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Found 10 Enz. Inhib. hit(s) with Target = 'C-terminal-binding protein 1'
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154571(4-Methylthio 2-oxobutyric acid (MTOB))
Affinity DataKd:  1.26E+6nMpH: 7.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154570(2-Hydroxyimino-3-phenylpropanoic acid (HIPP))
Affinity DataKd:  370nMpH: 7.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM154570(2-Hydroxyimino-3-phenylpropanoic acid (HIPP))
Affinity DataKd:  2.77E+3nMpH: 8.5Assay Description:Purified CtBP2 was dialyzed overnight against 500 mL of 50 mM glycylglycine at pH 8.5, 300 mM NaCl, 1 mM EDTA, and 2 mM TCEP, with or without 1.5 mM ...More data for this Ligand-Target Pair
TargetC-terminal-binding protein 1 [R266Q](Homo sapiens (Human))
Oregon Health And Science University

LigandPNGBDBM213227(Nicotinamide adenine dinucleotide (NAD))
Affinity DataKd:  1.60E+3nMAssay Description:Equilibrium dialysis was performed using purified recombinant CtBP proteins (10 μM) in binding buffer (25 mM Tris-Cl, 100 mM NaCl, 1 mM EDTA, 5%...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-terminal-binding protein 1 [E295A](Homo sapiens (Human))
Oregon Health And Science University

LigandPNGBDBM213227(Nicotinamide adenine dinucleotide (NAD))
Affinity DataKd:  2.40E+3nMAssay Description:Equilibrium dialysis was performed using purified recombinant CtBP proteins (10 μM) in binding buffer (25 mM Tris-Cl, 100 mM NaCl, 1 mM EDTA, 5%...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-terminal-binding protein 1 [H315A](Homo sapiens (Human))
Oregon Health And Science University

LigandPNGBDBM213227(Nicotinamide adenine dinucleotide (NAD))
Affinity DataKd:  7.90E+3nMAssay Description:Equilibrium dialysis was performed using purified recombinant CtBP proteins (10 μM) in binding buffer (25 mM Tris-Cl, 100 mM NaCl, 1 mM EDTA, 5%...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-terminal-binding protein 1 [V66R](Homo sapiens (Human))
Oregon Health And Science University

LigandPNGBDBM213227(Nicotinamide adenine dinucleotide (NAD))
Affinity DataKd:  500nMAssay Description:Equilibrium dialysis was performed using purified recombinant CtBP proteins (10 μM) in binding buffer (25 mM Tris-Cl, 100 mM NaCl, 1 mM EDTA, 5%...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-terminal-binding protein 1 [W318F](Homo sapiens (Human))
Oregon Health And Science University

LigandPNGBDBM213227(Nicotinamide adenine dinucleotide (NAD))
Affinity DataKd:  2.20E+3nMAssay Description:Equilibrium dialysis was performed using purified recombinant CtBP proteins (10 μM) in binding buffer (25 mM Tris-Cl, 100 mM NaCl, 1 mM EDTA, 5%...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-terminal-binding protein 1(Homo sapiens (Human))
University Of Massachusetts Medical School

LigandPNGBDBM213227(Nicotinamide adenine dinucleotide (NAD))
Affinity DataKd:  390nMAssay Description:Equilibrium dialysis was performed using purified recombinant CtBP proteins (10 μM) in binding buffer (25 mM Tris-Cl, 100 mM NaCl, 1 mM EDTA, 5%...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-terminal-binding protein 1 [A52D](Homo sapiens (Human))
Oregon Health And Science University

LigandPNGBDBM213227(Nicotinamide adenine dinucleotide (NAD))
Affinity DataKd:  500nMAssay Description:Equilibrium dialysis was performed using purified recombinant CtBP proteins (10 μM) in binding buffer (25 mM Tris-Cl, 100 mM NaCl, 1 mM EDTA, 5%...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed