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Found 357 Enz. Inhib. hit(s) with Target = 'Falcipain 2'
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23141(3-[(diethylamino)methyl]-2,4-dihydroxybenzaldehyde...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23157(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-{...)
Affinity DataIC50:  630nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23143(2,4-dihydroxy-3-(piperidin-1-ylmethyl)benzaldehyde...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23144(2,4-dihydroxy-3-(morpholin-4-ylmethyl)benzaldehyde...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23145(2,4-dihydroxy-3-[(4-methylpiperazin-1-yl)methyl]be...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23146(3-{[4-(7-chloroquinolin-4-yl)piperazin-1-yl]methyl...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23147([(E)-({3-[(diethylamino)methyl]-2,4-dihydroxypheny...)
Affinity DataIC50:  1.11E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23148([(E)-{[2,4-dihydroxy-3-(pyrrolidin-1-ylmethyl)phen...)
Affinity DataIC50:  5.85E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23149([(E)-{[2,4-dihydroxy-3-(piperidin-1-ylmethyl)pheny...)
Affinity DataIC50:  3.80E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23150([(E)-{[2,4-dihydroxy-3-(morpholin-4-ylmethyl)pheny...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23151([(E)-({2,4-dihydroxy-3-[(4-methylpiperazin-1-yl)me...)
Affinity DataIC50:  1.82E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23152([(E)-[(3-{[4-(7-chloroquinolin-4-yl)piperazin-1-yl...)
Affinity DataIC50:  2.25E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23153([(E)-[(3-{[4-(7-chloroquinolin-4-yl)piperazin-1-yl...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23154(2,4-dihydroxybenzaldehyde thiosemicarbazone | [(E)...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23158(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-{...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23159(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-(...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23160(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-[...)
Affinity DataIC50:  3.16E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23155(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-(...)
Affinity DataIC50:  2.60E+3nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23156(1-{2-[(7-chloroquinolin-4-yl)amino]ethyl}-3-[(E)-{...)
Affinity DataIC50:  720nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM23142(2,4-dihydroxy-3-(pyrrolidin-1-ylmethyl)benzaldehyd...)
Affinity DataIC50: >2.00E+4nMpH: 5.5 T: 2°CAssay Description:IC50 values against the recombinant falcipain-2 were determined by incubating protein with different concentrations of inhibitors in reaction buffer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50322349((R)-Methyl4-(2-(3-((adamantan-1-ylcarbamoyloxy)met...)
Affinity DataKi:  14nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50257018((E)-methyl4-(2-((R,Z)-3-((4-chloro-2-(trifluoromet...)
Affinity DataKi:  17nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371561(CHEMBL405741)
Affinity DataKi:  53nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371567(CHEMBL270278)
Affinity DataKi:  110nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371562(CHEMBL271992)
Affinity DataKi:  120nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371568(CHEMBL408071)
Affinity DataKi:  140nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074428(CHEMBL3409895)
Affinity DataKi:  200nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataKi:  290nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataKi:  290nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074133(CHEMBL3409912)
Affinity DataKi:  300nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074132(CHEMBL3409913)
Affinity DataKi:  300nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371564(CHEMBL403991)
Affinity DataKi:  320nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371566(CHEMBL407354)
Affinity DataKi:  370nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371563(CHEMBL272015)
Affinity DataKi:  390nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074143(CHEMBL3409902)
Affinity DataKi:  400nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074144(CHEMBL3409901)
Affinity DataKi:  400nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50183767((2R,3R)-dibenzyl 1-((S)-1-((S)-2-(tert-butoxycarbo...)
Affinity DataKi:  400nMAssay Description:Inhibition of Plasmodium falciparum falcipain 2 using Z-Phe-Arg-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50468724(CHEMBL4294334)
Affinity DataKi:  450nMAssay Description:Inhibition of Plasmodium falciparum falcipain 2 using Z-Phe-Arg-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50322342((R)-Methyl4-(2-(7-chloro-3-((4-chloro-2-(trifluoro...)
Affinity DataKi:  460nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50371565(CHEMBL402455)
Affinity DataKi:  600nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074130(CHEMBL3409915)
Affinity DataKi:  600nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074145(CHEMBL3409900)
Affinity DataKi:  800nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074131(CHEMBL3409914)
Affinity DataKi:  800nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074138(CHEMBL3409907)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50468723(CHEMBL4279824)
Affinity DataKi:  1.26E+3nMAssay Description:Inhibition of Plasmodium falciparum falcipain 2 using Z-Phe-Arg-AMC as substrate by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074137(CHEMBL3409908)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50322343((R)-Methyl4-(2-(5-(4-bromophenyl)-3-((4-chloro-2-(...)
Affinity DataKi:  1.56E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074434(CHEMBL3409894)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50322341(CHEMBL1171803 | Methyl4-(2-((R)-3-((4-chloro-2-(tr...)
Affinity DataKi:  2.22E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 after 10 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
University Of Cape Town

LigandPNGBDBM50074142(CHEMBL3409903)
Affinity DataKi:  2.53E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2 using ZFR-AMC as substrate after 30 mins by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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