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Found 2642 Enz. Inhib. hit(s) with Target = 'L-lactate dehydrogenase A'
TargetL-lactate dehydrogenase A chain(Mus musculus (Mouse))
Instituto Politécnico Nacional

LigandPNGBDBM23222(Oxalamic acid | Oxamate | Oxamate, 3 | Oxamidic Ac...)
Affinity DataIC50:  8.00E+4nMpH: 7.4Assay Description:Lactate dehydrogenase activity was determined by recording the absorbance change at 340 nm produced by the oxidation of NADH. Assays were performed a...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86138(LDHA Inhibitor, 34)
Affinity DataKd:  8nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Mus musculus (Mouse))
Instituto Politécnico Nacional

LigandPNGBDBM234444(N-Propyl oxamate)
Affinity DataIC50:  1.75E+6nMpH: 7.4Assay Description:Lactate dehydrogenase activity was determined by recording the absorbance change at 340 nm produced by the oxidation of NADH. Assays were performed a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Mus musculus (Mouse))
Instituto Politécnico Nacional

LigandPNGBDBM234445(N-Butyl oxamate)
Affinity DataIC50:  9.10E+6nMpH: 7.4Assay Description:Lactate dehydrogenase activity was determined by recording the absorbance change at 340 nm produced by the oxidation of NADH. Assays were performed a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Mus musculus (Mouse))
Instituto Politécnico Nacional

LigandPNGBDBM234446(N-Isobutyl oxamate)
Affinity DataIC50:  6.00E+6nMpH: 7.4Assay Description:Lactate dehydrogenase activity was determined by recording the absorbance change at 340 nm produced by the oxidation of NADH. Assays were performed a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Mus musculus (Mouse))
Instituto Politécnico Nacional

LigandPNGBDBM234447(N-sec-Butyl oxamate)
Affinity DataIC50:  1.25E+7nMpH: 7.4Assay Description:Lactate dehydrogenase activity was determined by recording the absorbance change at 340 nm produced by the oxidation of NADH. Assays were performed a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM86114(LDHA Inhibitor, 8)
Affinity DataKd:  1.28E+4nMpH: 7.4 T: 2°CAssay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86115(LDHA Inhibitor, 9)
Affinity DataKd:  1.60E+6nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86116(LDHA Inhibitor, 11)
Affinity DataKd:  3.00E+6nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86117(LDHA Inhibitor, 12)
Affinity DataKd:  7.70E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86124(LDHA Inhibitor, 20)
Affinity DataKd:  2.10E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86125(LDHA Inhibitor, 21)
Affinity DataKd:  2.80E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86126(LDHA Inhibitor, 22)
Affinity DataKd:  7.70E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86127(LDHA Inhibitor, 23)
Affinity DataKd:  3.50E+4nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86128(LDHA Inhibitor, 24)
Affinity DataKd:  1.60E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86129(LDHA Inhibitor, 25)
Affinity DataKd:  1.10E+6nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86130(LDHA Inhibitor, 26)
Affinity DataKd:  130nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86131(LDHA Inhibitor, 27)
Affinity DataKd:  46nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86132(LDHA Inhibitor, 28)
Affinity DataKd:  3.20E+3nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86133(LDHA Inhibitor, 29)
Affinity DataKd:  69nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86134(LDHA Inhibitor, 30)
Affinity DataKd:  1.20E+3nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86135(LDHA Inhibitor, 31)
Affinity DataKd:  60nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86136(LDHA Inhibitor, 32)
Affinity DataKd:  180nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86137(LDHA Inhibitor, 33)
Affinity DataKd:  93nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Mus musculus (Mouse))
Instituto Politécnico Nacional

LigandPNGBDBM234443(N-Ethyl oxamate)
Affinity DataIC50:  1.40E+5nMpH: 7.4Assay Description:Lactate dehydrogenase activity was determined by recording the absorbance change at 340 nm produced by the oxidation of NADH. Assays were performed a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86132(LDHA Inhibitor, 28)
Affinity DataIC50:  8.62E+4nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86133(LDHA Inhibitor, 29)
Affinity DataIC50:  1.90E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86134(LDHA Inhibitor, 30)
Affinity DataIC50:  2.95E+4nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86135(LDHA Inhibitor, 31)
Affinity DataIC50:  290nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86136(LDHA Inhibitor, 32)
Affinity DataIC50:  7.40E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86137(LDHA Inhibitor, 33)
Affinity DataIC50:  500nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86138(LDHA Inhibitor, 34)
Affinity DataIC50:  270nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM23251(1,2,5-Thiadiazole, TDA1 | 4-hydroxy-1,2,5-thiadiaz...)
Affinity DataIC50:  4.50E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50066974(7-Benzyl-2,3-dihydroxy-6-methyl-4-propyl-naphthale...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50339607(1-Hydroxy-6-phenyl-4-trifluoromethyl-1H-indole-2-c...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50219487(1-hydroxy-2-naphthoate | 1-hydroxy-2-naphthoic aci...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50192453(AMP(2-) | Adenosine-5-monophosphate | LDHA Inhibit...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM86113(LDHA Inhibitor, 7)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM86114(LDHA Inhibitor, 8)
Affinity DataIC50:  1.32E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50339607(1-Hydroxy-6-phenyl-4-trifluoromethyl-1H-indole-2-c...)
Affinity DataKd:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50219487(1-hydroxy-2-naphthoate | 1-hydroxy-2-naphthoic aci...)
Affinity DataKd:  6.40E+5nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50192453(AMP(2-) | Adenosine-5-monophosphate | LDHA Inhibit...)
Affinity DataKd:  6.50E+5nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM86113(LDHA Inhibitor, 7)
Affinity DataKd:  4.00E+6nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86115(LDHA Inhibitor, 9)
Affinity DataKd:  3.00E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM50078827(2-(pyridin-3-yl)-1H-benzo[d]imidazole | 2-Pyridin-...)
Affinity DataKd:  1.40E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86116(LDHA Inhibitor, 11)
Affinity DataKd:  2.40E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86117(LDHA Inhibitor, 12)
Affinity DataKd:  1.00E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86118(LDHA Inhibitor, 13)
Affinity DataKd:  4.00E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86119(LDHA Inhibitor, 14)
Affinity DataKd:  4.20E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86115(LDHA Inhibitor, 9)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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