4nM ΔG°: >-26.9kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91630(15t | alpha7 agonists 15t)
Affinity DataKi:  3.20E+4nM ΔG°:  -26.7kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
University Of California San Diego

LigandPNGBDBM91602(alpha7 agonists 4)
Affinity DataKi:  3.40E+4nM ΔG°:  -26.5kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Bayer Intellectual Property

US Patent
LigandPNGBDBM92417(PU04)
Affinity DataIC50:  1.00E+5nMpH: 7.4 T: 2°CAssay Description:The screening of the compound library at the h5-HT3A-HEK293 cell line and the subsequent functional characterization of the compounds were performed ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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